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SMILES: [H][C@]12CC[C@]([H])([C@@H](O)C1)[C@H](N2)C(=O)N1CC2(C1)CN(C2)c1c(cnc2sc(CC(F)(F)F)cc12)C(F)(F)F
InChI Key:
Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Histone-lysine N-methyltransferase 2A/Menin (Homo sapiens (Human)) | BDBM554120 (US11325921, Example 7) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 248 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Test for Evaluating the Inbinition of the Menin-MLL BindingMenin1-615 wherein 6× His tag and HA tag are inserted in the N-terminus, and myc tag is in... | Citation and Details BindingDB Entry DOI: 10.7270/Q2K64N9C | |||||||||||
More data for this Ligand-Target Pair |