Found 16 hits for monomerid = 50136493 Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
Imidazoline receptor 1 (I1R)
(Homo sapiens (Human)) | BDBM50136493
(1-Methyl-4,9-dihydro-3H-beta-carboline | 1-methyl-...)Show InChI InChI=1S/C12H12N2/c1-8-12-10(6-7-13-8)9-4-2-3-5-11(9)14-12/h2-5,14H,6-7H2,1H3 | PDB
UniProtKB/SwissProt
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| 46 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Virginia Commonwealth University
Curated by ChEMBL
| Assay Description Binding affinity towards Imidazoline I1 receptor |
Bioorg Med Chem Lett 13: 4421-5 (2003)
BindingDB Entry DOI: 10.7270/Q2D21X2G |
More data for this Ligand-Target Pair | |
Nischarin
(Homo sapiens (Human)) | BDBM50136493
(1-Methyl-4,9-dihydro-3H-beta-carboline | 1-methyl-...)Show InChI InChI=1S/C12H12N2/c1-8-12-10(6-7-13-8)9-4-2-3-5-11(9)14-12/h2-5,14H,6-7H2,1H3 | PDB
UniProtKB/SwissProt
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| 148 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Virginia Commonwealth University
Curated by ChEMBL
| Assay Description Binding affinity for rat 5-hydroxytryptamine 2A receptor using [3H]-DOB |
Bioorg Med Chem Lett 13: 4421-5 (2003)
BindingDB Entry DOI: 10.7270/Q2D21X2G |
More data for this Ligand-Target Pair | |
5-hydroxytryptamine receptor 7
(Homo sapiens (Human)) | BDBM50136493
(1-Methyl-4,9-dihydro-3H-beta-carboline | 1-methyl-...)Show InChI InChI=1S/C12H12N2/c1-8-12-10(6-7-13-8)9-4-2-3-5-11(9)14-12/h2-5,14H,6-7H2,1H3 | Reactome pathway KEGG
UniProtKB/SwissProt
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| 280 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Virginia Commonwealth University
Curated by ChEMBL
| Assay Description Binding affinity towards 5-hydroxytryptamine 7 receptor |
Bioorg Med Chem Lett 13: 4421-5 (2003)
BindingDB Entry DOI: 10.7270/Q2D21X2G |
More data for this Ligand-Target Pair | |
5-hydroxytryptamine receptor 5A
(Homo sapiens (Human)) | BDBM50136493
(1-Methyl-4,9-dihydro-3H-beta-carboline | 1-methyl-...)Show InChI InChI=1S/C12H12N2/c1-8-12-10(6-7-13-8)9-4-2-3-5-11(9)14-12/h2-5,14H,6-7H2,1H3 | KEGG
UniProtKB/SwissProt UniProtKB/TrEMBL
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| 845 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Virginia Commonwealth University
Curated by ChEMBL
| Assay Description Binding affinity towards 5-HT5A receptor |
Bioorg Med Chem Lett 13: 4421-5 (2003)
BindingDB Entry DOI: 10.7270/Q2D21X2G |
More data for this Ligand-Target Pair | |
5-hydroxytryptamine receptor 2A
(Rattus norvegicus (rat)) | BDBM50136493
(1-Methyl-4,9-dihydro-3H-beta-carboline | 1-methyl-...)Show InChI InChI=1S/C12H12N2/c1-8-12-10(6-7-13-8)9-4-2-3-5-11(9)14-12/h2-5,14H,6-7H2,1H3 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
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| 1.15E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Virginia Commonwealth University
Curated by ChEMBL
| Assay Description Binding affinity towards 5-hydroxytryptamine 2A receptor |
Bioorg Med Chem Lett 13: 4421-5 (2003)
BindingDB Entry DOI: 10.7270/Q2D21X2G |
More data for this Ligand-Target Pair | |
5-hydroxytryptamine receptor 6
(Homo sapiens (Human)) | BDBM50136493
(1-Methyl-4,9-dihydro-3H-beta-carboline | 1-methyl-...)Show InChI InChI=1S/C12H12N2/c1-8-12-10(6-7-13-8)9-4-2-3-5-11(9)14-12/h2-5,14H,6-7H2,1H3 | Reactome pathway KEGG
UniProtKB/SwissProt
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| 1.45E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Virginia Commonwealth University
