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SMILES: Cc1nc2cnccc2n1-c1ccc(cc1)C1=Nc2cc(C)c(C)cc2-n2nnnc2C1

InChI Key: InChIKey=RVZSGDUCSBXFBV-UHFFFAOYSA-N

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50033248   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kcal/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Platelet-activating factor receptor


(Cavia porcellus)		BDBM50033248
PNG
(8,9-Dimethyl-5-[4-(2-methyl-imidazo[4,5-c]pyridin-...)
Show SMILES Cc1nc2cnccc2n1-c1ccc(cc1)C1=Nc2cc(C)c(C)cc2-n2nnnc2C1 |t:19|
Show InChI InChI=1S/C24H20N8/c1-14-10-20-23(11-15(14)2)32-24(28-29-30-32)12-19(27-20)17-4-6-18(7-5-17)31-16(3)26-21-13-25-9-8-22(21)31/h4-11,13H,12H2,1-3H3
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n/an/a 11n/an/an/an/an/an/a



Pfizer Central Research

Curated by ChEMBL


Assay Description
In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit platelets

J Med Chem 38: 3524-35 (1995)


BindingDB Entry DOI: 10.7270/Q2JS9R2X
More data for this
Ligand-Target Pair