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24 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review
PMIDDataArticle TitleOrganization
10386934 15 Dual-acting agents with alpha1-adrenoceptor antagonistic and steroid 5alpha-reductase inhibitory activities. Synthesis and evaluation of arylpiperazine derivatives.EBI Zeria Pharmaceutical
9873656 17 Synthesis of benzanilide derivatives as dual acting agents with alpha 1-adrenoceptor antagonistic action and steroid 5-alpha reductase inhibitory activity.EBI Zeria Pharmaceutical
9873464 6 A practical synthesis of 3-substituted delta 3,5(6)-steroids as new potential 5 alpha-reductase inhibitor.EBI Chinese Academy of Science
26631442 6 Synthesis and activity of novel 16-dehydropregnenolone acetate derivatives as inhibitors of type 1 5a-reductase and on cancer cell line SK-LU-1.EBI Universidad Nacional Aut£Noma De M£Xico
25261928 17 Effect of dehydroepiandrosterone derivatives on the activity of 5a-reductase isoenzymes and on cancer cell line PC-3.EBI National University of Mexico
24951332 3 Conformational analysis of an anti-androgenic, (E,E)-8-hydroxygermacrene B, using NOESY and dynamic NMR spectroscopy.EBI Naresuan University
2308144 16 Steroidal A ring aryl carboxylic acids: a new class of steroid 5 alpha-reductase inhibitors.EBI Smith Kline & French Laboratories
12139451 41 Synthesis and evaluation of 2'-substituted 4-(4'-carboxy- or 4'-carboxymethylbenzylidene)-N-acylpiperidines: highly potent and in vivo active steroid 5alpha-reductase type 2 inhibitors.EBI Saarland University
9135028 114 Pharmacological options in the treatment of benign prostatic hyperplasia.EBI Pfizer
8978835 18 Indole derivatives as a new class of steroid 5 alpha-reductase inhibitors.EBI Kyowa Hakko Kogyo
7629802 48 Structure-activity relationships for inhibition of type 1 and 2 human 5 alpha-reductase and human adrenal 3 beta-hydroxy-delta 5-steroid dehydrogenase/3-keto-delta 5-steroid isomerase by 6-azaandrost-4-en-3-ones: optimization of the C17 substituent.EBI Glaxo Inc. Research Institute
3783591 225 Azasteroids: structure-activity relationships for inhibition of 5 alpha-reductase and of androgen receptor binding.EBI TBA
9871588 5 Structure activity relationship study of known inhibitors of the enzyme 5 alpha-reductase (5AR).EBI Kingston University
 3 The preparation and evaluation of (+/-)-trans-1-Diazo-8-methoxy-4a-methyl-1,2,3,4,4a,9,10,10a-octahydro-phenanthren-2-one as an inhibitor of human type-1 steroid 5α-reductaseEBI TBA
 2 Synthesis of a chemiluminescent probe useful for the purification of steroid 5α-reductaseEBI TBA
16420060 12 Novel 5alpha-reductase inhibitors: synthesis, structure-activity studies, and pharmacokinetic profile of phenoxybenzoylphenyl acetic acids.EBI Saarland University
10386944 7 N-substituted 4-(5-indolyl)benzoic acids. Synthesis and evaluation of steroid 5alpha-reductase type I and II inhibitory activity.EBI UniversitäT Des Saarlandes
29400967 136 Fluorine and Fluorinated Motifs in the Design and Application of Bioisosteres for Drug Design.EBI Bristol-Myers Squibb
9871560 17 Synthesis and 5 alpha-reductase inhibitory activities of benzofuran derivatives with a carbamoyl group.EBI Sankyo
11689062 8 Novel lead generation through hypothetical pharmacophore three-dimensional database searching: discovery of isoflavonoids as nonsteroidal inhibitors of rat 5 alpha-reductase.EBI TBA
7636849 52 (E)-4-(2-[[3-(indol-5-yl)-1-oxo-2-butenyl]amino]phenoxy)butyric acid derivatives: a new class of steroid 5 alpha-reductase inhibitors in the rat prostate. 1.EBI Kyowa Hakko Kogyo
30007568 3 Activity of steroid 4 and derivatives 4a-4f as inhibitors of the enzyme 5?-reductase 1.EBI Universidad Nacional Aut£Noma De M£Xico
2391687 16 Hydroxyperfluoroazobenzenes: novel inhibitors of enzymes of androgen biosynthesis.EBI Institute of Cancer Research
2308145 48 Inhibition of steroid 5 alpha-reductase by unsaturated 3-carboxysteroids.EBI Smith Kline & French Laboratories