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BDBM50503048 CHEMBL4457754
SMILES: [H][C@@]12CCN[C@]1(C)CN(c1ccccc1)c1ccccc21
InChI Key: InChIKey=OHCPINQLTJGNRS-FUHWJXTLSA-N
Data: 39 KI
| Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 5-hydroxytryptamine receptor 7 (Homo sapiens (Human)) | BDBM50503048 (CHEMBL4457754) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet  | PC cid PC sid UniChem | Article PubMed | 6.30 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Minnesota Twin Cities Curated by ChEMBL | Assay Description Displacement of [3H]-LSD from human recombinant 5-HT7 receptor expressed in stable HEK cells after 90 mins by microbeta scintillation counting method | ACS Med Chem Lett 10: 1436-1442 (2019) Article DOI: 10.1021/acsmedchemlett.9b00225 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| 5-hydroxytryptamine receptor 7 (Homo sapiens (Human)) | BDBM50503048 (CHEMBL4457754) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 6.30 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Minnesota Twin Cities Curated by ChEMBL | Assay Description Displacement of [3H]-LSD from human recombinant 5-HT7 receptor expressed in stable HEK cells after 90 mins by microbeta scintillation counting method | ACS Med Chem Lett 10: 1436-1442 (2019) Article DOI: 10.1021/acsmedchemlett.9b00225 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| 5-hydroxytryptamine receptor 2B (Homo sapiens (Human)) | BDBM50503048 (CHEMBL4457754) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 501 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Minnesota Twin Cities Curated by ChEMBL | Assay Description Displacement of [3H]-LSD from human recombinant 5-HT2B receptor stably expressed in HEK cells after 90 mins by microbeta scintillation counting metho... | ACS Med Chem Lett 10: 1436-1442 (2019) Article DOI: 10.1021/acsmedchemlett.9b00225 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Sigma non-opioid intracellular receptor 1 (Homo sapiens (Human)) | BDBM50503048 (CHEMBL4457754) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 501 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Minnesota Twin Cities Curated by ChEMBL | Assay Description Displacement of [3H]-Pentazocine from human recombinant sigma1 receptor expressed in HEKT cells after 90 mins by microbeta scintillation counting met... | ACS Med Chem Lett 10: 1436-1442 (2019) Article DOI: 10.1021/acsmedchemlett.9b00225 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Sigma intracellular receptor 2 (Homo sapiens (Human)) | BDBM50503048 (CHEMBL4457754) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Minnesota Twin Cities Curated by ChEMBL | Assay Description Displacement of [3H]-Pentazocine from human recombinant sigma2 receptor expressed in HEKT cells after 90 mins by microbeta scintillation counting met... | ACS Med Chem Lett 10: 1436-1442 (2019) Article DOI: 10.1021/acsmedchemlett.9b00225 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Adrenergic receptor (Homo sapiens (Human)) | BDBM50503048 (CHEMBL4457754) | Reactome pathway KEGG UniProtKB/SwissProt UniProtKB/TrEMBL DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Minnesota Twin Cities Curated by ChEMBL | Assay Description Displacement of [3H]-Prazosin from human recombinant adrenergic Alpha1D receptor expressed in cells after 90 mins by microbeta scintillation counting... | ACS Med Chem Lett 10: 1436-1442 (2019) Article DOI: 10.1021/acsmedchemlett.9b00225 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Adrenergic receptor (Homo sapiens (Human)) | BDBM50503048 (CHEMBL4457754) | PDB UniProtKB/SwissProt UniProtKB/TrEMBL antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Minnesota Twin Cities Curated by ChEMBL | Assay Description Displacement of [3H]-Rauwolscine from human recombinant adrenergic Alpha2C receptor expressed in stable MDCK cells after 90 mins by microbeta scintil... | ACS Med Chem Lett 10: 1436-1442 (2019) Article DOI: 10.1021/acsmedchemlett.9b00225 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Monoamine transporter (Homo sapiens (Human)) | BDBM50503048 (CHEMBL4457754) | Reactome pathway KEGG UniProtKB/SwissProt UniProtKB/TrEMBL DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 1.59E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Minnesota Twin Cities Curated by ChEMBL | Assay Description Displacement of [3H]-Nisoxetine from human recombinant NET receptor expressed in stable HEK cells after 90 mins by microbeta scintillation counting m... | ACS Med Chem Lett 10: 1436-1442 (2019) Article DOI: 10.1021/acsmedchemlett.9b00225 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Histamine H2 receptor (Homo sapiens (Human)) | BDBM50503048 (CHEMBL4457754) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 2.