BDBM50479455 CHEMBL492668
SMILES: CN(C)CCNC(=O)c1cc2ccccc2cc1O
InChI Key: InChIKey=PTYBNDTVHWXPPT-UHFFFAOYSA-N
Data: 1 KI
Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
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Voltage-dependent L-type calcium channel subunit alpha-1S (Rattus norvegicus) | BDBM50479455 (CHEMBL492668) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase PC cid PC sid UniChem | Article PubMed | 450 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Perugia Curated by ChEMBL | Assay Description Displacement of [3H]diltiazem from L-type calcium channel in Sprague-Dawley rat cardiac myocytes | J Med Chem 51: 5552-65 (2008) Article DOI: 10.1021/jm800151n BindingDB Entry DOI: 10.7270/Q24T6N5H | |||||||||||
More data for this Ligand-Target Pair |