BDBM50008404 CHEMBL3235541
SMILES: CCOc1ccc2nc(NC(=O)Cc3cccc(Cl)c3)sc2c1
InChI Key: InChIKey=DCFRVNRCHQVUOD-UHFFFAOYSA-N
Data: 1 IC50
Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Casein kinase I isoform delta (Homo sapiens (Human)) | BDBM50008404 (CHEMBL3235541) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.21E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
CSIC Curated by ChEMBL | Assay Description Inhibition of human recombinant CK-1delta using casein as substrate after 60 mins by Kinase-Glo assay | J Med Chem 57: 2755-72 (2014) Article DOI: 10.1021/jm500065f BindingDB Entry DOI: 10.7270/Q21N82NV | |||||||||||
More data for this Ligand-Target Pair |