Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Subtilisin-like protease 1 (Plasmodium falciparum) | BDBM50388064![]() (CHEMBL1237284 | TCMDC-123970) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Siena Curated by ChEMBL | Assay Description Inhibition of Plasmodium falciparum SUB1 by fluorimetric assay | Bioorg Med Chem Lett 22: 5317-21 (2012) Article DOI: 10.1016/j.bmcl.2012.06.023 BindingDB Entry DOI: 10.7270/Q2SF2X79 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Subtilisin-like protease 1 (Plasmodium falciparum) | BDBM50388063![]() (CHEMBL2059468) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Siena Curated by ChEMBL | Assay Description Inhibition of Plasmodium falciparum SUB1 by fluorimetric assay | Bioorg Med Chem Lett 22: 5317-21 (2012) Article DOI: 10.1016/j.bmcl.2012.06.023 BindingDB Entry DOI: 10.7270/Q2SF2X79 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Subtilisin-like protease 1 (Plasmodium falciparum) | BDBM50388062![]() (CHEMBL2059472) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 4.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Siena Curated by ChEMBL | Assay Description Inhibition of Plasmodium falciparum SUB1 by fluorimetric assay | Bioorg Med Chem Lett 22: 5317-21 (2012) Article DOI: 10.1016/j.bmcl.2012.06.023 BindingDB Entry DOI: 10.7270/Q2SF2X79 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Subtilisin-like protease 1 (Plasmodium falciparum) | BDBM50388061![]() (CHEMBL2057540) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 4.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Siena Curated by ChEMBL | Assay Description Inhibition of Plasmodium falciparum SUB1 by fluorimetric assay | Bioorg Med Chem Lett 22: 5317-21 (2012) Article DOI: 10.1016/j.bmcl.2012.06.023 BindingDB Entry DOI: 10.7270/Q2SF2X79 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Subtilisin-like protease 1 (Plasmodium falciparum) | BDBM50388066![]() (CHEMBL2059464) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | >5.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Siena Curated by ChEMBL | Assay Description Inhibition of Plasmodium falciparum SUB1 by fluorimetric assay | Bioorg Med Chem Lett 22: 5317-21 (2012) Article DOI: 10.1016/j.bmcl.2012.06.023 BindingDB Entry DOI: 10.7270/Q2SF2X79 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Subtilisin-like protease 1 (Plasmodium falciparum) | BDBM50388067![]() (CHEMBL2059462) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | >5.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Siena Curated by ChEMBL | Assay Description Inhibition of Plasmodium falciparum SUB1 by fluorimetric assay | Bioorg Med Chem Lett 22: 5317-21 (2012) Article DOI: 10.1016/j.bmcl.2012.06.023 BindingDB Entry DOI: 10.7270/Q2SF2X79 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Subtilisin-like protease 1 (Plasmodium falciparum) | BDBM50388065![]() (CHEMBL1237282 | TCMDC-142139) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 5.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Siena Curated by ChEMBL | Assay Description Inhibition of Plasmodium falciparum SUB1 by fluorimetric assay | Bioorg Med Chem Lett 22: 5317-21 (2012) Article DOI: 10.1016/j.bmcl.2012.06.023 BindingDB Entry DOI: 10.7270/Q2SF2X79 | |||||||||||
More data for this Ligand-Target Pair |