The following articles (labelled with PubMed ID or TBD) are for your review
PMID | Data | Article Title | Organization |
22475558 |
82 |
Discovery of an orally-bioavailable CC Chemokine Receptor 2 antagonist derived from an acyclic diaminoalcohol backbone. |
Bristol-Myers Squibb |
16198561 |
99 |
Novel CCR1 antagonists with oral activity in the mouse collagen induced arthritis. |
Novartis Institutes For Biomedical Research |
21295478 |
81 |
Discovery of INCB10820/PF-4178903, a potent, selective, and orally bioavailable dual CCR2 and CCR5 antagonist. |
Incyte |
21036044 |
43 |
Discovery of INCB3344, a potent, selective and orally bioavailable antagonist of human and murine CCR2. |
Incyte |
17389363 |
2 |
Naloxone acts as a potent analgesic in transgenic mouse models of sickle cell anemia. |
University of Minnesota |
12086500 |
59 |
Synthesis, SAR, and biological evaluation of oximino-piperidino-piperidine amides. 1. Orally bioavailable CCR5 receptor antagonists with potent anti-HIV activity. |
Schering-Plough Research Institute |
29425816 |
6 |
Recent updates for designing CCR5 antagonists as anti-retroviral agents. |
Nirma University |