null

SMILES: [C-]#[N+]c1[nH]nnc1-c1ccnc(c1)-c1cn(CC2CCCc3ccccc23)cn1

InChI Key:

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 319596   

Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50/IC50 nM	koff s-1	kon M-1s-1	pH	Temp °C
Histone lysine demethylase PHF8 (Homo sapiens (Human))	BDBM319596 (4-[2-[1-(1,2,3,4-tetrahydronaphthalen- 1-ylmethyl)...) Show SMILES [C-]#[N+]c1[nH]nnc1-c1ccnc(c1)-c1cn(CC2CCCc3ccccc23)cn1 Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	550	n/a	n/a	n/a	n/a	n/a	n/a
Celgene Quanticel Research, Inc. US Patent					Assay Description The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction conditions: 3 nM P...				US Patent US10174003 (2019) BindingDB Entry DOI: 10.7270/Q2417053
					More data for this Ligand-Target Pair
Lysine-specific demethylase 2B (Homo sapiens (Human))	BDBM319596 (4-[2-[1-(1,2,3,4-tetrahydronaphthalen- 1-ylmethyl)...) Show SMILES [C-]#[N+]c1[nH]nnc1-c1ccnc(c1)-c1cn(CC2CCCc3ccccc23)cn1 Show InChI	PDB UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<100	n/a	n/a	n/a	n/a	n/a	n/a
Celgene Quanticel Research, Inc. US Patent					Assay Description The ability of test compounds to inhibit the activity of FBXL10 was determined in 384-well plate format under the following reaction conditions: 0.3 ...				US Patent US10174003 (2019) BindingDB Entry DOI: 10.7270/Q2417053
					More data for this Ligand-Target Pair