Found 6 hits for monomerid = 50421512 Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
Alpha-1D adrenergic receptor
(Homo sapiens (Human)) | BDBM50421512
(CHEMBL95523)Show InChI InChI=1S/C12H16N4O/c1-13-12(17)9-4-2-3-5-10(9)16-8-11-14-6-7-15-11/h2-5,16H,6-8H2,1H3,(H,13,17)(H,14,15) | Reactome pathway KEGG
UniProtKB/SwissProt UniProtKB/TrEMBL
DrugBank antibodypedia GoogleScholar AffyNet
| CHEMBL PC cid PC sid UniChem
Similars
| PubMed
| n/a | n/a | 89 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline
Curated by ChEMBL
| Assay Description Concentration required for 50% inhibition of binding against human Alpha-1D adrenergic receptor |
Bioorg Med Chem Lett 11: 2871-4 (2001)
BindingDB Entry DOI: 10.7270/Q2CC1201 |
More data for this Ligand-Target Pair | |
Alpha-1A adrenergic receptor
(Homo sapiens (Human)) | BDBM50421512
(CHEMBL95523)Show InChI InChI=1S/C12H16N4O/c1-13-12(17)9-4-2-3-5-10(9)16-8-11-14-6-7-15-11/h2-5,16H,6-8H2,1H3,(H,13,17)(H,14,15) | Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet
| CHEMBL PC cid PC sid UniChem
Similars
| PubMed
| n/a | n/a | 214 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline
Curated by ChEMBL
| Assay Description Concentration required for 50% inhibition of binding against Alpha-1A adrenergic receptor in human |
Bioorg Med Chem Lett 11: 2871-4 (2001)
BindingDB Entry DOI: 10.7270/Q2CC1201 |
More data for this Ligand-Target Pair | |
Alpha adrenergic receptor (1a and 1d)
(Homo sapiens (Human)) | BDBM50421512
(CHEMBL95523)Show InChI InChI=1S/C12H16N4O/c1-13-12(17)9-4-2-3-5-10(9)16-8-11-14-6-7-15-11/h2-5,16H,6-8H2,1H3,(H,13,17)(H,14,15) | Reactome pathway KEGG
UniProtKB/SwissProt UniProtKB/TrEMBL
DrugBank antibodypedia GoogleScholar AffyNet
| CHEMBL PC cid PC sid UniChem
Similars
| PubMed
| n/a | n/a | n/a | n/a | 10 | n/a | n/a | n/a | n/a |
GlaxoSmithKline
Curated by ChEMBL
| Assay Description Potency against cloned human alpha 1D-adrenoceptor expressed in rat-1 fibroblasts. |
Bioorg Med Chem Lett 11: 2871-4 (2001)
BindingDB Entry DOI: 10.7270/Q2CC1201 |
More data for this Ligand-Target Pair | |
Adrenergic receptor alpha
(Homo sapiens (Human)) | BDBM50421512
(CHEMBL95523)Show InChI InChI=1S/C12H16N4O/c1-13-12(17)9-4-2-3-5-10(9)16-8-11-14-6-7-15-11/h2-5,16H,6-8H2,1H3,(H,13,17)(H,14,15) | UniProtKB/SwissProt
antibodypedia GoogleScholar AffyNet
| CHEMBL PC cid PC sid UniChem
Similars
| PubMed
| n/a | n/a | n/a | n/a | 1.60 | n/a | n/a | n/a | n/a |
GlaxoSmithKline
Curated by ChEMBL
| Assay Description Potency against cloned human alpha 1B adrenoceptor expressed in rat-1 fibroblasts. |
Bioorg Med Chem Lett 11: 2871-4 (2001)
BindingDB Entry DOI: 10.7270/Q2CC1201 |
More data for this Ligand-Target Pair | |
Alpha-1A adrenergic receptor
(Homo sapiens (Human)) | BDBM50421512
(CHEMBL95523)Show InChI InChI=1S/C12H16N4O/c1-13-12(17)9-4-2-3-5-10(9)16-8-11-14-6-7-15-11/h2-5,16H,6-8H2,1H3,(H,13,17)(H,14,15) | Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet
| CHEMBL PC cid PC sid UniChem
Similars
| PubMed
| n/a | n/a | n/a | n/a | 2.5 | n/a | n/a | n/a | n/a |
GlaxoSmithKline
Curated by ChEMBL
| Assay Description Agonist potency against cloned human alpha 1A adrenoceptor expressed in rat-1 fibroblasts. |
Bioorg Med Chem Lett 11: 2871-4 (2001)
BindingDB Entry DOI: 10.7270/Q2CC1201 |
More data for this Ligand-Target Pair | |
Adrenergic alpha1B
(Homo sapiens (Human)) | BDBM50421512
(CHEMBL95523)Show InChI InChI=1S/C12H16N4O/c1-13-12(17)9-4-2-3-5-10(9)16-8-11-14-6-7-15-11/h2-5,16H,6-8H2,1H3,(H,13,17)(H,14,15) | UniProtKB/SwissProt
antibodypedia GoogleScholar AffyNet
| CHEMBL PC cid PC sid UniChem
Similars
| PubMed
| n/a | n/a | 692 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline
Curated by ChEMBL
| Assay Description Concentration required for 50% inhibition of binding against human Alpha-1B adrenergic receptor |
Bioorg Med Chem Lett 11: 2871-4 (2001)
BindingDB Entry DOI: 10.7270/Q2CC1201 |
More data for this Ligand-Target Pair | |