Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
D(3) dopamine receptor (Rattus norvegicus (Rat)) | BDBM50219939 (CHEMBL240693 | N-((1r,4r)-4-(2-(4-(2,3-dichlorophe...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.200 | n/a | n/a | n/a | n/a | n/a | n/a |
Gedeon Richter Ltd Curated by ChEMBL | Assay Description Displacement of [3H]spiperone from rat dopamine D3 receptor expressed in Sf9 cells | Bioorg Med Chem Lett 17: 5340-4 (2007) Article DOI: 10.1016/j.bmcl.2007.08.015 BindingDB Entry DOI: 10.7270/Q22F7N5G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(3) dopamine receptor (Rattus norvegicus (Rat)) | BDBM50219946 (CHEMBL391700 | N-((1r,4r)-4-(2-(4-(3-(trifluoromet...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.300 | n/a | n/a | n/a | n/a | n/a | n/a |
Gedeon Richter Ltd Curated by ChEMBL | Assay Description Displacement of [3H]spiperone from rat dopamine D3 receptor expressed in Sf9 cells | Bioorg Med Chem Lett 17: 5340-4 (2007) Article DOI: 10.1016/j.bmcl.2007.08.015 BindingDB Entry DOI: 10.7270/Q22F7N5G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(3) dopamine receptor (Rattus norvegicus (Rat)) | BDBM50219943 (CHEMBL428910 | N-((1r,4r)-4-(2-(4-(3-cyano-5-(trif...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.400 | n/a | n/a | n/a | n/a | n/a | n/a |
Gedeon Richter Ltd Curated by ChEMBL | Assay Description Displacement of [3H]spiperone from rat dopamine D3 receptor expressed in Sf9 cells | Bioorg Med Chem Lett 17: 5340-4 (2007) Article DOI: 10.1016/j.bmcl.2007.08.015 BindingDB Entry DOI: 10.7270/Q22F7N5G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(3) dopamine receptor (Rattus norvegicus (Rat)) | BDBM50219944 (CHEMBL239847 | N-((1r,4r)-4-(2-(4-(4-bromo-2-metho...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 0.5 | n/a | n/a | n/a | n/a | n/a | n/a |
Gedeon Richter Ltd Curated by ChEMBL | Assay Description Displacement of [3H]spiperone from rat dopamine D3 receptor expressed in Sf9 cells | Bioorg Med Chem Lett 17: 5340-4 (2007) Article DOI: 10.1016/j.bmcl.2007.08.015 BindingDB Entry DOI: 10.7270/Q22F7N5G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(3) dopamine receptor (Rattus norvegicus (Rat)) | BDBM50219940 (CHEMBL240271 | N-((1r,4r)-4-(2-(4-(3-(trifluoromet...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 0.5 | n/a | n/a | n/a | n/a | n/a | n/a |
Gedeon Richter Ltd Curated by ChEMBL | Assay Description Displacement of [3H]spiperone from rat dopamine D3 receptor expressed in Sf9 cells | Bioorg Med Chem Lett 17: 5340-4 (2007) Article DOI: 10.1016/j.bmcl.2007.08.015 BindingDB Entry DOI: 10.7270/Q22F7N5G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(3) dopamine receptor (Rattus norvegicus (Rat)) | BDBM50219945 (CHEMBL240273 | N-((1r,4r)-4-(2-(4-(3-cyano-5-(trif...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 0.700 | n/a | n/a | n/a | n/a | n/a | n/a |
Gedeon Richter Ltd Curated by ChEMBL | Assay Description Displacement of [3H]spiperone from rat dopamine D3 receptor expressed in Sf9 cells | Bioorg Med Chem Lett 17: 5340-4 (2007) Article DOI: 10.1016/j.bmcl.2007.08.015 BindingDB Entry DOI: 10.7270/Q22F7N5G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(3) dopamine receptor (Rattus norvegicus (Rat)) | BDBM50219947 (CHEMBL429093 | N-((1r,4r)-4-(2-(4-(3-cyanophenyl)p...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 0.700 | n/a | n/a | n/a | n/a | n/a | n/a |
