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SMILES: Cc1nn(C)cc1-c1ccc(OC2CC3(C2)CCN(CC2CCOCC2)CC3)nn1

InChI Key:

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 521067   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kcal/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Muscarinic acetylcholine receptor M4


(Homo sapiens (Human))		BDBM521067
PNG
(2-[6-(1,3-dimethylpyrazol-4-yl)pyridazin-3- yl]oxy...)
Show SMILES Cc1nn(C)cc1-c1ccc(OC2CC3(C2)CCN(CC2CCOCC2)CC3)nn1
PDB

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PC cid
PC sid
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US Patent
n/an/a 4.43E+3n/an/an/an/an/an/a


TBA

Assay Description
For high throughput measurement of agonist-evoked increases in intracellular calcium, CHO-K1 cells stably expressing muscarinic receptors were plated...

Citation and Details

BindingDB Entry DOI: 10.7270/Q2XD14VC
More data for this
Ligand-Target Pair