Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Proto-oncogene tyrosine-protein kinase Src (Homo sapiens (Human)) | BDBM50314074 (2,6,9-Trisubstitute purine, 6 (AP23464) | 3-(2-(2-...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MMDB PC cid PC sid PDB UniChem Patents Similars | Article PubMed | n/a | n/a | 0.450 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Lille Curated by ChEMBL | Assay Description Inhibition of Src | Eur J Med Chem 45: 5678-84 (2010) Article DOI: 10.1016/j.ejmech.2010.09.022 BindingDB Entry DOI: 10.7270/Q2B27Z30 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gamma-aminobutyric acid type B receptor subunit 1/2 (Rattus norvegicus (Rat)) | BDBM24183 (4-amino-n-[2,3-3H]butyric acid | 4-aminobutanoic a...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG MMDB PC cid PC sid PDB UniChem Patents Similars | PDB PubMed | n/a | n/a | 30 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Displacement of [3H]baclofen from Gamma-aminobutyric acid type B receptor of rat brain membranes | J Med Chem 30: 743-6 (1987) BindingDB Entry DOI: 10.7270/Q22V2GPC | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Gamma-aminobutyric acid type B receptor subunit 1/2 (Rattus norvegicus (Rat)) | BDBM24183 (4-amino-n-[2,3-3H]butyric acid | 4-aminobutanoic a...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG MMDB PC cid PC sid PDB UniChem Patents Similars | PDB PubMed | n/a | n/a | 40 | n/a | n/a | n/a | n/a | n/a | n/a |
Laboratoire de Pharmacie Chimique, Facult� de Pharmacie, Lille, France. Curated by ChEMBL | Assay Description Inhibition of [3H]baclofen binding to rat gamma-aminobutyric acid type B receptor. | J Med Chem 34: 2557-60 (1991) BindingDB Entry DOI: 10.7270/Q2GQ6ZC0 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Similar to alpha-tubulin isoform 1 (Bos taurus) | BDBM50156464 (CHEMBL3793652) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 150 | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ de Lille Curated by ChEMBL | Assay Description Inhibition of bovine tubulin polymerization after 1 hr by fluorescence spectrometry | Eur J Med Chem 115: 393-405 (2016) Article DOI: 10.1016/j.ejmech.2016.03.056 BindingDB Entry DOI: 10.7270/Q2RN39RQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gamma-aminobutyric acid type B receptor subunit 1/2 (Rattus norvegicus (Rat)) | BDBM24182 (4-amino-3-(4-chlorophenyl)butanoic acid | Baclofen...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE PC cid PC sid PDB UniChem Patents Similars | PDB PubMed | n/a | n/a | 200 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Displacement of [3H]baclofen from Gamma-aminobutyric acid type B receptor of rat brain membranes | J Med Chem 30: 743-6 (1987) BindingDB Entry DOI: 10.7270/Q22V2GPC | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Gamma-aminobutyric acid type B receptor subunit 1/2 (Rattus norvegicus (Rat)) | BDBM24182 (4-amino-3-(4-chlorophenyl)butanoic acid | Baclofen...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE PC cid PC sid PDB UniChem Patents Similars | PDB PubMed | n/a | n/a | 330 | n/a | n/a | n/a | n/a | n/a | n/a |
Laboratoire de Pharmacie Chimique, Facult� de Pharmacie, Lille, France. Curated by ChEMBL | Assay Description Inhibition of [3H]baclofen binding to rat gamma-aminobutyric acid type B receptor. | J Med Chem 34: 2557-60 (1991) BindingDB Entry DOI: 10.7270/Q2GQ6ZC0 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Gamma-aminobutyric acid type B receptor subunit 1/2 (Rattus norvegicus (Rat)) | BDBM24182 (4-amino-3-(4-chlorophenyl)butanoic acid | Baclofen...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE PC cid PC sid PDB UniChem Patents Similars | PDB PubMed | n/a | n/a | 330 | n/a | n/a | n/a | n/a | n/a | n/a |
Laboratoire de Pharmacie Chimique, Facult� de Pharmacie, Lille, France. Curated by ChEMBL | Assay Description Inhibition of [3H]baclofen binding to rat gamma-aminobutyric acid type B receptor. | J Med Chem 34: 2557-60 (1991) BindingDB Entry DOI: 10.7270/Q2GQ6ZC0 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Gamma-aminobutyric acid type B receptor subunit 1/2 (Rattus norvegicus (Rat)) | BDBM50007118 (4-Amino-3-(5-chloro-thiophen-2-yl)-butyric acid | ...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 610 | n/a | n/a | n/a | n/a | n/a | n/a |