Gedeon Richter Ltd Curated by ChEMBL | Assay Description Displacement of [3H]spiperone from rat dopamine D3 receptor expressed in Sf9 cells | Bioorg Med Chem Lett 17: 5340-4 (2007) Article DOI: 10.1016/j.bmcl.2007.08.015 BindingDB Entry DOI: 10.7270/Q22F7N5G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(3) dopamine receptor (Rattus norvegicus (Rat)) | BDBM50219935 (CHEMBL392528 | N-[4-(4-{2-[4-(3-cyano-5-trifluorom...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.900 | n/a | n/a | n/a | n/a | n/a | n/a |
Gedeon Richter Ltd Curated by ChEMBL | Assay Description Displacement of [3H]spiperone from rat dopamine D3 receptor expressed in Sf9 cells | Bioorg Med Chem Lett 17: 5340-4 (2007) Article DOI: 10.1016/j.bmcl.2007.08.015 BindingDB Entry DOI: 10.7270/Q22F7N5G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(3) dopamine receptor (Rattus norvegicus (Rat)) | BDBM50219949 (3-oxo-N-((1r,4r)-4-(2-(4-(3-(trifluoromethyl)pheno...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1 | n/a | n/a | n/a | n/a | n/a | n/a |
Gedeon Richter Ltd Curated by ChEMBL | Assay Description Displacement of [3H]spiperone from rat dopamine D3 receptor expressed in Sf9 cells | Bioorg Med Chem Lett 17: 5340-4 (2007) Article DOI: 10.1016/j.bmcl.2007.08.015 BindingDB Entry DOI: 10.7270/Q22F7N5G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 2B (Rattus norvegicus (Rat)) | BDBM50204883 ((6-hydroxy-1H-benzimidazol-2-yl)-(4-p-tolyloxy-pip...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.10 | n/a | n/a | n/a | n/a | n/a | n/a |
Gedeon Richter Ltd. Curated by ChEMBL | Assay Description Antagonist activity at NR2B NMDA receptor in Wistar rat neocortical cells assessed as inhibition of NMDA-evoked elevation of intracellular calcium co... | J Med Chem 50: 901-14 (2007) Article DOI: 10.1021/jm060420k BindingDB Entry DOI: 10.7270/Q2DV1JJ4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 2B (Rattus norvegicus (Rat)) | BDBM50204865 (CHEMBL220611 | [4-(4-fluoro-benzyl)-piperidin-1-yl...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.20 | n/a | n/a | n/a | n/a | n/a | n/a |
Gedeon Richter Ltd. Curated by ChEMBL | Assay Description Antagonist activity at NR2B NMDA receptor in Wistar rat neocortical cells assessed as inhibition of NMDA-evoked elevation of intracellular calcium co... | J Med Chem 50: 901-14 (2007) Article DOI: 10.1021/jm060420k BindingDB Entry DOI: 10.7270/Q2DV1JJ4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 2B (Rattus norvegicus (Rat)) | BDBM50204868 (CHEMBL424752 | N-[2-(4-benzyl-piperidin-1-carbonyl...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.30 | n/a | n/a | n/a | n/a | n/a | n/a |
Gedeon Richter Ltd. Curated by ChEMBL | Assay Description Antagonist activity at NR2B NMDA receptor in Wistar rat neocortical cells assessed as inhibition of NMDA-evoked elevation of intracellular calcium co... | J Med Chem 50: 901-14 (2007) Article DOI: 10.1021/jm060420k BindingDB Entry DOI: 10.7270/Q2DV1JJ4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 2B (Rattus norvegicus (Rat)) | BDBM50204882 (CHEMBL375615 | [4-(4-chloro-phenoxy)-piperidin-1-y...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.70 | n/a | n/a | n/a | n/a | n/a | n/a |
