BindingDB logo
myBDB logout
Compile Data Set for Download or QSAR

Found 53 hits with Last Name = 'srinivas' and Initial = 'pa'   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Ubiquitin carboxyl-terminal hydrolase 30


(Homo sapiens (Human))
BDBM490051
PNG
((S)-N-(1-((4-(N-(tert- butyl)sulfamoyl)phenyl)amin...)
Show SMILES CC(C)(C)NS(=O)(=O)c1ccc(NC(=O)[C@H](Cc2cccs2)NC(=O)c2ccc(F)cc2)cc1 |r|
Show InChI InChI=1S/C24H26FN3O4S2/c1-24(2,3)28-34(31,32)20-12-10-18(11-13-20)26-23(30)21(15-19-5-4-14-33-19)27-22(29)16-6-8-17(25)9-7-16/h4-14,21,28H,15H2,1-3H3,(H,26,30)(H,27,29)/t21-/m0/s1
PDB

UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 20n/an/an/an/an/an/a


TBA

Assay Description
Inhibition of USP30 (unknown origin) using Ubiquitin-Rhodamine110-Glycine as substrate incubated for 15 mins followed by substrate addition and measu...


Citation and Details

Article DOI: 10.1016/j.bmcl.2018.05.013
BindingDB Entry DOI: 10.7270/Q2NK3JNN
More data for this
Ligand-Target Pair
Ubiquitin carboxyl-terminal hydrolase 30


(Homo sapiens (Human))
BDBM490037
PNG
((S)-N-(1-((4-(N-(tert- butyl)sulfamoyl)phenyl)amin...)
Show SMILES CC(C)(C)NS(=O)(=O)c1ccc(NC(=O)[C@H](CC2CCCCC2)NC(=O)c2ccc(F)cc2)cc1 |r|
Show InChI InChI=1S/C26H34FN3O4S/c1-26(2,3)30-35(33,34)22-15-13-21(14-16-22)28-25(32)23(17-18-7-5-4-6-8-18)29-24(31)19-9-11-20(27)12-10-19/h9-16,18,23,30H,4-8,17H2,1-3H3,(H,28,32)(H,29,31)/t23-/m0/s1
PDB

UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 20n/an/an/an/an/an/a


TBA

Assay Description
Inhibition of USP30 (unknown origin) using Ubiquitin-Rhodamine110-Glycine as substrate incubated for 15 mins followed by substrate addition and measu...


Citation and Details

Article DOI: 10.1016/j.bmcl.2018.05.013
BindingDB Entry DOI: 10.7270/Q2NK3JNN
More data for this
Ligand-Target Pair
Ubiquitin carboxyl-terminal hydrolase 30


(Homo sapiens (Human))
BDBM490029
PNG
((S)-N-(1-((4-(tert- butyl)sulfamoyl)phenyl)amino)-...)
Show SMILES CC(C)(C)NS(=O)(=O)c1ccc(NC(=O)[C@H](Cc2ccccc2)NC(=O)c2ccc(F)cc2)cc1 |r|
Show InChI InChI=1S/C26H28FN3O4S/c1-26(2,3)30-35(33,34)22-15-13-21(14-16-22)28-25(32)23(17-18-7-5-4-6-8-18)29-24(31)19-9-11-20(27)12-10-19/h4-16,23,30H,17H2,1-3H3,(H,28,32)(H,29,31)/t23-/m0/s1
PDB

UniProtKB/SwissProt

GoogleScholar
AffyNet 
Purchase

MCE
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 20n/an/an/an/an/an/a


TBA

Assay Description
Inhibition of USP30 (unknown origin) using Ubiquitin-Rhodamine110-Glycine as substrate incubated for 15 mins followed by substrate addition and measu...


Citation and Details

Article DOI: 10.1016/j.bmcl.2018.05.013
BindingDB Entry DOI: 10.7270/Q2NK3JNN
More data for this
Ligand-Target Pair
Ubiquitin carboxyl-terminal hydrolase 30


(Homo sapiens (Human))
BDBM490068
PNG
((S)-N-(1-((4-(N-(tert- butyl)sulfamoyl)phenyl)amin...)
Show SMILES CC(C)(C)NS(=O)(=O)c1ccc(NC(=O)[C@H](Cc2ccncc2)NC(=O)c2ccc(F)cc2)cc1 |r|
Show InChI InChI=1S/C25H27FN4O4S/c1-25(2,3)30-35(33,34)21-10-8-20(9-11-21)28-24(32)22(16-17-12-14-27-15-13-17)29-23(31)18-4-6-19(26)7-5-18/h4-15,22,30H,16H2,1-3H3,(H,28,32)(H,29,31)/t22-/m0/s1
PDB

UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 20n/an/an/an/an/an/a


TBA

Assay Description
Inhibition of USP30 (unknown origin) using Ubiquitin-Rhodamine110-Glycine as substrate incubated for 15 mins followed by substrate addition and measu...