Laboratoire de Pharmacie Chimique, Facult� de Pharmacie, Lille, France. Curated by ChEMBL | Assay Description Inhibition of [3H]baclofen binding to rat gamma-aminobutyric acid type B receptor. | J Med Chem 34: 2557-60 (1991) BindingDB Entry DOI: 10.7270/Q2GQ6ZC0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gamma-aminobutyric acid type B receptor subunit 1/2 (Rattus norvegicus (Rat)) | BDBM50007121 (4-Amino-3-(2-chloro-phenyl)-butyric acid | CHEMBL8...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 800 | n/a | n/a | n/a | n/a | n/a | n/a |
Laboratoire de Pharmacie Chimique, Facult� de Pharmacie, Lille, France. Curated by ChEMBL | Assay Description Inhibition of [3H]baclofen binding to rat gamma-aminobutyric acid type B receptor. | J Med Chem 34: 2557-60 (1991) BindingDB Entry DOI: 10.7270/Q2GQ6ZC0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gamma-aminobutyric acid type B receptor subunit 1/2 (Rattus norvegicus (Rat)) | BDBM50368295 (CHEMBL301492) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 1.33E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Laboratoire de Pharmacie Chimique, Facult� de Pharmacie, Lille, France. Curated by ChEMBL | Assay Description Inhibition of [3H]baclofen binding to rat gamma-aminobutyric acid type B receptor. | J Med Chem 34: 2557-60 (1991) BindingDB Entry DOI: 10.7270/Q2GQ6ZC0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gamma-aminobutyric acid type B receptor subunit 1/2 (Rattus norvegicus (Rat)) | BDBM50007107 (4-Amino-3-(5-methyl-thiophen-2-yl)-butyric acid | ...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 1.34E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Laboratoire de Pharmacie Chimique, Facult� de Pharmacie, Lille, France. Curated by ChEMBL | Assay Description Inhibition of [3H]baclofen binding to rat gamma-aminobutyric acid type B receptor. | J Med Chem 34: 2557-60 (1991) BindingDB Entry DOI: 10.7270/Q2GQ6ZC0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gamma-aminobutyric acid type B receptor subunit 1/2 (Rattus norvegicus (Rat)) | BDBM50007108 (4-Amino-3-(5-bromo-thiophen-2-yl)-butyric acid | C...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 1.86E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Laboratoire de Pharmacie Chimique, Facult� de Pharmacie, Lille, France. Curated by ChEMBL | Assay Description Inhibition of [3H]baclofen binding to rat gamma-aminobutyric acid type B receptor. | J Med Chem 34: 2557-60 (1991) BindingDB Entry DOI: 10.7270/Q2GQ6ZC0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Similar to alpha-tubulin isoform 1 (Bos taurus) | BDBM50156382 (CHEMBL3794202) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 4.26E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ de Lille Curated by ChEMBL | Assay Description Inhibition of bovine tubulin polymerization after 1 hr by fluorescence spectrometry | Eur J Med Chem 115: 393-405 (2016) Article DOI: 10.1016/j.ejmech.2016.03.056 BindingDB Entry DOI: 10.7270/Q2RN39RQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gamma-aminobutyric acid type B receptor subunit 1/2 (Rattus norvegicus (Rat)) | BDBM50021755 (4-Amino-3-(5-methoxy-benzofuran-2-yl)-butyric acid...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 5.60E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Displacement of [3H]baclofen from Gamma-aminobutyric acid type B receptor of rat brain membranes | J Med Chem 30: 743-6 (1987) BindingDB Entry DOI: 10.7270/Q22V2GPC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gamma-aminobutyric acid type B receptor subunit 1/2 (Rattus norvegicus (Rat)) | BDBM50007117 (4-Amino-3-thiophen-2-yl-butyric acid | CHEMBL31547...