Gedeon Richter Ltd. Curated by ChEMBL | Assay Description Antagonist activity at NR2B NMDA receptor in Wistar rat neocortical cells assessed as inhibition of NMDA-evoked elevation of intracellular calcium co... | J Med Chem 50: 901-14 (2007) Article DOI: 10.1021/jm060420k BindingDB Entry DOI: 10.7270/Q2DV1JJ4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(3) dopamine receptor (Rattus norvegicus (Rat)) | BDBM50219942 (CHEMBL240051 | N-((1r,4r)-4-(2-(4-(2,5-dichlorophe...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 2 | n/a | n/a | n/a | n/a | n/a | n/a |
Gedeon Richter Ltd Curated by ChEMBL | Assay Description Displacement of [3H]spiperone from rat dopamine D3 receptor expressed in Sf9 cells | Bioorg Med Chem Lett 17: 5340-4 (2007) Article DOI: 10.1016/j.bmcl.2007.08.015 BindingDB Entry DOI: 10.7270/Q22F7N5G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 2B (Rattus norvegicus (Rat)) | BDBM50204899 ((4-benzylpiperidine-1-yl)-[5(6)-hydroxy-1H-benzimi...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.20 | n/a | n/a | n/a | n/a | n/a | n/a |
Gedeon Richter Ltd. Curated by ChEMBL | Assay Description Antagonist activity at NR2B NMDA receptor in Wistar rat neocortical cells assessed as inhibition of NMDA-evoked elevation of intracellular calcium co... | J Med Chem 50: 901-14 (2007) Article DOI: 10.1021/jm060420k BindingDB Entry DOI: 10.7270/Q2DV1JJ4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 2B (Rattus norvegicus (Rat)) | BDBM50204887 ((6-hydroxy-1H-benzimidazol-2-yl)-[4-(3-methyl-benz...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.40 | n/a | n/a | n/a | n/a | n/a | n/a |
Gedeon Richter Ltd. Curated by ChEMBL | Assay Description Antagonist activity at NR2B NMDA receptor in Wistar rat neocortical cells assessed as inhibition of NMDA-evoked elevation of intracellular calcium co... | J Med Chem 50: 901-14 (2007) Article DOI: 10.1021/jm060420k BindingDB Entry DOI: 10.7270/Q2DV1JJ4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 2B (Rattus norvegicus (Rat)) | BDBM50204861 ((6-hydroxy-1H-benzimidazol-2-yl)-[4-(3-methoxy-ben...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.5 | n/a | n/a | n/a | n/a | n/a | n/a |
Gedeon Richter Ltd. Curated by ChEMBL | Assay Description Antagonist activity at NR2B NMDA receptor in Wistar rat neocortical cells assessed as inhibition of NMDA-evoked elevation of intracellular calcium co... | J Med Chem 50: 901-14 (2007) Article DOI: 10.1021/jm060420k BindingDB Entry DOI: 10.7270/Q2DV1JJ4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(3) dopamine receptor (Rattus norvegicus (Rat)) | BDBM50219948 (CHEMBL236407 | N-((1r,4r)-4-(2-(4-(3-(trifluoromet...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 2.60 | n/a | n/a | n/a | n/a | n/a | n/a |
Gedeon Richter Ltd Curated by ChEMBL | Assay Description Displacement of [3H]spiperone from rat dopamine D3 receptor expressed in Sf9 cells | Bioorg Med Chem Lett 17: 5340-4 (2007) Article DOI: 10.1016/j.bmcl.2007.08.015 BindingDB Entry DOI: 10.7270/Q22F7N5G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(3) dopamine receptor (Rattus norvegicus (Rat)) | BDBM50219938 (CHEMBL391699 | N-((1r,4r)-4-(2-(4-(3-(trifluoromet...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 2.80 | n/a | n/a | n/a | n/a | n/a | n/a |
