null

SMILES: CCCCc1ccc(cc1)C(=O)Nc1cccc2cnccc12

InChI Key: InChIKey=FBFHYVLRXNNMSE-UHFFFAOYSA-N

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50376282   

Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50/IC50 nM	koff s-1	kon M-1s-1	pH	Temp °C
Transient receptor potential cation channel subfamily V member 1 (Homo sapiens (Human))	BDBM50376282 (CHEMBL407762) Show SMILES CCCCc1ccc(cc1)C(=O)Nc1cccc2cnccc12 Show InChI InChI=1S/C20H20N2O/c1-2-3-5-15-8-10-16(11-9-15)20(23)22-19-7-4-6-17-14-21-13-12-18(17)19/h4,6-14H,2-3,5H2,1H3,(H,22,23)	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	72	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Johnson& Johnson Pharmaceutical Research and Development Curated by ChEMBL					Assay Description Displacement of [3H]RTX from human TRPV1 receptor expressed in HEK293 cells				Bioorg Med Chem Lett 18: 2730-4 (2008) Article DOI: 10.1016/j.bmcl.2008.02.075 BindingDB Entry DOI: 10.7270/Q27H1KF6
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily V member 1 (Homo sapiens (Human))	BDBM50376282 (CHEMBL407762) Show SMILES CCCCc1ccc(cc1)C(=O)Nc1cccc2cnccc12 Show InChI InChI=1S/C20H20N2O/c1-2-3-5-15-8-10-16(11-9-15)20(23)22-19-7-4-6-17-14-21-13-12-18(17)19/h4,6-14H,2-3,5H2,1H3,(H,22,23)	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	2.40E+3	n/a	n/a	n/a	n/a	n/a	n/a
Johnson& Johnson Pharmaceutical Research and Development Curated by ChEMBL					Assay Description Activity at human TRPV1 in HEK cells assessed by measuring capsaicin-induced calcium level by FLIPR technology				Bioorg Med Chem Lett 18: 2730-4 (2008) Article DOI: 10.1016/j.bmcl.2008.02.075 BindingDB Entry DOI: 10.7270/Q27H1KF6
					More data for this Ligand-Target Pair