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 9.72E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Laboratoire de Pharmacie Chimique, Facult� de Pharmacie, Lille, France. Curated by ChEMBL | Assay Description Inhibition of [3H]baclofen binding to rat gamma-aminobutyric acid type B receptor. | J Med Chem 34: 2557-60 (1991) BindingDB Entry DOI: 10.7270/Q2GQ6ZC0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Similar to alpha-tubulin isoform 1 (Bos taurus) | BDBM50156466 (CHEMBL3792479) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ de Lille Curated by ChEMBL | Assay Description Inhibition of bovine tubulin polymerization after 1 hr by fluorescence spectrometry | Eur J Med Chem 115: 393-405 (2016) Article DOI: 10.1016/j.ejmech.2016.03.056 BindingDB Entry DOI: 10.7270/Q2RN39RQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Similar to alpha-tubulin isoform 1 (Bos taurus) | BDBM50156467 (CHEMBL3794178) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ de Lille Curated by ChEMBL | Assay Description Inhibition of bovine tubulin polymerization after 1 hr by fluorescence spectrometry | Eur J Med Chem 115: 393-405 (2016) Article DOI: 10.1016/j.ejmech.2016.03.056 BindingDB Entry DOI: 10.7270/Q2RN39RQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Similar to alpha-tubulin isoform 1 (Bos taurus) | BDBM50156381 (CHEMBL3794460) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ de Lille Curated by ChEMBL | Assay Description Inhibition of bovine tubulin polymerization after 1 hr by fluorescence spectrometry | Eur J Med Chem 115: 393-405 (2016) Article DOI: 10.1016/j.ejmech.2016.03.056 BindingDB Entry DOI: 10.7270/Q2RN39RQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Similar to alpha-tubulin isoform 1 (Bos taurus) | BDBM50156465 (CHEMBL3793967) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ de Lille Curated by ChEMBL | Assay Description Inhibition of bovine tubulin polymerization after 1 hr by fluorescence spectrometry | Eur J Med Chem 115: 393-405 (2016) Article DOI: 10.1016/j.ejmech.2016.03.056 BindingDB Entry DOI: 10.7270/Q2RN39RQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Similar to alpha-tubulin isoform 1 (Bos taurus) | BDBM50156463 (CHEMBL3793124) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ de Lille Curated by ChEMBL | Assay Description Inhibition of bovine tubulin polymerization after 1 hr by fluorescence spectrometry | Eur J Med Chem 115: 393-405 (2016) Article DOI: 10.1016/j.ejmech.2016.03.056 BindingDB Entry DOI: 10.7270/Q2RN39RQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Similar to alpha-tubulin isoform 1 (Bos taurus) | BDBM50156462 (CHEMBL3793323) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ de Lille Curated by ChEMBL | Assay Description Inhibition of bovine tubulin polymerization after 1 hr by fluorescence spectrometry | Eur J Med Chem 115: 393-405 (2016) Article DOI: 10.1016/j.ejmech.2016.03.056 BindingDB Entry DOI: 10.7270/Q2RN39RQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Similar to alpha-tubulin isoform 1 (Bos taurus) | BDBM50156447 (CHEMBL3792513) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ de Lille Curated by ChEMBL | Assay Description Inhibition of bovine tubulin polymerization after 1 hr by fluorescence spectrometry | Eur J Med Chem 115: 393-405 (2016) Article DOI: 10.1016/j.ejmech.2016.03.056 BindingDB Entry DOI: 10.7270/Q2RN39RQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Similar to alpha-tubulin isoform 1 (Bos taurus) | BDBM50156445 (CHEMBL3793547) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ de Lille Curated by ChEMBL | Assay Description Inhibition of bovine tubulin polymerization after 1 hr by fluorescence spectrometry | Eur J Med Chem 115: 393-405 (2016) Article DOI: 10.1016/j.ejmech.2016.03.056 BindingDB Entry DOI: 10.7270/Q2RN39RQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Similar to alpha-tubulin isoform 1 (Bos taurus) | BDBM50156384 (CHEMBL3793564) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ de Lille Curated by ChEMBL | Assay Description Inhibition of bovine tubulin polymerization after 1 hr by fluorescence spectrometry | Eur J Med Chem 115: 393-405 (2016) Article DOI: 10.1016/j.ejmech.2016.03.056 BindingDB Entry DOI: 10.7270/Q2RN39RQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Similar to alpha-tubulin isoform 1 (Bos taurus) | BDBM50156444 (CHEMBL3792547) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ de Lille Curated by ChEMBL | Assay Description Inhibition of bovine tubulin polymerization after 1 hr by fluorescence spectrometry | Eur J Med Chem 115: 393-405 (2016) Article DOI: 10.1016/j.ejmech.2016.03.056 BindingDB Entry DOI: 10.7270/Q2RN39RQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gamma-aminobutyric acid type B receptor subunit 1/2 (Rattus norvegicus (Rat)) | BDBM50021756 (4-Amino-3-benzofuran-2-yl-butyric acid | CHEMBL349...