Gedeon Richter Ltd Curated by ChEMBL | Assay Description Displacement of [3H]spiperone from rat dopamine D3 receptor expressed in Sf9 cells | Bioorg Med Chem Lett 17: 5340-4 (2007) Article DOI: 10.1016/j.bmcl.2007.08.015 BindingDB Entry DOI: 10.7270/Q22F7N5G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 2B (Rattus norvegicus (Rat)) | BDBM50204864 (CHEMBL220474 | [4-(4-fluoro-phenoxy)-piperidin-1-y...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.90 | n/a | n/a | n/a | n/a | n/a | n/a |
Gedeon Richter Ltd. Curated by ChEMBL | Assay Description Antagonist activity at NR2B NMDA receptor in Wistar rat neocortical cells assessed as inhibition of NMDA-evoked elevation of intracellular calcium co... | J Med Chem 50: 901-14 (2007) Article DOI: 10.1021/jm060420k BindingDB Entry DOI: 10.7270/Q2DV1JJ4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 2B (Rattus norvegicus (Rat)) | BDBM50204861 ((6-hydroxy-1H-benzimidazol-2-yl)-[4-(3-methoxy-ben...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3 | n/a | n/a | n/a | n/a | n/a | n/a |
Gedeon Richter Ltd. Curated by ChEMBL | Assay Description Displacement of [3H]Ro 25,6981 from NR2B NMDA receptor in rat forebrain | J Med Chem 50: 901-14 (2007) Article DOI: 10.1021/jm060420k BindingDB Entry DOI: 10.7270/Q2DV1JJ4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 2B (Rattus norvegicus (Rat)) | BDBM50204863 ((4-benzyl-piperidin-1-yl)-[4(7)-hydroxy-1H-benzimi...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3 | n/a | n/a | n/a | n/a | n/a | n/a |
Gedeon Richter Ltd. Curated by ChEMBL | Assay Description Antagonist activity at NR2B NMDA receptor in Wistar rat neocortical cells assessed as inhibition of NMDA-evoked elevation of intracellular calcium co... | J Med Chem 50: 901-14 (2007) Article DOI: 10.1021/jm060420k BindingDB Entry DOI: 10.7270/Q2DV1JJ4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 2B (Rattus norvegicus (Rat)) | BDBM50204868 (CHEMBL424752 | N-[2-(4-benzyl-piperidin-1-carbonyl...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3 | n/a | n/a | n/a | n/a | n/a | n/a |
Gedeon Richter Ltd. Curated by ChEMBL | Assay Description Displacement of [3H]Ro 25,6981 from NR2B NMDA receptor in rat forebrain | J Med Chem 50: 901-14 (2007) Article DOI: 10.1021/jm060420k BindingDB Entry DOI: 10.7270/Q2DV1JJ4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 2B (Rattus norvegicus (Rat)) | BDBM50204883 ((6-hydroxy-1H-benzimidazol-2-yl)-(4-p-tolyloxy-pip...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3 | n/a | n/a | n/a | n/a | n/a | n/a |
Gedeon Richter Ltd. Curated by ChEMBL | Assay Description Displacement of [3H]Ro 25,6981 from NR2B NMDA receptor in rat forebrain | J Med Chem 50: 901-14 (2007) Article DOI: 10.1021/jm060420k BindingDB Entry DOI: 10.7270/Q2DV1JJ4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(3) dopamine receptor (Rattus norvegicus (Rat)) | BDBM50219937 (4-chloro-N-((1r,4r)-4-(2-(4-(3-(trifluoromethyl)ph...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3 | n/a | n/a | n/a | n/a | n/a | n/a |
