The following articles (labelled with PubMed ID or TBD) are for your review
PMID | Data | Article Title | Organization |
10386934 |
15 |
Dual-acting agents with alpha1-adrenoceptor antagonistic and steroid 5alpha-reductase inhibitory activities. Synthesis and evaluation of arylpiperazine derivatives. |
Zeria Pharmaceutical |
9873656 |
17 |
Synthesis of benzanilide derivatives as dual acting agents with alpha 1-adrenoceptor antagonistic action and steroid 5-alpha reductase inhibitory activity. |
Zeria Pharmaceutical |
9873464 |
6 |
A practical synthesis of 3-substituted delta 3,5(6)-steroids as new potential 5 alpha-reductase inhibitor. |
Chinese Academy of Science |
26631442 |
6 |
Synthesis and activity of novel 16-dehydropregnenolone acetate derivatives as inhibitors of type 1 5a-reductase and on cancer cell line SK-LU-1. |
Universidad Nacional Aut£Noma De M£Xico |
25261928 |
17 |
Effect of dehydroepiandrosterone derivatives on the activity of 5a-reductase isoenzymes and on cancer cell line PC-3. |
National University of Mexico |
24951332 |
3 |
Conformational analysis of an anti-androgenic, (E,E)-8-hydroxygermacrene B, using NOESY and dynamic NMR spectroscopy. |
Naresuan University |
2308144 |
16 |
Steroidal A ring aryl carboxylic acids: a new class of steroid 5 alpha-reductase inhibitors. |
Smith Kline & French Laboratories |
12139451 |
41 |
Synthesis and evaluation of 2'-substituted 4-(4'-carboxy- or 4'-carboxymethylbenzylidene)-N-acylpiperidines: highly potent and in vivo active steroid 5alpha-reductase type 2 inhibitors. |
Saarland University |
9135028 |
114 |
Pharmacological options in the treatment of benign prostatic hyperplasia. |
Pfizer |
8978835 |
18 |
Indole derivatives as a new class of steroid 5 alpha-reductase inhibitors. |
Kyowa Hakko Kogyo |
7629802 |
48 |
Structure-activity relationships for inhibition of type 1 and 2 human 5 alpha-reductase and human adrenal 3 beta-hydroxy-delta 5-steroid dehydrogenase/3-keto-delta 5-steroid isomerase by 6-azaandrost-4-en-3-ones: optimization of the C17 substituent. |
Glaxo Inc. Research Institute |
3783591 |
225 |
Azasteroids: structure-activity relationships for inhibition of 5 alpha-reductase and of androgen receptor binding. |
TBA |
9871588 |
5 |
Structure activity relationship study of known inhibitors of the enzyme 5 alpha-reductase (5AR). |
Kingston University |
| 3 |
The preparation and evaluation of (+/-)-trans-1-Diazo-8-methoxy-4a-methyl-1,2,3,4,4a,9,10,10a-octahydro-phenanthren-2-one as an inhibitor of human type-1 steroid 5α-reductase |
TBA |
| 2 |
Synthesis of a chemiluminescent probe useful for the purification of steroid 5α-reductase |
TBA |
16420060 |
12 |
Novel 5alpha-reductase inhibitors: synthesis, structure-activity studies, and pharmacokinetic profile of phenoxybenzoylphenyl acetic acids. |
Saarland University |
10386944 |
7 |
N-substituted 4-(5-indolyl)benzoic acids. Synthesis and evaluation of steroid 5alpha-reductase type I and II inhibitory activity. |
UniversitäT Des Saarlandes |
29400967 |
136 |
Fluorine and Fluorinated Motifs in the Design and Application of Bioisosteres for Drug Design. |
Bristol-Myers Squibb |
9871560 |
17 |
Synthesis and 5 alpha-reductase inhibitory activities of benzofuran derivatives with a carbamoyl group. |
Sankyo |
11689062 |
8 |
Novel lead generation through hypothetical pharmacophore three-dimensional database searching: discovery of isoflavonoids as nonsteroidal inhibitors of rat 5 alpha-reductase. |
TBA |
7636849 |
52 |
(E)-4-(2-[[3-(indol-5-yl)-1-oxo-2-butenyl]amino]phenoxy)butyric acid derivatives: a new class of steroid 5 alpha-reductase inhibitors in the rat prostate. 1. |
Kyowa Hakko Kogyo |
30007568 |
3 |
Activity of steroid 4 and derivatives 4a-4f as inhibitors of the enzyme 5?-reductase 1. |
Universidad Nacional Aut£Noma De M£Xico |
2391687 |
16 |
Hydroxyperfluoroazobenzenes: novel inhibitors of enzymes of androgen biosynthesis. |
Institute of Cancer Research |
2308145 |
48 |
Inhibition of steroid 5 alpha-reductase by unsaturated 3-carboxysteroids. |
Smith Kline & French Laboratories |