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Minnesota Twin Cities Curated by ChEMBL | Assay Description Displacement of [125I]-Iodoaminopotentidine from human recombinant histamine H2 receptor expressed in stable HEK cells after 90 mins by microbeta sci... | ACS Med Chem Lett 10: 1436-1442 (2019) Article DOI: 10.1021/acsmedchemlett.9b00225 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Beta-1 adrenergic receptor (Homo sapiens (Human)) | BDBM50503048 (CHEMBL4457754) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 3.16E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Minnesota Twin Cities Curated by ChEMBL | Assay Description Displacement of [125I]-pindolol from human recombinant adrenergic Beta1 receptor expressed in Flp-In CHO cells after 90 mins by microbeta scintillati... | ACS Med Chem Lett 10: 1436-1442 (2019) Article DOI: 10.1021/acsmedchemlett.9b00225 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Muscarinic acetylcholine receptor M2 and M5 (Homo sapiens (Human)) | BDBM50503048 (CHEMBL4457754) | PDB UniProtKB/SwissProt UniProtKB/TrEMBL antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | <1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Minnesota Twin Cities Curated by ChEMBL | Assay Description Displacement of [3H]-QNB/[3H]-NMS from human recombinant Muscarinic acetylcholine M2 receptor expressed in stable CHO cells after 90 mins by microbet... | ACS Med Chem Lett 10: 1436-1442 (2019) Article DOI: 10.1021/acsmedchemlett.9b00225 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Muscarinic acetylcholine receptor M3 (Homo sapiens (Human)) | BDBM50503048 (CHEMBL4457754) | Reactome pathway KEGG UniProtKB/SwissProt UniProtKB/TrEMBL DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | <1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Minnesota Twin Cities Curated by ChEMBL | Assay Description Displacement of [3H]-QNB/[3H]-NMS from human recombinant Muscarinic acetylcholine M3 receptor expressed in stable CHO cells after 90 mins by microbet... | ACS Med Chem Lett 10: 1436-1442 (2019) Article DOI: 10.1021/acsmedchemlett.9b00225 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Muscarinic acetylcholine receptor M2 and M4 (Homo sapiens (Human)) | BDBM50503048 (CHEMBL4457754) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | <1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Minnesota Twin Cities Curated by ChEMBL | Assay Description Displacement of [3H]-QNB/[3H]-NMS from human recombinant Muscarinic acetylcholine M4 receptor expressed in stable CHO cells after 90 mins by microbet... | ACS Med Chem Lett 10: 1436-1442 (2019) Article DOI: 10.1021/acsmedchemlett.9b00225 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Kappa-type opioid receptor (Homo sapiens (Human)) | BDBM50503048 (CHEMBL4457754) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | <1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Minnesota Twin Cities Curated by ChEMBL | Assay Description Displacement of [3H]-U69593 from human recombinant KOR receptor expressed in stable HEK cells after 90 mins by microbeta scintillation counting metho... | ACS Med Chem Lett 10: 1436-1442 (2019) Article DOI: 10.1021/acsmedchemlett.9b00225 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Sodium-dependent dopamine transporter (Homo sapiens (Human)) | BDBM50503048 (CHEMBL4457754) | NCI pathway Reactome pathway KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | <1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Minnesota Twin Cities Curated by ChEMBL | Assay Description Displacement of [3H]-Win35428 from human recombinant DAT receptor expressed in stable HEK cells after 90 mins by microbeta scintillation counting met... | ACS Med Chem Lett 10: 1436-1442 (2019) Article DOI: 10.1021/acsmedchemlett.9b00225 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Adrenergic receptor (Homo sapiens (Human)) | BDBM50503048 (CHEMBL4457754) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | <1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Minnesota Twin