BDBM101538 US8530494, 208::US8530652, 116::US8530652, 65
SMILES: CN(C)C[C@@H](NC(=O)N1Cc2c(Nc3ccnc(C)n3)[nH]nc2C1(C)C)c1ccccc1
InChI Key: InChIKey=HEYDCDKYVGFDOG-GOSISDBHSA-N
Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Serine/threonine-protein kinase PAK 4 (Homo sapiens (Human)) | BDBM101538 (US8530494, 208 | US8530652, 116 | US8530652, 65) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt UniProtKB/TrEMBL B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | 680 | n/a | n/a | n/a | 67.1 | n/a | n/a | n/a | n/a |
Agouron Pharmaceuticals, Inc.; Pfizer Inc. US Patent | Assay Description The enzymatic activity of PAK4 KD was measured by its ability to catalyzed the transfer of a phosphate residue from a nucleoside triphosphate to an a... | US Patent US8530652 (2013) BindingDB Entry DOI: 10.7270/Q2F18XC4 | |||||||||||
More data for this Ligand-Target Pair |