Gedeon Richter Ltd Curated by ChEMBL | Assay Description Displacement of [3H]spiperone from rat dopamine D3 receptor expressed in Sf9 cells | Bioorg Med Chem Lett 17: 5340-4 (2007) Article DOI: 10.1016/j.bmcl.2007.08.015 BindingDB Entry DOI: 10.7270/Q22F7N5G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(3) dopamine receptor (Rattus norvegicus (Rat)) | BDBM50219936 (4-bromo-N-((1r,4r)-4-(2-(4-(3-cyano-5-(trifluorome...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.30 | n/a | n/a | n/a | n/a | n/a | n/a |
Gedeon Richter Ltd Curated by ChEMBL | Assay Description Displacement of [3H]spiperone from rat dopamine D3 receptor expressed in Sf9 cells | Bioorg Med Chem Lett 17: 5340-4 (2007) Article DOI: 10.1016/j.bmcl.2007.08.015 BindingDB Entry DOI: 10.7270/Q22F7N5G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 2B (Rattus norvegicus (Rat)) | BDBM50204862 (CHEMBL436521 | N-(2-((4-benzylpiperidin-1-yl)methy...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.5 | n/a | n/a | n/a | n/a | n/a | n/a |
Gedeon Richter Ltd. Curated by ChEMBL | Assay Description Displacement of [3H]Ro 25,6981 from NR2B NMDA receptor in rat forebrain | J Med Chem 50: 901-14 (2007) Article DOI: 10.1021/jm060420k BindingDB Entry DOI: 10.7270/Q2DV1JJ4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(3) dopamine receptor (Rattus norvegicus (Rat)) | BDBM50219934 (CHEMBL399833 | N-((1r,4r)-4-(2-(4-(3-(trifluoromet...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.80 | n/a | n/a | n/a | n/a | n/a | n/a |
Gedeon Richter Ltd Curated by ChEMBL | Assay Description Displacement of [3H]spiperone from rat dopamine D3 receptor expressed in Sf9 cells | Bioorg Med Chem Lett 17: 5340-4 (2007) Article DOI: 10.1016/j.bmcl.2007.08.015 BindingDB Entry DOI: 10.7270/Q22F7N5G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(2) dopamine receptor (Rattus norvegicus (rat)) | BDBM50219939 (CHEMBL240693 | N-((1r,4r)-4-(2-(4-(2,3-dichlorophe...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 4 | n/a | n/a | n/a | n/a | n/a | n/a |
Gedeon Richter Ltd Curated by ChEMBL | Assay Description Displacement of [3H]spiperone from dopamine D2 receptor in rat striatal membranes | Bioorg Med Chem Lett 17: 5340-4 (2007) Article DOI: 10.1016/j.bmcl.2007.08.015 BindingDB Entry DOI: 10.7270/Q22F7N5G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 2B (Rattus norvegicus (Rat)) | BDBM50204865 (CHEMBL220611 | [4-(4-fluoro-benzyl)-piperidin-1-yl...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 4 | n/a | n/a | n/a | n/a | n/a | n/a |
Gedeon Richter Ltd. Curated by ChEMBL | Assay Description Displacement of [3H]Ro 25,6981 from NR2B NMDA receptor in rat forebrain | J Med Chem 50: 901-14 (2007) Article DOI: 10.1021/jm060420k BindingDB Entry DOI: 10.7270/Q2DV1JJ4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 2B (Rattus norvegicus (Rat)) | BDBM50204884 (6-(2-(4-(4-fluorobenzyl)piperidin-1-yl)ethylsulfin...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Patents | Article PubMed | n/a | n/a | 4 | n/a | n/a | n/a | n/a | n/a | n/a |
Gedeon Richter Ltd. Curated by ChEMBL | Assay Description Displacement of [3H]Ro 25,6981 from NR2B NMDA receptor in rat forebrain | J Med Chem 50: 901-14 (2007) Article DOI: 10.1021/jm060420k BindingDB Entry DOI: 10.7270/Q2DV1JJ4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 2B (Rattus norvegicus (Rat)) | BDBM50204899 ((4-benzylpiperidine-1-yl)-[5(6)-hydroxy-1H-benzimi...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 4 | n/a | n/a | n/a | n/a | n/a | n/a |
