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SMILES: Cc1nc2cnccc2n1-c1ccc(cc1)C1=Nc2nc(C)cc(C)c2NC(=O)C1

InChI Key: InChIKey=HPDPZQPMNFMUFQ-UHFFFAOYSA-N

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50033227   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kcal/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Platelet-activating factor receptor


(Cavia porcellus)		BDBM50033227
PNG
(7,9-Dimethyl-4-[4-(2-methyl-imidazo[4,5-c]pyridin-...)
Show SMILES Cc1nc2cnccc2n1-c1ccc(cc1)C1=Nc2nc(C)cc(C)c2NC(=O)C1 |t:19|
Show InChI InChI=1S/C23H20N6O/c1-13-10-14(2)25-23-22(13)28-21(30)11-18(27-23)16-4-6-17(7-5-16)29-15(3)26-19-12-24-9-8-20(19)29/h4-10,12H,11H2,1-3H3,(H,28,30)
MMDB

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n/an/a 21n/an/an/an/an/an/a



Pfizer Central Research

Curated by ChEMBL


Assay Description
In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit platelets

J Med Chem 38: 3524-35 (1995)


BindingDB Entry DOI: 10.7270/Q2JS9R2X
More data for this
Ligand-Target Pair