BDBM183387 US9150546, I-561::US9688643, I-561::US9718790, I-0570
SMILES: CC(C)Oc1ccc(cc1Cl)\N=c1/[nH]c(=O)n([C@H](C)CC(O)=O)c(=O)n1Cc1ccc(Cl)cc1
InChI Key:
Data: 3 IC50
Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
P2X purinoceptor 3 (Homo sapiens (Human)) | BDBM183387 (US9150546, I-561 | US9688643, I-561 | US9718790, I...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 8 | n/a | n/a | n/a | n/a | 7.5 | 37 |
SHIONOGI & CO., LTD. US Patent | Assay Description Stably expressing cell line (C6BU-1 cell transfected with human P2X3 receptor gene (GenBank accession number Y07683)) was used. The cells were seeded... | US Patent US9150546 (2015) BindingDB Entry DOI: 10.7270/Q2416VV1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P2X purinoceptor 3 (Homo sapiens (Human)) | BDBM183387 (US9150546, I-561 | US9688643, I-561 | US9718790, I...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 8 | n/a | n/a | n/a | n/a | 7.5 | n/a |
SHIONOGI & CO., LTD. US Patent | Assay Description Stably expressing cell line (C6BU-1 transfected with human P2X3 receptor gene (GenBank accession number Y07683) was used. The cells were seeded in a ... | US Patent US9718790 (2017) BindingDB Entry DOI: 10.7270/Q22809KB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucocorticoid receptor (Homo sapiens (Human)) | BDBM183387 (US9150546, I-561 | US9688643, I-561 | US9718790, I...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 8 | n/a | n/a | n/a | n/a | n/a | n/a |
SRMLSC US Patent | Assay Description Stably expressing cell line (C6BU-1 cell transfected with human P2X3 receptor gene (GenBank accession number Y07683)) was used. The cells were seeded... | US Patent US9688643 (2017) BindingDB Entry DOI: 10.7270/Q2M32SZ2 | |||||||||||
More data for this Ligand-Target Pair |