Curated by ChEMBL
| Assay Description Binding affinity towards human 5-hydroxytryptamine 6 receptor |
Bioorg Med Chem Lett 13: 4421-5 (2003)
BindingDB Entry DOI: 10.7270/Q2D21X2G |
More data for this Ligand-Target Pair | |
5-hydroxytryptamine receptor 1A
(Homo sapiens (Human)) | BDBM50136493
(1-Methyl-4,9-dihydro-3H-beta-carboline | 1-methyl-...)Show InChI InChI=1S/C12H12N2/c1-8-12-10(6-7-13-8)9-4-2-3-5-11(9)14-12/h2-5,14H,6-7H2,1H3 | PDB
UniProtKB/SwissProt UniProtKB/TrEMBL
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| >1.67E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Virginia Commonwealth University
Curated by ChEMBL
| Assay Description Binding affinity towards 5-hydroxytryptamine 1A receptor |
Bioorg Med Chem Lett 13: 4421-5 (2003)
BindingDB Entry DOI: 10.7270/Q2D21X2G |
More data for this Ligand-Target Pair | |
5-hydroxytryptamine receptor 2C
(Homo sapiens (Human)) | BDBM50136493
(1-Methyl-4,9-dihydro-3H-beta-carboline | 1-methyl-...)Show InChI InChI=1S/C12H12N2/c1-8-12-10(6-7-13-8)9-4-2-3-5-11(9)14-12/h2-5,14H,6-7H2,1H3 | Reactome pathway KEGG
UniProtKB/SwissProt
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| 1.86E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Virginia Commonwealth University
Curated by ChEMBL
| Assay Description Binding affinity towards 5-hydroxytryptamine 2C receptor |
Bioorg Med Chem Lett 13: 4421-5 (2003)
BindingDB Entry DOI: 10.7270/Q2D21X2G |
More data for this Ligand-Target Pair | |
Dopamine receptor
(Homo sapiens (Human)) | BDBM50136493
(1-Methyl-4,9-dihydro-3H-beta-carboline | 1-methyl-...)Show InChI InChI=1S/C12H12N2/c1-8-12-10(6-7-13-8)9-4-2-3-5-11(9)14-12/h2-5,14H,6-7H2,1H3 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt UniProtKB/TrEMBL
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| >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Virginia Commonwealth University
Curated by ChEMBL
| Assay Description Binding affinity towards cloned rat Inhibition of binding towards 5-hydroxytryptamine 2A receptor at 100 nM concentration was determined using [3H]-D... |
Bioorg Med Chem Lett 13: 4421-5 (2003)
BindingDB Entry DOI: 10.7270/Q2D21X2G |
More data for this Ligand-Target Pair | |
Muscarinic acetylcholine receptor
(Homo sapiens (Human)) | BDBM50136493
(1-Methyl-4,9-dihydro-3H-beta-carboline | 1-methyl-...)Show InChI InChI=1S/C12H12N2/c1-8-12-10(6-7-13-8)9-4-2-3-5-11(9)14-12/h2-5,14H,6-7H2,1H3 | PDB MMDB
NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt UniProtKB/TrEMBL
B.MOAD DrugBank antibodypedia antibodypedia antibodypedia antibodypedia antibodypedia GoogleScholar AffyNet
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| >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Virginia Commonwealth University
Curated by ChEMBL
| Assay Description Binding affinity for rat 5-hydroxytryptamine 2A receptor using [3H]-DOB |
Bioorg Med Chem Lett 13: 4421-5 (2003)
BindingDB Entry DOI: 10.7270/Q2D21X2G |
More data for this Ligand-Target Pair | |
Metabotropic glutamate receptor
(Rattus norvegicus-Rattus norvegicus (Rat)-RAT) | BDBM50136493
(1-Methyl-4,9-dihydro-3H-beta-carboline | 1-methyl-...)Show InChI InChI=1S/C12H12N2/c1-8-12-10(6-7-13-8)9-4-2-3-5-11(9)14-12/h2-5,14H,6-7H2,1H3 | PDB
UniProtKB/SwissProt UniProtKB/TrEMBL
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| >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Virginia Commonwealth University
Curated by ChEMBL
| Assay Description Binding affinity towards Alpha-2B adrenergic receptor |
