The following articles (labelled with PubMed ID or TBD) are for your review
PMID | Data | Article Title | Organization |
26191358 |
105 |
Optimization of Novel Antagonists to the Neurokinin-3 Receptor for the Treatment of Sex-Hormone Disorders (Part II). |
Euroscreen |
25738882 |
210 |
Discovery and optimization of novel antagonists to the human neurokinin-3 receptor for the treatment of sex-hormone disorders (Part I). |
Euroscreen |
25247671 |
30 |
Development of novel neurokinin 3 receptor (NK3R) selective agonists with resistance to proteolytic degradation. |
Kyoto University |
7678430 |
23 |
Cyclic peptides as selective tachykinin antagonists. |
Merck Sharp and Dohme Research Laboratories |
16950620 |
36 |
N',2-diphenylquinoline-4-carbohydrazide based NK3 receptor antagonists. |
Merck Sharp & Dohme Research Laboratories |
8648606 |
72 |
Use of a dipeptide chemical library in the development of non-peptide tachykinin NK3 receptor selective antagonists. |
Cambridge University Forvie Site |
7515443 |
79 |
Design and synthesis of side-chain conformationally restricted phenylalanines and their use for structure-activity studies on tachykinin NK-1 receptor. |
Universit£ |
1331460 |
54 |
Conformationally constrained tachykinin analogues: potent and highly selective neurokinin NK-2 receptor agonists. |
Glaxo Group Research |
1851847 |
22 |
Imidazo[4,5-b]quinoxaline cyanines as neurokinin antagonists. |
Rochester |
21376585 |
120 |
Discovery of 3-aryl-5-acylpiperazinyl-pyrazoles as antagonists to the NK3 receptor. |
Euroscreen |
| 10 |
The dipeptide neurokinin-1 receptor antagonist S19752 is a potent and long-acting inhibitor of bronchoconstriction when administered by aerosol to the guinea pig in vivo |
TBA |
8759639 |
33 |
Synthesis and biological activity of NK-1 selective, N-backbone cyclic analogs of the C-terminal hexapeptide of substance P. |
Hebrew University of Jerusalem |
8576917 |
79 |
3-Aryl-1,2-diacetamidopropane derivatives as novel and potent NK-1 receptor antagonists. |
Eli Lilly |