null

SMILES: Cn1ncc2c(NC(=O)NCc3cc(nn3-c3ccc(F)cc3)C(F)(F)F)cccc12

InChI Key:

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50553848   

Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50/IC50 nM	koff s-1	kon M-1s-1	pH	Temp °C
Transient receptor potential cation channel subfamily V member 1 (Homo sapiens (Human))	BDBM50553848 (CHEMBL4751349) Show SMILES Cn1ncc2c(NC(=O)NCc3cc(nn3-c3ccc(F)cc3)C(F)(F)F)cccc12 Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	8.40	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Antagonist activity at human TRPV1 expressed in CHO-K1 cells assessed as inhibition of capsaicin-induced Ca2+ response treated with compound 6 mins p...				Citation and Details Article DOI: 10.1016/j.bmcl.2020.127548 BindingDB Entry DOI: 10.7270/Q2VD733R
					More data for this Ligand-Target Pair