Cities Curated by ChEMBL | Assay Description Displacement of [3H]-Prazosin from human recombinant adrenergic Alpha1B receptor expressed in HEKT cells after 90 mins by microbeta scintillation cou... | ACS Med Chem Lett 10: 1436-1442 (2019) Article DOI: 10.1021/acsmedchemlett.9b00225 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Delta-type opioid receptor (Homo sapiens (Human)) | BDBM50503048 (CHEMBL4457754) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | <1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Minnesota Twin Cities Curated by ChEMBL | Assay Description Displacement of [3H]-DADLE from human recombinant DOR receptor expressed in stable HEK cells after 90 mins by microbeta scintillation counting method | ACS Med Chem Lett 10: 1436-1442 (2019) Article DOI: 10.1021/acsmedchemlett.9b00225 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Muscarinic acetylcholine receptor M5 (Homo sapiens (Human)) | BDBM50503048 (CHEMBL4457754) | Reactome pathway KEGG UniProtKB/SwissProt UniProtKB/TrEMBL DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | <1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Minnesota Twin Cities Curated by ChEMBL | Assay Description Displacement of [3H]-QNB/[3H]-NMS from human recombinant Muscarinic acetylcholine M5 receptor expressed in stable CHO cells after 90 mins by microbet... | ACS Med Chem Lett 10: 1436-1442 (2019) Article DOI: 10.1021/acsmedchemlett.9b00225 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| D(3) dopamine receptor (Homo sapiens (Human)) | BDBM50503048 (CHEMBL4457754) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | <1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Minnesota Twin Cities Curated by ChEMBL | Assay Description Displacement of [3H]-N-methylspiperone from human recombinant dopamine D3 receptor expressed in HEKT cells after 90 mins by microbeta scintillation c... | ACS Med Chem Lett 10: 1436-1442 (2019) Article DOI: 10.1021/acsmedchemlett.9b00225 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| 5-hydroxytryptamine receptor 2C (Homo sapiens (Human)) | BDBM50503048 (CHEMBL4457754) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | <1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Minnesota Twin Cities Curated by ChEMBL | Assay Description Displacement of [3H]-Mesulergine from human recombinant 5-HT2C receptor expressed in HEKT cells after 90 mins by microbeta scintillation counting met... | ACS Med Chem Lett 10: 1436-1442 (2019) Article DOI: 10.1021/acsmedchemlett.9b00225 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Beta-2 adrenergic receptor and beta-3 adrenergic receptor (Homo sapiens (Human)) | BDBM50503048 (CHEMBL4457754) | PDB Reactome pathway KEGG UniProtKB/SwissProt UniProtKB/TrEMBL DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | <1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Minnesota Twin Cities Curated by ChEMBL | Assay Description Displacement of [3H]-CGP12177 from human recombinant adrenergic Beta3 receptor expressed in Flp-In HEK cells after 90 mins by microbeta scintillation... | ACS Med Chem Lett 10: 1436-1442 (2019) Article DOI: 10.1021/acsmedchemlett.9b00225 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Adrenergic receptor (Homo sapiens (Human)) | BDBM50503048 (CHEMBL4457754) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | <1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Minnesota Twin Cities Curated by ChEMBL | Assay Description Displacement of [3H]-Rauwolscine from human recombinant adrenergic Alpha2B receptor expressed in HEKT cells after 90 mins by microbeta scintillation ... | ACS Med Chem Lett 10: 1436-1442 (2019) Article DOI: 10.1021/acsmedchemlett.9b00225 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Serotonin (5-HT) receptor (Homo sapiens (Human)) | BDBM50503048 (CHEMBL4457754) | PDB Reactome pathway KEGG UniProtKB/SwissProt UniProtKB/TrEMBL DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | <1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Minnesota Twin Cities Curated by ChEMBL | Assay Description Displacement of [3H]5-CT from human recombinant 5-HT1B receptor expressed in stable HEK cells after 90 mins by microbeta scintillation counting metho... | ACS Med Chem Lett 10: 1436-1442 (2019) Article DOI: 10.1021/acsmedchemlett.9b00225 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Histamine H1 receptor (Homo sapiens (Human)) | BDBM50503048 (CHEMBL4457754) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | <1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Minnesota Twin Cities Curated by ChEMBL | Assay Description Displacement of [3H]-Pyrilamine from human recombinant histamine H1 receptor expressed in stable HEK cells after 90 mins by microbeta scintillation c... | ACS Med Chem Lett 10: 1436-1442 (2019) Article DOI: 10.1021/acsmedchemlett.9b00225 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Muscarinic acetylcholine receptor M1 (Homo sapiens (Human)) | BDBM50503048 (CHEMBL4457754) | UniProtKB/SwissProt UniProtKB/TrEMBL antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | <1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Minnesota Twin Cities Curated by ChEMBL | Assay Description Displacement of [3H]-QNB/[3H]-NMS from human recombinant Muscarinic acetylcholine M1 receptor expressed in stable CHO cells after 90 mins by microbet... | ACS Med Chem Lett 10: 1436-1442 (2019) Article DOI: 10.1021/acsmedchemlett.9b00225 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Mu-type opioid receptor (Homo sapiens (Human)) | BDBM50503048 (CHEMBL4457754) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | <1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Minnesota Twin Cities Curated by ChEMBL | Assay Description Displacement of [3H]-DAMGO from human recombinant MOR receptor expressed in stable HEK cells after 90 mins by microbeta scintillation counting method | ACS Med Chem Lett 10: 1436-1442 (2019) Article DOI: 10.1021/acsmedchemlett.9b00225 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| D(4) dopamine receptor (Homo sapiens (Human)) | BDBM50503048 (CHEMBL4457754) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | <1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Minnesota Twin Cities Curated by ChEMBL | Assay Description Displacement of [3H]-methylspiperone from human recombinant dopamine D4 receptor expressed in Stable HEK cells after 90 mins by microbeta scintillati... | ACS Med Chem Lett 10: 1436-1442 (2019) Article DOI: 10.1021/acsmedchemlett.9b00225 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Serotonin (5-HT) receptor (Homo sapiens (Human)) | BDBM50503048 (CHEMBL4457754) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | <1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Minnesota Twin Cities Curated by ChEMBL | Assay Description Displacement of [3H]5-CT from human recombinant 5-HT1D receptor transiently expressed in HEKT cells after 90 mins by microbeta scintillation counting... | ACS Med Chem Lett 10: 1436-1442 (2019) Article DOI: 10.1021/acsmedchemlett.9b00225 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Histamine receptor (H3 and H4) (Homo sapiens (Human)) | BDBM50503048 (CHEMBL4457754) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | <1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Minnesota Twin Cities Curated by ChEMBL | Assay Description Displacement of [3H]-Histamine from human recombinant histamine H4 receptor expressed in HEKT cells after 90 mins by microbeta scintillation counting... | ACS Med Chem Lett 10: 1436-1442 (2019) Article DOI: 10.1021/acsmedchemlett.9b00225 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Serotonin (5-HT) receptor (Homo sapiens (Human)) | BDBM50503048 (CHEMBL4457754) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | <1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Minnesota Twin Cities Curated by ChEMBL | Assay Description Displacement of [3H]-HT from human recombinant 5-HT1E receptor expressed in stable HEK cells after 90 mins by microbeta scintillation counting method | ACS Med Chem Lett 10: 1436-1442 (2019) Article DOI: 10.1021/acsmedchemlett.9b00225 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| 5-hydroxytryptamine receptor 3A (Homo sapiens (Human)) | BDBM50503048 (CHEMBL4457754) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | <1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Minnesota Twin Cities Curated by ChEMBL | Assay Description Displacement of [3H]-GR65630 from human recombinant 5-HT3 receptor expressed in HEKT cells after 90 mins by microbeta scintillation counting method | ACS Med Chem Lett 10: 1436-1442 (2019) Article DOI: 10.1021/acsmedchemlett.9b00225 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| 5-hydroxytryptamine receptor 6 (Homo sapiens (Human)) | BDBM50503048 (CHEMBL4457754) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | <1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Minnesota Twin Cities Curated by ChEMBL | Assay Description Displacement of [3H]-LSD from human recombinant 5-HT6 receptor expressed in stable HEK cells after 90 mins by microbeta scintillation counting method | ACS Med Chem Lett 10: 1436-1442 (2019) Article DOI: 10.1021/acsmedchemlett.9b00225 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Alpha-1A adrenergic receptor (Homo sapiens (Human)) | BDBM50503048 (CHEMBL4457754) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | <1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Minnesota Twin Cities Curated by ChEMBL | Assay Description Displacement of [3H]-Prazosin from human recombinant adrenergic alpha1A receptor expressed in cells after 90 mins by microbeta scintillation counting... | ACS Med Chem Lett 10: 1436-1442 (2019) Article DOI: 10.1021/acsmedchemlett.9b00225 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| D(1A) dopamine receptor (Homo sapiens (Human)) | BDBM50503048 (CHEMBL4457754) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | <1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Minnesota Twin Cities Curated by ChEMBL | Assay Description Displacement of [3H]-SCH23390 from human recombinant dopamine D1 receptor expressed in HEKT cells after 90 mins by microbeta scintillation counting m... | ACS Med Chem Lett 10: 1436-1442 (2019) Article DOI: 10.1021/acsmedchemlett.9b00225 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| D(2) dopamine receptor (Homo sapiens (Human)) | BDBM50503048 (CHEMBL4457754) | PDB Reactome pathway KEGG UniProtKB/SwissProt UniProtKB/TrEMBL DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | <1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Minnesota Twin Cities Curated by ChEMBL | Assay Description Displacement of [3H]-N-methylspiperone from human recombinant dopamine D2 receptor expressed in stable fibroblast cells after 90 mins by microbeta sc... | ACS Med Chem Lett 10: 1436-1442 (2019) Article DOI: 10.1021/acsmedchemlett.9b00225 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| D(1B) dopamine receptor (Homo sapiens (Human)) | BDBM50503048 (CHEMBL4457754) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | <1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Minnesota Twin Cities Curated by ChEMBL | Assay Description Displacement of [3H]-SCH23390 from human recombinant dopamine D5 receptor expressed in HEKT cells after 90 mins by microbeta scintillation counting m... | ACS Med Chem Lett 10: 1436-1442 (2019) Article DOI: 10.1021/acsmedchemlett.9b00225 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| 5-hydroxytryptamine receptor 1A (Homo sapiens (Human)) | BDBM50503048 (CHEMBL4457754) | PDB UniProtKB/SwissProt UniProtKB/TrEMBL antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Minnesota Twin Cities Curated by ChEMBL | Assay Description Displacement of [3H]-Way100635 from human recombinant 5-HT1A expressed in stable CHO cells after 90 mins by microbeta scintillation counting method | ACS Med Chem Lett 10: 1436-1442 (2019) Article DOI: 10.1021/acsmedchemlett.9b00225 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Beta-2 adrenergic receptor (Homo sapiens (Human)) | BDBM50503048 (CHEMBL4457754) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt UniProtKB/TrEMBL B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | <1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Minnesota Twin Cities Curated by ChEMBL | Assay Description Displacement of [3H]-CGP12177 from human recombinant adrenergic Beta2 receptor expressed in Flp-In HEK cells after 90 mins by microbeta scintillation... | ACS Med Chem Lett 10: 1436-1442 (2019) Article DOI: 10.1021/acsmedchemlett.9b00225 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| 5-hydroxytryptamine receptor 1A (Homo sapiens (Human)) | BDBM50503048 (CHEMBL4457754) | PDB UniProtKB/SwissProt UniProtKB/TrEMBL antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | <1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Minnesota Twin Cities Curated by ChEMBL | Assay Description Displacement of [3H]-Way100635 from human recombinant 5-HT1A expressed in stable CHO cells after 90 mins by microbeta scintillation counting method | ACS Med Chem Lett 10: 1436-1442 (2019) Article DOI: 10.1021/acsmedchemlett.9b00225 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
