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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Gamma-aminobutyric acid type B receptor subunit 1/2' and Ligand = 'BDBM50021763'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Gamma-aminobutyric acid type B receptor subunit 1/2


(Rattus norvegicus (Rat))		BDBM50021763
PNG
(4-Amino-3-(3-methyl-2-oxo-2,3-dihydro-benzooxazol-...)
Show SMILES Cn1c2ccc(cc2oc1=O)C(CN)CC(O)=O
Show InChI InChI=1S/C12H14N2O4/c1-14-9-3-2-7(4-10(9)18-12(14)17)8(6-13)5-11(15)16/h2-4,8H,5-6,13H2,1H3,(H,15,16)
PDB

KEGG

UniProtKB/SwissProt

GoogleScholar
AffyNet 
CHEMBL
PC cid
PC sid
UniChem
PubMed
n/an/a>1.00E+5n/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
Displacement of [3H]baclofen from Gamma-aminobutyric acid type B receptor of rat brain membranes

J Med Chem 30: 743-6 (1987)


BindingDB Entry DOI: 10.7270/Q22V2GPC
More data for this
Ligand-Target Pair