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16 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review
PMIDDataArticle TitleOrganization
10464022 25 Design and in vivo analysis of potent non-thiol inhibitors of farnesyl protein transferase.EBI Merck Research Laboratories
9651171 29 N-Arylalkyl pseudopeptide inhibitors of farnesyltransferase.EBI Merck Research Laboratories
8145221 28 Pseudopeptide inhibitors of Ras farnesyl-protein transferase.EBI Merck Research Laboratories
10450988 51 Synthesis and evaluation of hydroxyproline-derived isoprenyltransferase inhibitors.EBI Eisai Research Institute
 21 DIARYLETHER INHIBITORS OF FARNESYL-PROTEIN TRANSFERASEEBI TBA
15582430 123 Design and synthesis of o-trifluoromethylbiphenyl substituted 2-amino-nicotinonitriles as inhibitors of farnesyltransferase.EBI Abbott Laboratories
15454229 86 Synthesis and activity of 1-aryl-1'-imidazolyl methyl ethers as non-thiol farnesyltransferase inhibitors.EBI Abbott Laboratories
15454228 17 Design, synthesis, and activity of 4-quinolone and pyridone compounds as nonthiol-containing farnesyltransferase inhibitors.EBI Abbott Laboratories
15324873 21 Synthesis of 1H-pyridin-2-one derivatives as potent and selective farnesyltransferase inhibitors.EBI Abbott Laboratories
12699757 72 Discovery of potent imidazole and cyanophenyl containing farnesyltransferase inhibitors with improved oral bioavailability.EBI Abbott Laboratories
12657284 31 Novel and selective imidazole-containing biphenyl inhibitors of protein farnesyltransferase.EBI Abbott Laboratories
8691462 14 2-substituted piperazines as constrained amino acids. Application to the synthesis of potent, non carboxylic acid inhibitors of farnesyltransferase.EBI Merck Research Laboratories
7562930 34 Pseudodipeptide inhibitors of protein farnesyltransferase.EBI Merck Research Laboratories
12657282 13 Aryl tetrahydropyridine inhibitors of farnesyltransferase: glycine, phenylalanine and histidine derivatives.BDB Abbott Laboratories
15808463 35 Design, synthesis, and activity of achiral analogs of 2-quinolones and indoles as non-thiol farnesyltransferase inhibitors.BDB Abbott Laboratories
15911281 30 Benzimidazolones and indoles as non-thiol farnesyltransferase inhibitors based on tipifarnib scaffold: synthesis and activity.BDB Abbott Laboratories