Citation and Details

Article DOI: 10.1016/j.bmcl.2018.05.013
BindingDB Entry DOI: 10.7270/Q2NK3JNN
More data for this
Ligand-Target Pair
Ubiquitin carboxyl-terminal hydrolase 30


(Homo sapiens (Human))
BDBM490042
PNG
((S)-N-(1-((4-(N-(tert- butyl)sulfamoyl)phenyl)amin...)
Show SMILES CC(C)(C)NS(=O)(=O)c1ccc(NC(=O)[C@H](CC2CCCCC2)NC(=O)c2ccc(F)c(F)c2)cc1 |r|
Show InChI InChI=1S/C26H33F2N3O4S/c1-26(2,3)31-36(34,35)20-12-10-19(11-13-20)29-25(33)23(15-17-7-5-4-6-8-17)30-24(32)18-9-14-21(27)22(28)16-18/h9-14,16-17,23,31H,4-8,15H2,1-3H3,(H,29,33)(H,30,32)/t23-/m0/s1
PDB

UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 30n/an/an/an/an/an/a


TBA

Assay Description
Inhibition of USP30 (unknown origin) using Ubiquitin-Rhodamine110-Glycine as substrate incubated for 15 mins followed by substrate addition and measu...


Citation and Details

Article DOI: 10.1016/j.bmcl.2018.05.013
BindingDB Entry DOI: 10.7270/Q2NK3JNN
More data for this
Ligand-Target Pair
Ubiquitin carboxyl-terminal hydrolase 30


(Homo sapiens (Human))
BDBM490045
PNG
((S)-N-(1-((4-(N-(tert- butyl)sulfamoyl)phenyl)amin...)
Show SMILES CC(C)(C)NS(=O)(=O)c1ccc(NC(=O)[C@H](Cc2cccs2)NC(=O)C2CCCCC2)cc1 |r|
Show InChI InChI=1S/C24H33N3O4S2/c1-24(2,3)27-33(30,31)20-13-11-18(12-14-20)25-23(29)21(16-19-10-7-15-32-19)26-22(28)17-8-5-4-6-9-17/h7,10-15,17,21,27H,4-6,8-9,16H2,1-3H3,(H,25,29)(H,26,28)/t21-/m0/s1
PDB

UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 30n/an/an/an/an/an/a


TBA

Assay Description
Inhibition of USP30 (unknown origin) using Ubiquitin-Rhodamine110-Glycine as substrate incubated for 15 mins followed by substrate addition and measu...


Citation and Details

Article DOI: 10.1016/j.bmcl.2018.05.013
BindingDB Entry DOI: 10.7270/Q2NK3JNN
More data for this
Ligand-Target Pair
Ubiquitin carboxyl-terminal hydrolase 30


(Homo sapiens (Human))
BDBM489719
PNG
((S)-N-(1-((5-(N-(tert- butyl)sulfamoyl)naphthalen-...)
Show SMILES CC(C)(C)NS(=O)(=O)c1cccc2c(NC(=O)[C@H](Cc3ccccc3)NC(=O)c3ccc(F)cc3)cccc12 |r|
Show InChI InChI=1S/C30H30FN3O4S/c1-30(2,3)34-39(37,38)27-14-8-11-23-24(27)12-7-13-25(23)32-29(36)26(19-20-9-5-4-6-10-20)33-28(35)21-15-17-22(31)18-16-21/h4-18,26,34H,19H2,1-3H3,(H,32,36)(H,33,35)/t26-/m0/s1
PDB

UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 49n/an/an/an/an/an/a


TBA

Assay Description
Inhibition of USP30 (unknown origin) using Ubiquitin-Rhodamine110-Glycine as substrate incubated for 15 mins followed by substrate addition and measu...


