BDBM50018339 3'-(Cyclohepta-1,3,5-trienyloxy)-biphenyl-4-carboxylic acid (4-pyridin-3-yl-butyl)-amide::CHEMBL50050
SMILES: O=C(NCCCCc1cccnc1)c1ccc(cc1)-c1cccc(OC2=CC=CC=CC2)c1
InChI Key: InChIKey=OXVZHFKZGCMBCC-UHFFFAOYSA-N
Data: 1 IC50
Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Platelet-activating factor receptor (Homo sapiens (Human)) | BDBM50018339 (3'-(Cyclohepta-1,3,5-trienyloxy)-biphenyl-4-carbox...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | PubMed | n/a | n/a | 700 | n/a | n/a | n/a | n/a | n/a | n/a |
Roche Research Center Curated by ChEMBL | Assay Description Inhibition of platelet-activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand. | J Med Chem 32: 1814-20 (1989) BindingDB Entry DOI: 10.7270/Q2SQ8ZCJ | |||||||||||
More data for this Ligand-Target Pair |