BDBM101503 US8524710, 81::US8530652, 30::US8530652, 74
SMILES: CC1(C)N(Cc2c(Nc3ccnc(n3)C(F)(F)F)[nH]nc12)C(=O)NC1C[C@@H]1c1ccccc1
InChI Key: InChIKey=OLUNGVPQMWVIAU-AFYYWNPRSA-N
Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Serine/threonine-protein kinase PAK 4 (Homo sapiens (Human)) | BDBM101503 (US8524710, 81 | US8530652, 30 | US8530652, 74) | PDB MMDB Reactome pathway KEGG B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | 80 | n/a | n/a | n/a | 968 | n/a | n/a | n/a | n/a |
Agouron Pharmaceuticals, Inc.; Pfizer Inc. US Patent | Assay Description The enzymatic activity of PAK4 KD was measured by its ability to catalyzed the transfer of a phosphate residue from a nucleoside triphosphate to an a... | US Patent US8530652 (2013) BindingDB Entry DOI: 10.7270/Q2F18XC4 | |||||||||||
More data for this Ligand-Target Pair |