Gedeon Richter Ltd. Curated by ChEMBL | Assay Description Displacement of [3H]Ro 25,6981 from NR2B NMDA receptor in rat forebrain | J Med Chem 50: 901-14 (2007) Article DOI: 10.1021/jm060420k BindingDB Entry DOI: 10.7270/Q2DV1JJ4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(3) dopamine receptor (Rattus norvegicus (Rat)) | BDBM50219941 (CHEMBL240909 | N-((1r,4r)-4-(2-(4-(3-cyano-5-(trif...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 4.20 | n/a | n/a | n/a | n/a | n/a | n/a |
Gedeon Richter Ltd Curated by ChEMBL | Assay Description Displacement of [3H]spiperone from rat dopamine D3 receptor expressed in Sf9 cells | Bioorg Med Chem Lett 17: 5340-4 (2007) Article DOI: 10.1016/j.bmcl.2007.08.015 BindingDB Entry DOI: 10.7270/Q22F7N5G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 2B (Rattus norvegicus (Rat)) | BDBM50204895 ((4-amino-1H-indol-2-yl)-(4-benzyl-piperidin-1-yl)-...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 4.30 | n/a | n/a | n/a | n/a | n/a | n/a |
Gedeon Richter Ltd. Curated by ChEMBL | Assay Description Antagonist activity at NR2B NMDA receptor in Wistar rat neocortical cells assessed as inhibition of NMDA-evoked elevation of intracellular calcium co... | J Med Chem 50: 901-14 (2007) Article DOI: 10.1021/jm060420k BindingDB Entry DOI: 10.7270/Q2DV1JJ4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(2) dopamine receptor (Rattus norvegicus (rat)) | BDBM50219940 (CHEMBL240271 | N-((1r,4r)-4-(2-(4-(3-(trifluoromet...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 4.30 | n/a | n/a | n/a | n/a | n/a | n/a |
Gedeon Richter Ltd Curated by ChEMBL | Assay Description Displacement of [3H]spiperone from dopamine D2 receptor in rat striatal membranes | Bioorg Med Chem Lett 17: 5340-4 (2007) Article DOI: 10.1016/j.bmcl.2007.08.015 BindingDB Entry DOI: 10.7270/Q22F7N5G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 2B (Rattus norvegicus (Rat)) | BDBM50204873 ((4-benzylpiperidin-1-yl)-(3,6-dihydro-pirrolo[3,2-...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 5 | n/a | n/a | n/a | n/a | n/a | n/a |
Gedeon Richter Ltd. Curated by ChEMBL | Assay Description Displacement of [3H]Ro 25,6981 from NR2B NMDA receptor in rat forebrain | J Med Chem 50: 901-14 (2007) Article DOI: 10.1021/jm060420k BindingDB Entry DOI: 10.7270/Q2DV1JJ4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 2B (Rattus norvegicus (Rat)) | BDBM50204887 ((6-hydroxy-1H-benzimidazol-2-yl)-[4-(3-methyl-benz...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 5 | n/a | n/a | n/a | n/a | n/a | n/a |
Gedeon Richter Ltd. Curated by ChEMBL | Assay Description Displacement of [3H]Ro 25,6981 from NR2B NMDA receptor in rat forebrain | J Med Chem 50: 901-14 (2007) Article DOI: 10.1021/jm060420k BindingDB Entry DOI: 10.7270/Q2DV1JJ4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(2) dopamine receptor (Rattus norvegicus (rat)) | BDBM50219949 (3-oxo-N-((1r,4r)-4-(2-(4-(3-(trifluoromethyl)pheno...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 5.30 | n/a | n/a | n/a | n/a | n/a | n/a |
