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BDBM50471520 CHEMBL117691

SMILES:

InChI Key: InChIKey=GNYILBXSHNUBSS-AATRIKPKSA-M

Data: 1 KI

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Similarity at least:  must be >=0.5
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50471520   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kcal/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Glutamate receptor ionotropic, NMDA 1


(RAT)
BDBM50471520
PNG
(CHEMBL117691)
Show InChI InChI=1S/C19H14Cl2N4O4/c20-9-7-13(21)16-12(17(18(27)28)25-14(16)8-9)5-6-15(26)23-10-1-3-11(4-2-10)24-19(22)29/h1-8,25H,(H,23,26)(H,27,28)(H3,22,24,29)/p-1/b6-5+
PDB

UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
1.60n/an/an/an/an/an/an/an/a



Glaxo Wellcome S.p.A.

Curated by ChEMBL


Assay Description
Inhibition of [3H]glycine to glycine binding site, associated with the N-methyl-D-aspartate glutamate receptor 1 in crude synaptic membranes prepared...


J Med Chem 40: 841-50 (1997)


Article DOI: 10.1021/jm960644a
BindingDB Entry DOI: 10.7270/Q2DJ5JBV
More data for this
Ligand-Target Pair