The following articles (labelled with PubMed ID or TBD) are for your review
| PMID | Data | Article Title | Organization |
|---|
| 1310115 |
11 |
Synthesis, antinociceptive activity, and opioid receptor profiles of substituted trans-3-(decahydro- and octahydro-4a-isoquinolinyl)phenols. |
Glaxo Group Research |
| 2475628 |
5 |
Opioid agonist and antagonist activities of peripherally selective derivatives of naltrexamine and oxymorphamine. |
University of Minnesota |
| 2872334 |
16 |
Synthesis and opioid activity of dermorphin tetrapeptides bearing D-methionine S-oxide at position 2. |
TBA |
| 3020245 |
4 |
Synthesis and biological activity of analogues of beta-chlornaltrexamine and beta-funaltrexamine at opioid receptors. |
TBA |
| 6312042 |
7 |
Different receptor sites mediate opioid agonism and antagonism. |
TBA |
| 6283082 |
3 |
Stereochemical studies on medicinal agents. 25. Absolute configuration and analgetic potency of beta-1,2-dimethyl-2-phenyl-4-(propionyloxy)piperidine enantiomers. |
TBA |
| 6106064 |
20 |
Synthesis and biological activity of fluoroalkylamine derivatives of narcotic analgesics. |
TBA |
| 1361580 |
25 |
N-terminal alkylated derivatives of [D-Pro10]dynorphin A-(1-11) are highly selective for kappa-opioid receptors. |
Oregon State University |
| 1335078 |
76 |
O3-(2-carbomethoxyallyl) ethers of opioid ligands derived from oxymorphone, naltrexone, etorphine, diprenorphine, norbinaltorphimine, and naltrindole. Unexpected O3-dealkylation in the opioid radioligand displacement assay. |
University of Washington |
| 1320121 |
48 |
Electrophilic opioid ligands. Oxygen tethered alpha-methylene-gamma-lactone, acrylate, isothiocyanate, and epoxide derivatives of 6 beta-naltrexol. |
University of Washington |
| 2153826 |
11 |
Conjugate addition ligands of opioid antagonists. Methacrylate esters and ethers of 6 alpha- and 6 beta-naltrexol. |
University of Washington |
| 9873602 |
11 |
A high affinity, mu-opioid receptor-selective enkephalin analogue lacking an N-terminal tyrosine. |
University of Michigan |
| 16722631 |
87 |
An integrated in silico 3D model-driven discovery of a novel, potent, and selective amidosulfonamide 5-HT1A agonist (PRX-00023) for the treatment of anxiety and depression. |
Predix Pharmaceuticals |
| 197237 |
3 |
3-Hydroxy-17-aralkylmorphinans as potential opiate receptor-site-directed alkylating agents. |
TBA |
| 894682 |
12 |
Stereochemical studies on medicinal agents. 23. Synthesis and biological evaluation of 6-amino derivatives of naloxone and naltrexone. |
TBA |
| 513062 |
2 |
4-(p-Bromophenyl)-4-(dimethylamino)-1-phenethylcyclohexanol, an extremely potent respresentative of a new analgesic series. |
TBA |
| 1972964 |
40 |
Design and synthesis of highly potent and selective cyclic dynorphin A analogues. |
University of Arizona |
| 1652019 |
12 |
Electrophilic gamma-lactone kappa-opioid receptor probes. Analogues of 2'-hydroxy-2-tetrahydrofurfuryl-5,9-dimethyl-6,7-benzomorphan diastereomers. |
University of Washington |
Search and Browse