Gedeon Richter Ltd Curated by ChEMBL | Assay Description Displacement of [3H]spiperone from dopamine D2 receptor in rat striatal membranes | Bioorg Med Chem Lett 17: 5340-4 (2007) Article DOI: 10.1016/j.bmcl.2007.08.015 BindingDB Entry DOI: 10.7270/Q22F7N5G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(3) dopamine receptor (Rattus norvegicus (Rat)) | BDBM50219950 (3-cyano-N-((1r,4r)-4-(2-(4-(3-cyano-5-(trifluorome...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 5.80 | n/a | n/a | n/a | n/a | n/a | n/a |
Gedeon Richter Ltd Curated by ChEMBL | Assay Description Displacement of [3H]spiperone from rat dopamine D3 receptor expressed in Sf9 cells | Bioorg Med Chem Lett 17: 5340-4 (2007) Article DOI: 10.1016/j.bmcl.2007.08.015 BindingDB Entry DOI: 10.7270/Q22F7N5G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 2B (Rattus norvegicus (Rat)) | BDBM50204891 ((4-benzylpiperidin-1-yl)-(3,6-dihydro-imidazo[4,5-...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 6 | n/a | n/a | n/a | n/a | n/a | n/a |
Gedeon Richter Ltd. Curated by ChEMBL | Assay Description Displacement of [3H]Ro 25,6981 from NR2B NMDA receptor in rat forebrain | J Med Chem 50: 901-14 (2007) Article DOI: 10.1021/jm060420k BindingDB Entry DOI: 10.7270/Q2DV1JJ4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 2B (Rattus norvegicus (Rat)) | BDBM50204864 (CHEMBL220474 | [4-(4-fluoro-phenoxy)-piperidin-1-y...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 6 | n/a | n/a | n/a | n/a | n/a | n/a |
Gedeon Richter Ltd. Curated by ChEMBL | Assay Description Displacement of [3H]Ro 25,6981 from NR2B NMDA receptor in rat forebrain | J Med Chem 50: 901-14 (2007) Article DOI: 10.1021/jm060420k BindingDB Entry DOI: 10.7270/Q2DV1JJ4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 2B (Rattus norvegicus (Rat)) | BDBM50134652 ((4-Benzyl-piperidin-1-yl)-(4,6-dihydroxy-1H-indol-...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 6 | n/a | n/a | n/a | n/a | n/a | n/a |
Gedeon Richter Ltd. Curated by ChEMBL | Assay Description Displacement of [3H]Ro 25,6981 from NR2B NMDA receptor in rat forebrain | J Med Chem 50: 901-14 (2007) Article DOI: 10.1021/jm060420k BindingDB Entry DOI: 10.7270/Q2DV1JJ4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 2B (Rattus norvegicus (Rat)) | BDBM50080029 (4-((1R,2S)-3-(4-benzylpiperidin-1-yl)-1-hydroxy-2-...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE MMDB PC cid PC sid PDB UniChem Patents Similars | PDB Article PubMed | n/a | n/a | 6 | n/a | n/a | n/a | n/a | n/a | n/a |
Gedeon Richter Ltd. Curated by ChEMBL | Assay Description Displacement of [3H]Ro 25,6981 from NR2B NMDA receptor in rat forebrain | J Med Chem 50: 901-14 (2007) Article DOI: 10.1021/jm060420k BindingDB Entry DOI: 10.7270/Q2DV1JJ4 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Glutamate receptor ionotropic, NMDA 2B (Rattus norvegicus (Rat)) | BDBM50134652 ((4-Benzyl-piperidin-1-yl)-(4,6-dihydroxy-1H-indol-...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 6.5 | n/a | n/a | n/a | n/a | n/a | n/a |
Gedeon Richter Ltd. Curated by ChEMBL | Assay Description Antagonist activity at NR2B NMDA receptor in Wistar rat neocortical cells assessed as inhibition of NMDA-evoked elevation of intracellular calcium co... | J Med Chem 50: 901-14 (2007) Article DOI: 10.1021/jm060420k BindingDB Entry DOI: 10.7270/Q2DV1JJ4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 2B (Rattus norvegicus (Rat)) | BDBM50204884 (6-(2-(4-(4-fluorobenzyl)piperidin-1-yl)ethylsulfin...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Patents | Article PubMed | n/a | n/a | 6.60 | n/a | n/a | n/a | n/a | n/a | n/a |
