The following articles (labelled with PubMed ID or TBD) are for your review
PMID | Data | Article Title | Organization |
25101488 |
50 |
Discovery of the CCR1 antagonist, BMS-817399, for the treatment of rheumatoid arthritis. |
Bristol-Myers Squibb |
23374868 |
76 |
1-(4-Phenylpiperazin-1-yl)-2-(1H-pyrazol-1-yl)ethanones as novel CCR1 antagonists. |
Chemocentryx |
23075267 |
85 |
Discovery and lead optimization of a novel series of CC chemokine receptor 1 (CCR1)-selective piperidine antagonists via parallel synthesis. |
Bristol-Myers Squibb |
22931505 |
69 |
Chemokine receptor antagonists. |
National Heart and Lung Institute |
16198561 |
99 |
Novel CCR1 antagonists with oral activity in the mouse collagen induced arthritis. |
Novartis Institutes For Biomedical Research |
21036044 |
43 |
Discovery of INCB3344, a potent, selective and orally bioavailable antagonist of human and murine CCR2. |
Incyte |
17446072 |
68 |
Structure-activity relationships of novel, highly potent, selective, and orally active CCR1 antagonists. |
Tanabe Research Laboratories |
11311066 |
76 |
Design, synthesis, and discovery of a novel CCR1 antagonist. |
Banyu Tsukuba Research Institute In Collaboration With Merck Research Laboratories |
30595446 |
63 |
Identification of novel azaindazole CCR1 antagonist clinical candidates. |
Boehringer Ingelheim Pharmaceuticals |