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BDBM234297 Met-ψ[P(O)(OH)CH2]-Ala (5)

SMILES: CSCCC(N)P(O)(=O)CC(C)C(O)=O

InChI Key: InChIKey=KVCYRBIAXSOETM-UHFFFAOYNA-N

Data: 1 KI

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 234297   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kcal/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Leucine aminopeptidase (LAP)


(Sus scrofa (Pig))
BDBM234297
PNG
(Met-ψ[P(O)(OH)CH2]-Ala (5))
Show SMILES CSCCC(N)P(O)(=O)CC(C)C(O)=O
Show InChI InChI=1/C8H18NO4PS/c1-6(8(10)11)5-14(12,13)7(9)3-4-15-2/h6-7H,3-5,9H2,1-2H3,(H,10,11)(H,12,13)
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
3.64E+3 -7.41n/an/an/an/an/a8.425



Academy of Sciences of the Czech Republic



Assay Description
LAP was assayed in 75 mM triethanolamine hydrochloride buffer (pH = 8.4, containing 5 mM MgCl2) at 25C. The substrate (L-leucine-p-nitroanilide) was...


J Enzyme Inhib Med Chem 26: 155-61 (2011)


Article DOI: 10.3109/14756366.2010.482047
More data for this
Ligand-Target Pair