Bioorg Med Chem Lett 13: 4421-5 (2003)
BindingDB Entry DOI: 10.7270/Q2D21X2G |
More data for this Ligand-Target Pair | |
SLC6A3
(BOVINE) | BDBM50136493
(1-Methyl-4,9-dihydro-3H-beta-carboline | 1-methyl-...)Show InChI InChI=1S/C12H12N2/c1-8-12-10(6-7-13-8)9-4-2-3-5-11(9)14-12/h2-5,14H,6-7H2,1H3 | UniProtKB/SwissProt
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| >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Virginia Commonwealth University
Curated by ChEMBL
| Assay Description Binding affinity towards DAT (bovine) |
Bioorg Med Chem Lett 13: 4421-5 (2003)
BindingDB Entry DOI: 10.7270/Q2D21X2G |
More data for this Ligand-Target Pair | |
5-hydroxytryptamine receptor 1D
(Homo sapiens (Human)) | BDBM50136493
(1-Methyl-4,9-dihydro-3H-beta-carboline | 1-methyl-...)Show InChI InChI=1S/C12H12N2/c1-8-12-10(6-7-13-8)9-4-2-3-5-11(9)14-12/h2-5,14H,6-7H2,1H3 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet
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CHEMBL PC cid PC sid UniChem
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| >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Virginia Commonwealth University
Curated by ChEMBL
| Assay Description Binding affinity towards 5-hydroxytryptamine 1D receptor |
Bioorg Med Chem Lett 13: 4421-5 (2003)
BindingDB Entry DOI: 10.7270/Q2D21X2G |
More data for this Ligand-Target Pair | |
Sodium-dependent serotonin transporter
(Homo sapiens (Human)) | BDBM50136493
(1-Methyl-4,9-dihydro-3H-beta-carboline | 1-methyl-...)Show InChI InChI=1S/C12H12N2/c1-8-12-10(6-7-13-8)9-4-2-3-5-11(9)14-12/h2-5,14H,6-7H2,1H3 | PDB
KEGG
UniProtKB/SwissProt
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CHEMBL PC cid PC sid UniChem
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| >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Virginia Commonwealth University
Curated by ChEMBL
| Assay Description Binding affinity towards Serotonin transporter |
Bioorg Med Chem Lett 13: 4421-5 (2003)
BindingDB Entry DOI: 10.7270/Q2D21X2G |
More data for this Ligand-Target Pair | |
Sodium-dependent noradrenaline transporter
(Homo sapiens (Human)) | BDBM50136493
(1-Methyl-4,9-dihydro-3H-beta-carboline | 1-methyl-...)Show InChI InChI=1S/C12H12N2/c1-8-12-10(6-7-13-8)9-4-2-3-5-11(9)14-12/h2-5,14H,6-7H2,1H3 | Reactome pathway KEGG
UniProtKB/SwissProt UniProtKB/TrEMBL
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CHEMBL PC cid PC sid UniChem
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| >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Virginia Commonwealth University
Curated by ChEMBL
| Assay Description Binding affinity towards NET |
Bioorg Med Chem Lett 13: 4421-5 (2003)
BindingDB Entry DOI: 10.7270/Q2D21X2G |
More data for this Ligand-Target Pair | |
5-hydroxytryptamine receptor 1B
(Homo sapiens (Human)) | BDBM50136493
(1-Methyl-4,9-dihydro-3H-beta-carboline | 1-methyl-...)Show InChI InChI=1S/C12H12N2/c1-8-12-10(6-7-13-8)9-4-2-3-5-11(9)14-12/h2-5,14H,6-7H2,1H3 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt UniProtKB/TrEMBL
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CHEMBL PC cid PC sid UniChem
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| >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Virginia Commonwealth University
Curated by ChEMBL
| Assay Description Binding affinity towards 5-hydroxytryptamine 1B receptor |
Bioorg Med Chem Lett 13: 4421-5 (2003)
BindingDB Entry DOI: 10.7270/Q2D21X2G |
More data for this Ligand-Target Pair | |