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32 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review
PMIDDataArticle TitleOrganization
27326332 66 Discovery and Preclinical Evaluation of BMS-711939, an Oxybenzylglycine Based PPARa Selective Agonist.EBI Bristol-Myers Squibb
26990539 79 Discovery of a Novel, Orally Efficacious Liver X Receptor (LXR)ß Agonist.EBI Vitae Pharmaceuticals
 61 Synthesis and structure-activity relationships of potent conformationally restricted retinoid X receptor ligandsEBI TBA
 22 Synthesis and receptor binding affinity of conformationally restricted retinoic acid analoguesEBI TBA
 83 Synthesis of highly potent RXR-specific retinoids: The use of a cyclopropyl group as a double bond isostereEBI TBA
 54 Differential RXR & RAR activity of stilbene retinoid analogs bearing thiazole and imidazole carboxylic acidsEBI TBA
19095448 24 Replacing alkyl sulfonamide with aromatic sulfonamide in sulfonamide-type RXR agonists favors switch towards antagonist activity.EBI Okayama University Graduate School of Medicine
16364638 99 Aza-retinoids as novel retinoid X receptor-specific agonists.EBI Ligand Pharmaceuticals
15006411 126 Design, synthesis and structure-activity relationship of novel RXR-selective modulators.EBI Ligand Pharmaceuticals
14592510 150 Design and synthesis of novel RXR-selective modulators with improved pharmacological profile.EBI Ligand Pharmaceuticals
12482435 75 Retinoic acid receptor ligands based on the 6-cyclopropyl-2,4-hexadienoic acid.EBI Ligand Pharmaceuticals
12161154 11 An improved synthesis of the C-linked glucuronide of N-(4-hydroxyphenyl)retinamide.EBI The Ohio State University
11428923 39 Enantioselective syntheses of potent retinoid X receptor ligands: differential biological activities of individual antipodes.EBI Allergan
30776227 38 Discovery of Second Generation ROR? Inhibitors Composed of an Azole Scaffold.EBI Kyoto Prefectural University of Medicine
27592633 13 Modeling, Synthesis, and Biological Evaluation of Potential Retinoid X Receptor (RXR)-Selective Agonists: Analogues of 4-[1-(3,5,5,8,8-Pentamethyl-5,6,7,8-tetrahydro-2-naphthyl)ethynyl]benzoic Acid (Bexarotene) and 6-(Ethyl(5,5,8,8-tetrahydronaphthalen-2-yl)amino)nicotinic Acid (NEt-TMN).EBI Arizona State University
30702885 256 Tuning Nuclear Receptor Selectivity of Wy14,643 towards Selective Retinoid X Receptor Modulation.EBI Goethe University Frankfurt
10585206 45 Structure-activity relationship studies of novel heteroretinoids: induction of apoptosis in the HL-60 cell line by a novel isoxazole-containing heteroretinoid.EBI Università
10098670 24 Stereoselective synthesis and receptor activity of conformationally defined retinoid X receptor selective ligands.EBI Allergan
10052980 138 Synthesis of retinoid X receptor-specific ligands that are potent inducers of adipogenesis in 3T3-L1 cells.EBI Ligand Pharmaceuticals
30783504 87 Computer-Assisted Discovery and Structural Optimization of a Novel Retinoid X Receptor Agonist Chemotype.EBI Goethe-University Frankfurt
9435893 46 Regulation of retinoidal actions by diazepinylbenzoic acids. Retinoid synergists which activate the RXR-RAR heterodimers.EBI University of Tokyo
30594433 90 Discovery of potent and selective PPAR?/? dual antagonists and initial biological studies.EBI Inception Sciences
8784454 76 Synthesis and structure-activity relationships of retinoid X receptor selective diaryl sulfide analogs of retinoic acid.EBI Allergan
31531208 46 A Novel Biphenyl-based Chemotype of Retinoid X Receptor Ligands Enables Subtype and Heterodimer Preferences.EBI Goethe-University Frankfurt
8765503 39 Identification of the first retinoid X, receptor homodimer antagonist.EBI Ligand Pharmaceuticals
8709094 41 Discovery of novel retinoic acid receptor agonists having potent antiproliferative activity in cervical cancer cells.EBI Ligand Pharmaceuticals
8308867 72 Synthesis of high specific activity [3H]-9-cis-retinoic acid and its application for identifying retinoids with unusual binding properties.EBI Ligand Pharmaceuticals
23217961 2 Structure-activity relationship study on benzoic acid part of diphenylamine-based retinoids.EBI Tohoku Pharmaceutical University
7650690 64 Conformational effects on retinoid receptor selectivity. 2. Effects of retinoid bridging group on retinoid X receptor activity and selectivity.EBI Sri International
29901398 29 Computer-Assisted Discovery of Retinoid X Receptor Modulating Natural Products and Isofunctional Mimetics.EBI Swiss Federal Institute of Technology (Eth)
28850227 85 Natural-Products-Inspired Use of the gem-Dimethyl Group in Medicinal Chemistry.EBI St. John'S University