Gedeon Richter Ltd. Curated by ChEMBL | Assay Description Antagonist activity at NR2B NMDA receptor in Wistar rat neocortical cells assessed as inhibition of NMDA-evoked elevation of intracellular calcium co... | J Med Chem 50: 901-14 (2007) Article DOI: 10.1021/jm060420k BindingDB Entry DOI: 10.7270/Q2DV1JJ4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 2B (Rattus norvegicus (Rat)) | BDBM50134648 ((6-Hydroxy-1H-indol-2-yl)-(4-phenoxymethyl-piperid...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 7 | n/a | n/a | n/a | n/a | n/a | n/a |
Gedeon Richter Ltd. Curated by ChEMBL | Assay Description Displacement of [3H]Ro 25,6981 from NR2B NMDA receptor in rat forebrain | J Med Chem 50: 901-14 (2007) Article DOI: 10.1021/jm060420k BindingDB Entry DOI: 10.7270/Q2DV1JJ4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 2B (Rattus norvegicus (Rat)) | BDBM50032651 (1-((1S,2S)-1-hydroxy-1-(4-hydroxyphenyl)propan-2-y...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 7 | n/a | n/a | n/a | n/a | n/a | n/a |
Gedeon Richter Ltd. Curated by ChEMBL | Assay Description Displacement of [3H]Ro 25,6981 from NR2B NMDA receptor in rat forebrain | J Med Chem 50: 901-14 (2007) Article DOI: 10.1021/jm060420k BindingDB Entry DOI: 10.7270/Q2DV1JJ4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 2B (Rattus norvegicus (Rat)) | BDBM50204870 (2-[(4-benzyl-piperidin-1-yl)-imino-methyl]-1H-indo...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 8.5 | n/a | n/a | n/a | n/a | n/a | n/a |
Gedeon Richter Ltd. Curated by ChEMBL | Assay Description Antagonist activity at NR2B NMDA receptor in Wistar rat neocortical cells assessed as inhibition of NMDA-evoked elevation of intracellular calcium co... | J Med Chem 50: 901-14 (2007) Article DOI: 10.1021/jm060420k BindingDB Entry DOI: 10.7270/Q2DV1JJ4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 2B (Rattus norvegicus (Rat)) | BDBM50204862 (CHEMBL436521 | N-(2-((4-benzylpiperidin-1-yl)methy...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 8.60 | n/a | n/a | n/a | n/a | n/a | n/a |
Gedeon Richter Ltd. Curated by ChEMBL | Assay Description Antagonist activity at NR2B NMDA receptor in Wistar rat neocortical cells assessed as inhibition of NMDA-evoked elevation of intracellular calcium co... | J Med Chem 50: 901-14 (2007) Article DOI: 10.1021/jm060420k BindingDB Entry DOI: 10.7270/Q2DV1JJ4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(2) dopamine receptor (Rattus norvegicus (rat)) | BDBM50219942 (CHEMBL240051 | N-((1r,4r)-4-(2-(4-(2,5-dichlorophe...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 9 | n/a | n/a | n/a | n/a | n/a | n/a |
Gedeon Richter Ltd Curated by ChEMBL | Assay Description Displacement of [3H]spiperone from dopamine D2 receptor in rat striatal membranes | Bioorg Med Chem Lett 17: 5340-4 (2007) Article DOI: 10.1016/j.bmcl.2007.08.015 BindingDB Entry DOI: 10.7270/Q22F7N5G | |||||||||||
More data for this Ligand-Target Pair |
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