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18 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review
PMIDDataArticle TitleOrganization
11055335 27 Highly potent and selective peptide-based inhibitors of the hepatitis C virus serine protease: towards smaller inhibitors.EBI Boehringer Ingelheim Pharmaceuticals
10360758 10 Metallopeptide approach to the design of biologically active ligands: design of specific human neutrophil elastase inhibitors.EBI Palatin Technologies
 45 A comparative SAR and computer modeling study of benzisothiazolone, mechanism-based inhibitors with porcine pancreatic and human leukocyte elastaseEBI TBA
 27 Synthesis and porcine pancreatic elastase inhibitory evaluation of 6α-(sulfonyl)oxy-and 6α-chloropenicillanate sulfone esters and 3α-(acyloxy)methyl-6α-chloropenam sulfonesEBI TBA
 30 Enantioselective synthesis and antielastase activity of 1,3,4-trisubstituted and 3,4-disubstituted β-lactam antibioticsEBI TBA
12565935 5 Synthesis and evaluation of delta-lactams (piperazones) as elastase inhibitors.EBI The Oxford Centre For Molecular Sciences and The Dyson Perrins Laboratory
10866385 13 Mass spectrometry reveals elastase inhibitors from the reactive centre loop of alpha1-antitrypsin.EBI The Oxford Centre For Molecular Sciences
10698435 150 Structure-activity relationship studies of chloromethyl ketone derivatives for selective human chymase inhibitors.EBI Kyoto Pharmaceutical University
10091694 90 Symmetrical anhydride-type serine protease inhibitors: structure-activity relationship studies of human chymase inhibitors.EBI Nippon Steel
9925737 57 N-[2,2-dimethyl-3-(N-(4-cyanobenzoyl)amino)nonanoyl]-L-phenylalanine ethyl ester as a stable ester-type inhibitor of chymotrypsin-like serine proteases: structural requirements for potent inhibition of alpha-chymotrypsin.EBI Nippon Steel
9871780 85 Inhibition of human cytomegalovirus protease N(o) with monocyclic beta-lactams.EBI Boehringer Ingelheim (Canada)
9406601 109 Peptidomimetic inhibitors of the human cytomegalovirus protease.EBI Boehringer Ingelheim
9379436 46 Orally active trifluoromethyl ketone inhibitors of human leukocyte elastase.EBI Zeneca Pharmaceuticals
9341917 69 7-alkylidenecephalosporin esters as inhibitors of human leukocyte elastase.EBI Southern Methodist University
9191969 31 Dual inhibition of human leukocyte elastase and lipid peroxidation: in vitro and in vivo activities of azabicyclo[2.2.2]octane and perhydroindole derivatives.EBI Institut De Recherche Servier
7932558 30 Nonpeptidic inhibitors of human leukocyte elastase. 2. Design, synthesis, and in vitro activity of a series of 3-amino-6-arylopyridin-2-one trifluoromethyl ketones.EBI Zeneca Pharmaceuticals Group
7739010 118 Characterization of a class of peptide boronates with neutral P1 side chains as highly selective inhibitors of thrombin.EBI Thrombosis Research Institute
7562931 41 Peptidyl alpha-ketoheterocyclic inhibitors of human neutrophil elastase. 3. In vitro and in vivo potency of a series of peptidyl alpha-ketobenzoxazoles.EBI Zeneca Pharmaceuticals