null
SMILES: Cc1cc2c(NC(=O)N[C@H]3CC[C@@H](C3)c3ccccc3F)c(F)ccc2cn1
InChI Key: InChIKey=PJVXUKARZNCIRA-HOCLYGCPSA-N
Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Transient receptor potential cation channel subfamily V member 1 (Homo sapiens (Human)) | BDBM128902 (US8802711, 71) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 8.60 | n/a | n/a | n/a | n/a | n/a | n/a |
AbbVie Inc. US Patent | Assay Description The functional activity of compounds at the TRPV1 receptor was determined by measurement of intracellular Ca2+ levels ([Ca2+]i) using the Fluorescenc... | US Patent US8802711 (2014) BindingDB Entry DOI: 10.7270/Q2QZ28NC | |||||||||||
More data for this Ligand-Target Pair |