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16 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review
PMIDDataArticle TitleOrganization
25766632 31 Synthesis and biological evaluation of spirocyclic antagonists of CCR2 (chemokine CC receptor subtype 2).EBI Westf£Lische Wilhelms-Universit£T M£Nster
20627722 89 Identification of a sulfonamide series of CCR2 antagonists.EBI Glaxosmithkline
23079519 86 In vivo activity of an azole series of CCR2 antagonists.EBI Glaxosmithkline
24900425 72 Discovery of a 4-Azetidinyl-1-thiazoyl-cyclohexane CCR2 Antagonist as a Development Candidate.EBI TBA
22608963 109 The design and synthesis of novel, potent and orally bioavailable N-aryl piperazine-1-carboxamide CCR2 antagonists with very high hERG selectivity.EBI Astrazeneca
24900280 81 Discovery of INCB8761/PF-4136309, a Potent, Selective, and Orally Bioavailable CCR2 Antagonist.EBI TBA
22475558 82 Discovery of an orally-bioavailable CC Chemokine Receptor 2 antagonist derived from an acyclic diaminoalcohol backbone.EBI Bristol-Myers Squibb
24900329 49 Discovery of INCB3284, a Potent, Selective, and Orally Bioavailable hCCR2 Antagonist.EBI TBA
21341682 37 Discovery, optimization, and pharmacological characterization of novel heteroaroylphenylureas antagonists of C-C chemokine ligand 2 function.EBI Telik
21295478 81 Discovery of INCB10820/PF-4178903, a potent, selective, and orally bioavailable dual CCR2 and CCR5 antagonist.EBI Incyte
21036044 43 Discovery of INCB3344, a potent, selective and orally bioavailable antagonist of human and murine CCR2.EBI Incyte
17929797 34 Synthesis, structure-activity relationship and in vivo antiinflammatory efficacy of substituted dipiperidines as CCR2 antagonists.EBI Johnson & Johnson Pharmaceutical Research and Development
17482462 60 3-Amino-1-alkyl-cyclopentane carboxamides as small molecule antagonists of the human and murine CC chemokine receptor 2.EBI Merck Research Laboratories
17461566 11 Discovery of 3-piperidinyl-1-cyclopentanecarboxamide as a novel scaffold for highly potent CC chemokine receptor 2 antagonists.EBI Merck Research Laboratories
17092717 59 Alpha-aminothiazole-gamma-aminobutanoic amides as potent, small molecule CCR2 receptor antagonists.EBI Merck Research Laboratories