Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Transcriptional enhancer factor TEF-3 (Homo sapiens) | BDBM50547124 (CHEMBL242708 | NCI-0001009) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 2.60E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Reversible inhibition of CPM binding to nonacylated N-terminal His6-tagged human TEAD4 (217 to 434 residues) expressed in Escherichia coli BL21-Codon... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01275 BindingDB Entry DOI: 10.7270/Q2QN6BC1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcriptional enhancer factor TEF-3 (Homo sapiens) | BDBM50547126 (CHEMBL4763473) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | Article PubMed | 1.04E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of CPM binding to N-terminal His6-tagged human TEAD4 (217 to 434 residues) expressed in Escherichia coli BL21-CodonPlus (DE3)-RIPL cells p... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01275 BindingDB Entry DOI: 10.7270/Q2QN6BC1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcriptional enhancer factor TEF-3 (Homo sapiens) | BDBM50547124 (CHEMBL242708 | NCI-0001009) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 70 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Binding affinity to nonacylated N-terminal His6-tagged human TEAD4 (217 to 434 residues) expressed in Escherichia coli BL21-CodonPlus (DE3)-RIPL cell... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01275 BindingDB Entry DOI: 10.7270/Q2QN6BC1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcriptional enhancer factor TEF-3 (Homo sapiens) | BDBM50547134 (CHEMBL4787565) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 100 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of FITC-labeled palmitate tracer binding to N-terminal His6-tagged human TEAD4 (217 to 434 residues) expressed in Escherichia coli BL21-Co... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01275 BindingDB Entry DOI: 10.7270/Q2QN6BC1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcriptional enhancer factor TEF-3 (Homo sapiens) | BDBM50547124 (CHEMBL242708 | NCI-0001009) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 200 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of FITC-labeled palmitate tracer binding to N-terminal His6-tagged human TEAD4 (217 to 434 residues) expressed in Escherichia coli BL21-Co... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01275 BindingDB Entry DOI: 10.7270/Q2QN6BC1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcriptional enhancer factor TEF-3 (Homo sapiens) | BDBM50547154 (CHEMBL4745831) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 200 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of FITC-labeled palmitate tracer binding to N-terminal His6-tagged human TEAD4 (217 to 434 residues) expressed in Escherichia coli BL21-Co... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01275 BindingDB Entry DOI: 10.7270/Q2QN6BC1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcriptional enhancer factor TEF-3 (Homo sapiens) | BDBM50547135 (CHEMBL4776143) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 200 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of FITC-labeled palmitate tracer binding to N-terminal His6-tagged human TEAD4 (217 to 434 residues) expressed in Escherichia coli BL21-Co... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01275 BindingDB Entry DOI: 10.7270/Q2QN6BC1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcriptional enhancer factor TEF-3 (Homo sapiens) | BDBM50547146 (CHEMBL4745853) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 200 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of FITC-labeled palmitate tracer binding to N-terminal His6-tagged human TEAD4 (217 to 434 residues) expressed in Escherichia coli BL21-Co... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01275 BindingDB Entry DOI: 10.7270/Q2QN6BC1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcriptional enhancer factor TEF-3 (Homo sapiens) | BDBM50547136 (CHEMBL4757924) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 200 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of FITC-labeled palmitate tracer binding to N-terminal His6-tagged human TEAD4 (217 to 434 residues) expressed in Escherichia coli BL21-Co... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01275 BindingDB Entry DOI: 10.7270/Q2QN6BC1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcriptional enhancer factor TEF-3 (Homo sapiens) | BDBM50547142 (CHEMBL4757369) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 200 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of FITC-labeled palmitate tracer binding to N-terminal His6-tagged human TEAD4 (217 to 434 residues) expressed in Escherichia coli BL21-Co... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01275 BindingDB Entry DOI: 10.7270/Q2QN6BC1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcriptional enhancer factor TEF-3 (Homo sapiens) | BDBM50547143 (CHEMBL4789889) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 300 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of FITC-labeled palmitate tracer binding to N-terminal His6-tagged human TEAD4 (217 to 434 residues) expressed in Escherichia coli BL21-Co... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01275 BindingDB Entry DOI: 10.7270/Q2QN6BC1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcriptional enhancer factor TEF-3 (Homo sapiens) | BDBM50547148 (CHEMBL4797833) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 300 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of FITC-labeled palmitate tracer binding to N-terminal His6-tagged human TEAD4 (217 to 434 residues) expressed in Escherichia coli BL21-Co... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01275 BindingDB Entry DOI: 10.7270/Q2QN6BC1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcriptional enhancer factor TEF-3 (Homo sapiens) | BDBM50547130 (CHEMBL1701986) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 300 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of FITC-labeled palmitate tracer binding to N-terminal His6-tagged human TEAD4 (217 to 434 residues) expressed in Escherichia coli BL21-Co... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01275 BindingDB Entry DOI: 10.7270/Q2QN6BC1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcriptional enhancer factor TEF-3 (Homo sapiens) | BDBM50547156 (CHEMBL4783341) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 300 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of FITC-labeled palmitate tracer binding to N-terminal His6-tagged human TEAD4 (217 to 434 residues) expressed in Escherichia coli BL21-Co... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01275 BindingDB Entry DOI: 10.7270/Q2QN6BC1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcriptional enhancer factor TEF-3 (Homo sapiens) | BDBM50547155 (CHEMBL4744235) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 300 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of FITC-labeled palmitate tracer binding to N-terminal His6-tagged human TEAD4 (217 to 434 residues) expressed in Escherichia coli BL21-Co... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01275 BindingDB Entry DOI: 10.7270/Q2QN6BC1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcriptional enhancer factor TEF-3 (Homo sapiens) | BDBM50547152 (CHEMBL4750726) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 300 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of FITC-labeled palmitate tracer binding to N-terminal His6-tagged human TEAD4 (217 to 434 residues) expressed in Escherichia coli BL21-Co... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01275 BindingDB Entry DOI: 10.7270/Q2QN6BC1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcriptional enhancer factor TEF-3 (Homo sapiens) | BDBM50547145 (CHEMBL4750624) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 400 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of FITC-labeled palmitate tracer binding to N-terminal His6-tagged human TEAD4 (217 to 434 residues) expressed in Escherichia coli BL21-Co... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01275 BindingDB Entry DOI: 10.7270/Q2QN6BC1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcriptional enhancer factor TEF-3 (Homo sapiens) | BDBM50547131 (CHEMBL4800702) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 400 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of FITC-labeled palmitate tracer binding to N-terminal His6-tagged human TEAD4 (217 to 434 residues) expressed in Escherichia coli BL21-Co... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01275 BindingDB Entry DOI: 10.7270/Q2QN6BC1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcriptional enhancer factor TEF-3 (Homo sapiens) | BDBM50547133 (CHEMBL4757939) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 500 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of FITC-labeled palmitate tracer binding to N-terminal His6-tagged human TEAD4 (217 to 434 residues) expressed in Escherichia coli BL21-Co... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01275 BindingDB Entry DOI: 10.7270/Q2QN6BC1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcriptional enhancer factor TEF-3 (Homo sapiens) | BDBM50547134 (CHEMBL4787565) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 700 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of CPM binding to N-terminal His6-tagged human TEAD4 (217 to 434 residues) expressed in Escherichia coli BL21-CodonPlus (DE3)-RIPL cells p... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01275 BindingDB Entry DOI: 10.7270/Q2QN6BC1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcriptional enhancer factor TEF-3 (Homo sapiens) | BDBM50547126 (CHEMBL4763473) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | 800 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of CPM binding to N-terminal His6-tagged human TEAD4 (217 to 434 residues) expressed in Escherichia coli BL21-CodonPlus (DE3)-RIPL cells p... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01275 BindingDB Entry DOI: 10.7270/Q2QN6BC1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcriptional enhancer factor TEF-3 (Homo sapiens) | BDBM50547125 (CHEMBL4784286) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 900 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of FITC-labeled palmitate tracer binding to N-terminal His6-tagged human TEAD4 (217 to 434 residues) expressed in Escherichia coli BL21-Co... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01275 BindingDB Entry DOI: 10.7270/Q2QN6BC1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcriptional enhancer factor TEF-3 (Homo sapiens) | BDBM50547136 (CHEMBL4757924) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of CPM binding to N-terminal His6-tagged human TEAD4 (217 to 434 residues) expressed in Escherichia coli BL21-CodonPlus (DE3)-RIPL cells p... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01275 BindingDB Entry DOI: 10.7270/Q2QN6BC1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcriptional enhancer factor TEF-3 (Homo sapiens) | BDBM50547132 (CHEMBL4797545) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of FITC-labeled palmitate tracer binding to N-terminal His6-tagged human TEAD4 (217 to 434 residues) expressed in Escherichia coli BL21-Co... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01275 BindingDB Entry DOI: 10.7270/Q2QN6BC1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcriptional enhancer factor TEF-3 (Homo sapiens) | BDBM50547135 (CHEMBL4776143) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of CPM binding to N-terminal His6-tagged human TEAD4 (217 to 434 residues) expressed in Escherichia coli BL21-CodonPlus (DE3)-RIPL cells p... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01275 BindingDB Entry DOI: 10.7270/Q2QN6BC1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcriptional enhancer factor TEF-3 (Homo sapiens) | BDBM50547146 (CHEMBL4745853) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.20E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of CPM binding to N-terminal His6-tagged human TEAD4 (217 to 434 residues) expressed in Escherichia coli BL21-CodonPlus (DE3)-RIPL cells p... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01275 BindingDB Entry DOI: 10.7270/Q2QN6BC1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcriptional enhancer factor TEF-3 (Homo sapiens) | BDBM50547142 (CHEMBL4757369) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of CPM binding to N-terminal His6-tagged human TEAD4 (217 to 434 residues) expressed in Escherichia coli BL21-CodonPlus (DE3)-RIPL cells p... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01275 BindingDB Entry DOI: 10.7270/Q2QN6BC1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcriptional enhancer factor TEF-3 (Homo sapiens) | BDBM50547154 (CHEMBL4745831) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of CPM binding to N-terminal His6-tagged human TEAD4 (217 to 434 residues) expressed in Escherichia coli BL21-CodonPlus (DE3)-RIPL cells p... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01275 BindingDB Entry DOI: 10.7270/Q2QN6BC1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcriptional enhancer factor TEF-3 (Homo sapiens) | BDBM50547144 (CHEMBL4778316) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of FITC-labeled palmitate tracer binding to N-terminal His6-tagged human TEAD4 (217 to 434 residues) expressed in Escherichia coli BL21-Co... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01275 BindingDB Entry DOI: 10.7270/Q2QN6BC1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcriptional enhancer factor TEF-3 (Homo sapiens) | BDBM50547148 (CHEMBL4797833) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of CPM binding to N-terminal His6-tagged human TEAD4 (217 to 434 residues) expressed in Escherichia coli BL21-CodonPlus (DE3)-RIPL cells p... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01275 BindingDB Entry DOI: 10.7270/Q2QN6BC1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcriptional enhancer factor TEF-3 (Homo sapiens) | BDBM50547152 (CHEMBL4750726) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.70E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of CPM binding to N-terminal His6-tagged human TEAD4 (217 to 434 residues) expressed in Escherichia coli BL21-CodonPlus (DE3)-RIPL cells p... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01275 BindingDB Entry DOI: 10.7270/Q2QN6BC1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcriptional enhancer factor TEF-3 (Homo sapiens) | BDBM50547143 (CHEMBL4789889) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.90E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of CPM binding to N-terminal His6-tagged human TEAD4 (217 to 434 residues) expressed in Escherichia coli BL21-CodonPlus (DE3)-RIPL cells p... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01275 BindingDB Entry DOI: 10.7270/Q2QN6BC1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcriptional enhancer factor TEF-3 (Homo sapiens) | BDBM50547124 (CHEMBL242708 | NCI-0001009) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 2.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of CPM binding to N-terminal His6-tagged human TEAD4 (217 to 434 residues) expressed in Escherichia coli BL21-CodonPlus (DE3)-RIPL cells p... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01275 BindingDB Entry DOI: 10.7270/Q2QN6BC1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcriptional enhancer factor TEF-3 (Homo sapiens) | BDBM50547156 (CHEMBL4783341) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 2.40E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of CPM binding to N-terminal His6-tagged human TEAD4 (217 to 434 residues) expressed in Escherichia coli BL21-CodonPlus (DE3)-RIPL cells p... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01275 BindingDB Entry DOI: 10.7270/Q2QN6BC1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcriptional enhancer factor TEF-4 (Homo sapiens) | BDBM50547124 (CHEMBL242708 | NCI-0001009) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 2.60E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of CPM binding to nonacylated N-terminal His6-tagged human TEAD2 (217 to 447 residues) expressed in Escherichia coli BL21-CodonPlus (DE3)-... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01275 BindingDB Entry DOI: 10.7270/Q2QN6BC1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcriptional enhancer factor TEF-5 (Homo sapiens) | BDBM50547124 (CHEMBL242708 | NCI-0001009) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 2.60E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of CPM binding to N-terminal His6-tagged human TEAD3 (216 to 434 residues) expressed in Escherichia coli BL21-CodonPlus (DE3)-RIPL cells p... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01275 BindingDB Entry DOI: 10.7270/Q2QN6BC1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcriptional enhancer factor TEF-1 (Homo sapiens) | BDBM50547124 (CHEMBL242708 | NCI-0001009) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 2.60E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of CPM binding to nonacylated N-terminal His6/GST-tagged human TEAD1 (209 to 426 residues) expressed in Escherichia coli BL21-CodonPlus (D... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01275 BindingDB Entry DOI: 10.7270/Q2QN6BC1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcriptional enhancer factor TEF-3 (Homo sapiens) | BDBM50547155 (CHEMBL4744235) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of CPM binding to N-terminal His6-tagged human TEAD4 (217 to 434 residues) expressed in Escherichia coli BL21-CodonPlus (DE3)-RIPL cells p... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01275 BindingDB Entry DOI: 10.7270/Q2QN6BC1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcriptional enhancer factor TEF-3 (Homo sapiens) | BDBM50547130 (CHEMBL1701986) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.20E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of CPM binding to N-terminal His6-tagged human TEAD4 (217 to 434 residues) expressed in Escherichia coli BL21-CodonPlus (DE3)-RIPL cells p... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01275 BindingDB Entry DOI: 10.7270/Q2QN6BC1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcriptional enhancer factor TEF-3 (Homo sapiens) | BDBM50547130 (CHEMBL1701986) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.20E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of CPM binding to N-terminal His6-tagged human TEAD4 (217 to 434 residues) expressed in Escherichia coli BL21-CodonPlus (DE3)-RIPL cells p... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01275 BindingDB Entry DOI: 10.7270/Q2QN6BC1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcriptional enhancer factor TEF-3 (Homo sapiens) | BDBM50547131 (CHEMBL4800702) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.70E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of CPM binding to N-terminal His6-tagged human TEAD4 (217 to 434 residues) expressed in Escherichia coli BL21-CodonPlus (DE3)-RIPL cells p... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01275 BindingDB Entry DOI: 10.7270/Q2QN6BC1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcriptional enhancer factor TEF-3 (Homo sapiens) | BDBM50547145 (CHEMBL4750624) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 4.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of CPM binding to N-terminal His6-tagged human TEAD4 (217 to 434 residues) expressed in Escherichia coli BL21-CodonPlus (DE3)-RIPL cells p... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01275 BindingDB Entry DOI: 10.7270/Q2QN6BC1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Catenin beta-1 (Homo sapiens (Human)) | BDBM50436054 (CHEMBL2397077) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 5.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Chemical Genomics Centre of the Max Planck Society Curated by ChEMBL | Assay Description Inhibition of beta-catenin-mediated transcriptional activity in Wnt3a-stimulated human HeLa cells after 24 hrs by Dual-Glo luciferase reporter gene a... | Bioorg Med Chem 21: 4020-6 (2013) Article DOI: 10.1016/j.bmc.2013.02.050 BindingDB Entry DOI: 10.7270/Q2BP046Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Catenin beta-1 (Homo sapiens (Human)) | BDBM50436055 (CHEMBL2397076) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 5.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Chemical Genomics Centre of the Max Planck Society Curated by ChEMBL | Assay Description Inhibition of beta-catenin-mediated transcriptional activity in Wnt3a-stimulated human HeLa cells after 24 hrs by Dual-Glo luciferase reporter gene a... | Bioorg Med Chem 21: 4020-6 (2013) Article DOI: 10.1016/j.bmc.2013.02.050 BindingDB Entry DOI: 10.7270/Q2BP046Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcriptional enhancer factor TEF-3 (Homo sapiens) | BDBM50547153 (CHEMBL4751604) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 5.60E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of FITC-labeled palmitate tracer binding to N-terminal His6-tagged human TEAD4 (217 to 434 residues) expressed in Escherichia coli BL21-Co... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01275 BindingDB Entry DOI: 10.7270/Q2QN6BC1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcriptional enhancer factor TEF-3 (Homo sapiens) | BDBM85507 (CAS_4394-00-7 | NSC_4488 | Niflumic acid | Niflumi...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase DrugBank MCE KEGG MMDB PC cid PC sid PDB UniChem Patents | Article PubMed | n/a | n/a | 5.90E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of FITC-labeled palmitate tracer binding to N-terminal His6-tagged human TEAD4 (217 to 434 residues) expressed in Escherichia coli BL21-Co... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01275 BindingDB Entry DOI: 10.7270/Q2QN6BC1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcriptional enhancer factor TEF-3 (Homo sapiens) | BDBM50547151 (CHEMBL4781890) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 6.40E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of FITC-labeled palmitate tracer binding to N-terminal His6-tagged human TEAD4 (217 to 434 residues) expressed in Escherichia coli BL21-Co... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01275 BindingDB Entry DOI: 10.7270/Q2QN6BC1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcriptional enhancer factor TEF-3 (Homo sapiens) | BDBM50547137 (CHEMBL4750499) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 8.70E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of CPM binding to N-terminal His6-tagged human TEAD4 (217 to 434 residues) expressed in Escherichia coli BL21-CodonPlus (DE3)-RIPL cells p... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01275 BindingDB Entry DOI: 10.7270/Q2QN6BC1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcriptional enhancer factor TEF-3 (Homo sapiens) | BDBM50547132 (CHEMBL4797545) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 9.20E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of CPM binding to N-terminal His6-tagged human TEAD4 (217 to 434 residues) expressed in Escherichia coli BL21-CodonPlus (DE3)-RIPL cells p... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01275 BindingDB Entry DOI: 10.7270/Q2QN6BC1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcriptional enhancer factor TEF-3 (Homo sapiens) | BDBM50547123 (CHEMBL4786804) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 9.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Binding affinity to nonacylated N-terminal His6-tagged human TEAD4 (217 to 434 residues) expressed in Escherichia coli BL21-CodonPlus (DE3)-RIPL cell... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01275 BindingDB Entry DOI: 10.7270/Q2QN6BC1 | |||||||||||
More data for this Ligand-Target Pair |
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