The following articles (labelled with PubMed ID or TBD) are for your review
PMID | Data | Article Title | Organization |
17267215 |
27 |
Oxazolidinones as novel human CCR8 antagonists. |
Glaxosmithkline |
19954248 |
85 |
Increasing selectivity of CC chemokine receptor 8 antagonists by engineering nondesolvation related interactions with the intended and off-target binding sites. |
Astrazeneca |
18257512 |
33 |
Overcoming undesirable HERG potency of chemokine receptor antagonists using baseline lipophilicity relationships. |
Astrazeneca |
22957890 |
174 |
Modulation in selectivity and allosteric properties of small-molecule ligands for CC-chemokine receptors. |
University of Copenhagen |
17266208 |
104 |
Design, synthesis, and evaluation of naphthalene-sulfonamide antagonists of human CCR8. |
Millennium Pharmaceuticals |
16698264 |
37 |
Discovery of 3,5-bis(trifluoromethyl)benzyl L-arylglycinamide based potent CCR2 antagonists. |
Merck Research Laboratories |
16640325 |
41 |
Design, synthesis, and progress toward optimization of potent small molecule antagonists of CC chemokine receptor 8 (CCR8). |
Millennium Pharmaceuticals |
31913038 |
13 |
Preventing Morphine-Seeking Behavior through the Re-Engineering of Vincamine's Biological Activity. |
University of Florida |
23409871 |
48 |
Synthesis and structure-activity relationships of indazole arylsulfonamides as allosteric CC-chemokine receptor 4 (CCR4) antagonists. |
Glaxosmithkline |
29406702 |
128 |
Discovery of Novel 1-Cyclopentenyl-3-phenylureas as Selective, Brain Penetrant, and Orally Bioavailable CXCR2 Antagonists. |
Gsk Pharmaceuticals R & D |