BDBM260769 US9533989, 80
SMILES: Cc1cccc(c1)C(=O)N1CCc2ccc(Nc3nc(N[C@@H]4CCCC[C@@H]4N)ncc3C(N)=O)cc2C1
InChI Key: InChIKey=OSFSLYLWSVRCJL-BJKOFHAPSA-N
Data: 1 IC50
Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Tyrosine-protein kinase SYK (Homo sapiens (Human)) | BDBM260769 (US9533989, 80) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt UniProtKB/TrEMBL B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 36.4 | n/a | n/a | n/a | n/a | n/a | n/a |
Ziarco Pharma Ltd. US Patent | Assay Description The Promega ADP-Glo Kinase Assay is a luminescent ADP detection assay that provides a universal, homogeneous, high-throughput screening method to mea... | US Patent US9533989 (2017) BindingDB Entry DOI: 10.7270/Q2VQ31M7 | |||||||||||
More data for this Ligand-Target Pair |