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 1.80E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Displacement of [3H]baclofen from Gamma-aminobutyric acid type B receptor of rat brain membranes | J Med Chem 30: 743-6 (1987) BindingDB Entry DOI: 10.7270/Q22V2GPC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gamma-aminobutyric acid type B receptor subunit 1/2 (Rattus norvegicus (Rat)) | BDBM50007109 (4-Amino-3-(3-chloro-phenyl)-butyric acid | CHEMBL3...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 2.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Laboratoire de Pharmacie Chimique, Facult� de Pharmacie, Lille, France. Curated by ChEMBL | Assay Description Inhibition of [3H]baclofen binding to rat gamma-aminobutyric acid type B receptor. | J Med Chem 34: 2557-60 (1991) BindingDB Entry DOI: 10.7270/Q2GQ6ZC0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gamma-aminobutyric acid type B receptor subunit 1/2 (Rattus norvegicus (Rat)) | BDBM50007113 (4-Amino-3-thiophen-3-yl-butyric acid | CHEMBL87856) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 2.09E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Laboratoire de Pharmacie Chimique, Facult� de Pharmacie, Lille, France. Curated by ChEMBL | Assay Description Inhibition of [3H]baclofen binding to rat gamma-aminobutyric acid type B receptor. | J Med Chem 34: 2557-60 (1991) BindingDB Entry DOI: 10.7270/Q2GQ6ZC0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gamma-aminobutyric acid type B receptor subunit 1/2 (Rattus norvegicus (Rat)) | BDBM50007110 (4-Amino-3-(4-bromo-thiophen-2-yl)-butyric acid | C...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 3.91E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Laboratoire de Pharmacie Chimique, Facult� de Pharmacie, Lille, France. Curated by ChEMBL | Assay Description Inhibition of [3H]baclofen binding to rat gamma-aminobutyric acid type B receptor. | J Med Chem 34: 2557-60 (1991) BindingDB Entry DOI: 10.7270/Q2GQ6ZC0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gamma-aminobutyric acid type B receptor subunit 1/2 (Rattus norvegicus (Rat)) | BDBM50007111 (4-Amino-3-(4-chloro-thiophen-2-yl)-butyric acid | ...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 4.53E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Laboratoire de Pharmacie Chimique, Facult� de Pharmacie, Lille, France. Curated by ChEMBL | Assay Description Inhibition of [3H]baclofen binding to rat gamma-aminobutyric acid type B receptor. | J Med Chem 34: 2557-60 (1991) BindingDB Entry DOI: 10.7270/Q2GQ6ZC0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gamma-aminobutyric acid type B receptor subunit 1/2 (Rattus norvegicus (Rat)) | BDBM50007120 (4-Amino-3-(4-hydroxy-phenyl)-butyric acid | CHEMBL...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Laboratoire de Pharmacie Chimique, Facult� de Pharmacie, Lille, France. Curated by ChEMBL | Assay Description Inhibition of [3H]baclofen binding to rat gamma-aminobutyric acid type B receptor. | J Med Chem 34: 2557-60 (1991) BindingDB Entry DOI: 10.7270/Q2GQ6ZC0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gamma-aminobutyric acid type B receptor subunit 1/2 (Rattus norvegicus (Rat)) | BDBM50007119 (4-Amino-3-phenyl-butyric acid | CHEMBL53073) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Laboratoire de Pharmacie Chimique, Facult� de Pharmacie, Lille, France. Curated by ChEMBL | Assay Description Inhibition of [3H]baclofen binding to rat gamma-aminobutyric acid type B receptor. | J Med Chem 34: 2557-60 (1991) BindingDB Entry DOI: 10.7270/Q2GQ6ZC0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gamma-aminobutyric acid type B receptor subunit 1/2 (Rattus norvegicus (Rat)) | BDBM50007114 (4-Amino-3-furan-2-yl-butyric acid | CHEMBL85880) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | PubMed | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Laboratoire de Pharmacie Chimique, Facult� de Pharmacie, Lille, France. Curated by ChEMBL | Assay Description Inhibition of [3H]baclofen binding to rat gamma-aminobutyric acid type B receptor. | J Med Chem 34: 2557-60 (1991) BindingDB Entry DOI: 10.7270/Q2GQ6ZC0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gamma-aminobutyric acid type B receptor subunit 1/2 (Rattus norvegicus (Rat)) | BDBM50007112 (4-Amino-3-(5-methyl-furan-2-yl)-butyric acid | CHE...