The following articles (labelled with PubMed ID or TBD) are for your review
PMID | Data | Article Title | Organization |
16610792 |
15 |
Refinement of the benzodiazepine receptor site topology by structure-activity relationships of new N-(heteroarylmethyl)indol-3-ylglyoxylamides. |
Universit£ |
7799410 |
46 |
Four amino acid exchanges convert a diazepam-insensitive, inverse agonist-preferring GABAA receptor into a diazepam-preferring GABAA receptor. |
Heidelberg |
17335185 |
21 |
Novel N-substituted indol-3-ylglyoxylamides probing the LDi and L1/L2 lipophilic regions of the benzodiazepine receptor site in search for subtype-selective ligands. |
Università |
17306981 |
8 |
Novel 3-iodo-8-ethoxypyrazolo[5,1-c][1,2,4]benzotriazine 5-oxide as promising lead for design of alpha5-inverse agonist useful tools for therapy of mnemonic damage. |
Università |
15828832 |
14 |
High affinity central benzodiazepine receptor ligands: synthesis and biological evaluation of a series of phenyltriazolobenzotriazindione derivatives. |
Università |
12519068 |
32 |
Synthesis and benzodiazepine receptor affinity of pyrazolo[1,5-a]pyrimidine derivatives. 3. New 6-(3-thienyl) series as alpha 1 selective ligands. |
University of Firenze |
12477354 |
8 |
Benzodiazepine receptor ligands. 7. Synthesis and pharmacological evaluation of new 3-esters of the 8-chloropyrazolo[5,1-c][1,2,4]benzotriazine 5-oxide. 3-(2-Thienylmethoxycarbonyl) derivative: an anxioselective agent in rodents. |
Università |
11428922 |
21 |
Novel N-(arylalkyl)indol-3-ylglyoxylylamides targeted as ligands of the benzodiazepine receptor: synthesis, biological evaluation, and molecular modeling analysis of the structure-activity relationships. |
Università |
20684859 |
12 |
Homology modeling and atomic level binding study of GABA(A) receptor with novel enaminone amides. |
Wuhan Institute of Technology |
29657102 |
19 |
Agonists of the ?-aminobutyric acid type B (GABA |
University of Mississippi |
29650463 |
17 |
A new class of pyrazolo[5,1-c][1,2,4]triazines as ?-aminobutyric type A (GABA |
Universit£ |
29146472 |
71 |
Discovery of the first low-shift positive allosteric modulators for the muscarinic M1 receptor. |
Roche Pharma Research and Early Development |