BindingDB logo
myBDB logout

BDBM308046 (S)-1-(1H- benzo[d]imidazol-5-yl)-5-(4- propoxyphenyl)imidazolidin- 2-one::US9650362, 14

SMILES: CCCOc1ccc(cc1)[C@H]1CNC(=O)N1c1ccc2[nH]cnc2c1

InChI Key:

Data: 1 KI  1 IC50

Find this compound or compounds like it in BindingDB or PDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 308046   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kcal/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Glutaminyl-peptide cyclotransferase


(Homo sapiens (Human))
BDBM308046
PNG
((S)-1-(1H- benzo[d]imidazol-5-yl)-5-(4- propoxyphe...)
Show SMILES CCCOc1ccc(cc1)[C@H]1CNC(=O)N1c1ccc2[nH]cnc2c1 |r|
PDB
MMDB

KEGG

UniProtKB/SwissProt

B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet 
Purchase

PC cid
PC sid
UniChem
US Patent
37.4n/an/an/an/an/an/an/an/a



PROBIODRUG AG

US Patent


Assay Description
All measurements were performed with a BioAssay Reader HTS-7000Plus for microplates (Perkin Elmer) at 30° C. QC activity was evaluated fluorometrical...


US Patent US9650362 (2017)


BindingDB Entry DOI: 10.7270/Q2VD71H9
More data for this
Ligand-Target Pair
Glutaminyl-peptide cyclotransferase


(Homo sapiens (Human))
BDBM308046
PNG
((S)-1-(1H- benzo[d]imidazol-5-yl)-5-(4- propoxyphe...)
Show SMILES CCCOc1ccc(cc1)[C@H]1CNC(=O)N1c1ccc2[nH]cnc2c1 |r|
PDB
MMDB

KEGG

UniProtKB/SwissProt

B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet 
Purchase

PC cid
PC sid
UniChem
US Patent
n/an/a 238n/an/an/an/an/an/a



PROBIODRUG AG

US Patent


Assay Description
All measurements were performed with a BioAssay Reader HTS-7000Plus for microplates (Perkin Elmer) at 30° C. QC activity was evaluated fluorometrical...


US Patent US9650362 (2017)


BindingDB Entry DOI: 10.7270/Q2VD71H9
More data for this
Ligand-Target Pair