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | PubMed | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Laboratoire de Pharmacie Chimique, Facult� de Pharmacie, Lille, France. Curated by ChEMBL | Assay Description Inhibition of [3H]baclofen binding to rat gamma-aminobutyric acid type B receptor. | J Med Chem 34: 2557-60 (1991) BindingDB Entry DOI: 10.7270/Q2GQ6ZC0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gamma-aminobutyric acid type B receptor subunit 1/2 (Rattus norvegicus (Rat)) | BDBM50021761 (4-Amino-3-[4-(4-fluoro-benzyloxy)-phenyl]-butyric ...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Displacement of [3H]baclofen from Gamma-aminobutyric acid type B receptor of rat brain membranes | J Med Chem 30: 743-6 (1987) BindingDB Entry DOI: 10.7270/Q22V2GPC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gamma-aminobutyric acid type B receptor subunit 1/2 (Rattus norvegicus (Rat)) | BDBM50021759 (4-Amino-3-(5-methoxy-2,3-dihydro-benzofuran-2-yl)-...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Displacement of [3H]baclofen from Gamma-aminobutyric acid type B receptor of rat brain membranes | J Med Chem 30: 743-6 (1987) BindingDB Entry DOI: 10.7270/Q22V2GPC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gamma-aminobutyric acid type B receptor subunit 1/2 (Rattus norvegicus (Rat)) | BDBM50021763 (4-Amino-3-(3-methyl-2-oxo-2,3-dihydro-benzooxazol-...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | PubMed | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Displacement of [3H]baclofen from Gamma-aminobutyric acid type B receptor of rat brain membranes | J Med Chem 30: 743-6 (1987) BindingDB Entry DOI: 10.7270/Q22V2GPC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gamma-aminobutyric acid type B receptor subunit 1/2 (Rattus norvegicus (Rat)) | BDBM50021758 (4-Amino-3-(2,3-dihydro-benzofuran-2-yl)-butyric ac...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Displacement of [3H]baclofen from Gamma-aminobutyric acid type B receptor of rat brain membranes | J Med Chem 30: 743-6 (1987) BindingDB Entry DOI: 10.7270/Q22V2GPC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gamma-aminobutyric acid type B receptor subunit 1/2 (Rattus norvegicus (Rat)) | BDBM50007120 (4-Amino-3-(4-hydroxy-phenyl)-butyric acid | CHEMBL...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Displacement of [3H]baclofen from Gamma-aminobutyric acid type B receptor of rat brain membranes | J Med Chem 30: 743-6 (1987) BindingDB Entry DOI: 10.7270/Q22V2GPC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gamma-aminobutyric acid type B receptor subunit 1/2 (Rattus norvegicus (Rat)) | BDBM50021757 (4-Amino-3-(4-benzyloxy-phenyl)-butyric acid; hydro...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Displacement of [3H]baclofen from Gamma-aminobutyric acid type B receptor of rat brain membranes | J Med Chem 30: 743-6 (1987) BindingDB Entry DOI: 10.7270/Q22V2GPC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gamma-aminobutyric acid type B receptor subunit 1/2 (Rattus norvegicus (Rat)) | BDBM50007116 (4-Amino-3-(3-methyl-thiophen-2-yl)-butyric acid | ...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 1.24E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Laboratoire de Pharmacie Chimique, Facult� de Pharmacie, Lille, France. Curated by ChEMBL | Assay Description Inhibition of [3H]baclofen binding to rat gamma-aminobutyric acid type B receptor. | J Med Chem 34: 2557-60 (1991) BindingDB Entry DOI: 10.7270/Q2GQ6ZC0 | |||||||||||
More data for this Ligand-Target Pair |