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SMILES: Cc1nc2cnccc2n1-c1ccc(cc1)C1=Nc2cccnc2NC(=O)C1

InChI Key: InChIKey=SEZZDCVZNXXFKS-UHFFFAOYSA-N

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50033259   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kcal/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Platelet-activating factor receptor


(Cavia porcellus)		BDBM50033259
PNG
(2-[4-(2-Methyl-imidazo[4,5-c]pyridin-1-yl)-phenyl]...)
Show SMILES Cc1nc2cnccc2n1-c1ccc(cc1)C1=Nc2cccnc2NC(=O)C1 |t:19|
Show InChI InChI=1S/C21H16N6O/c1-13-24-18-12-22-10-8-19(18)27(13)15-6-4-14(5-7-15)17-11-20(28)26-21-16(25-17)3-2-9-23-21/h2-10,12H,11H2,1H3,(H,23,26,28)
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n/an/a 130n/an/an/an/an/an/a



Pfizer Central Research

Curated by ChEMBL


Assay Description
In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit platelets

J Med Chem 38: 3524-35 (1995)


BindingDB Entry DOI: 10.7270/Q2JS9R2X
More data for this
Ligand-Target Pair