Citation and Details

Article DOI: 10.1016/j.bmcl.2018.05.013
BindingDB Entry DOI: 10.7270/Q2NK3JNN
More data for this
Ligand-Target Pair
Ubiquitin carboxyl-terminal hydrolase 30


(Homo sapiens (Human))
BDBM490041
PNG
((S)-N-(1-((4-(N-(tert- butyl)sulfamoyl)phenyl)amin...)
Show SMILES CC(C)(C)NS(=O)(=O)c1ccc(NC(=O)[C@H](CC2CCCCC2)NC(=O)c2cccc(F)c2)cc1 |r|
Show InChI InChI=1S/C26H34FN3O4S/c1-26(2,3)30-35(33,34)22-14-12-21(13-15-22)28-25(32)23(16-18-8-5-4-6-9-18)29-24(31)19-10-7-11-20(27)17-19/h7,10-15,17-18,23,30H,4-6,8-9,16H2,1-3H3,(H,28,32)(H,29,31)/t23-/m0/s1
PDB

UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 60n/an/an/an/an/an/a


TBA

Assay Description
Inhibition of USP30 (unknown origin) using Ubiquitin-Rhodamine110-Glycine as substrate incubated for 15 mins followed by substrate addition and measu...


Citation and Details

Article DOI: 10.1016/j.bmcl.2018.05.013
BindingDB Entry DOI: 10.7270/Q2NK3JNN
More data for this
Ligand-Target Pair
Ubiquitin carboxyl-terminal hydrolase 30


(Homo sapiens (Human))
BDBM490026
PNG
((S)-N-(1-((4-(N-(tert- butyl)sulfamoyl)phenyl)amin...)
Show SMILES CC(C)(C)NS(=O)(=O)c1ccc(NC(=O)[C@H](Cc2ccccc2)NC(=O)C2CCCCC2)cc1 |r|
Show InChI InChI=1S/C26H35N3O4S/c1-26(2,3)29-34(32,33)22-16-14-21(15-17-22)27-25(31)23(18-19-10-6-4-7-11-19)28-24(30)20-12-8-5-9-13-20/h4,6-7,10-11,14-17,20,23,29H,5,8-9,12-13,18H2,1-3H3,(H,27,31)(H,28,30)/t23-/m0/s1
PDB

UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 60n/an/an/an/an/an/a


TBA

Assay Description
Inhibition of USP30 (unknown origin) using Ubiquitin-Rhodamine110-Glycine as substrate incubated for 15 mins followed by substrate addition and measu...


Citation and Details

Article DOI: 10.1016/j.bmcl.2018.05.013
BindingDB Entry DOI: 10.7270/Q2NK3JNN
More data for this
Ligand-Target Pair
Ubiquitin carboxyl-terminal hydrolase 30


(Homo sapiens (Human))
BDBM490036
PNG
((S)-N-(1-((4-(N-(tert- butyl)sulfamoyl)phenyl)amin...)
Show SMILES CC(C)(C)NS(=O)(=O)c1ccc(NC(=O)[C@H](CC2CCCCC2)NC(=O)C2CCCCC2)cc1 |r|
Show InChI InChI=1S/C26H41N3O4S/c1-26(2,3)29-34(32,33)22-16-14-21(15-17-22)27-25(31)23(18-19-10-6-4-7-11-19)28-24(30)20-12-8-5-9-13-20/h14-17,19-20,23,29H,4-13,18H2,1-3H3,(H,27,31)(H,28,30)/t23-/m0/s1
PDB

UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 80n/an/an/an/an/an/a


TBA

Assay Description
Inhibition of USP30 (unknown origin) using Ubiquitin-Rhodamine110-Glycine as substrate incubated for 15 mins followed by substrate addition and measu...


Citation and Details

Article DOI: 10.1016/j.bmcl.2018.05.013
BindingDB Entry DOI: 10.7270/Q2NK3JNN
More data for this
Ligand-Target Pair
Ubiquitin carboxyl-terminal hydrolase 30


(Homo sapiens (Human))
BDBM490016
PNG
((S)-N-(1-((5-(N-(tert- butyl)sulfamoyl)naphthalen-...)
Show SMILES COc1ccc(C[C@H](NC(=O)c2ccccc2)C(=O)Nc2cccc3c(cccc23)S(=O)(=O)NC(C)(C)C)cc1 |r|
Show InChI InChI=1S/C31H33N3O5S/c1-31(2,3)34-40(37,38)28-15-9-12-24-25(28)13-8-14-26(24)32-30(36)27(20-21-16-18-23(39-4)19-17-21)33-29(35)22-10-6-5-7-11-22/h5-19,27,34H,20H2,1-4H3,(H,32,36)(H,33,35)/t27-/m0/s1
PDB

UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 90n/an/an/an/an/an/a


TBA

Assay Description
Inhibition of USP30 (unknown origin) using Ubiquitin-Rhodamine110-Glycine as substrate incubated for 15 mins followed by substrate addition and measu...


Citation and Details

Article DOI: 10.1016/j.bmcl.2018.05.013
BindingDB Entry DOI: 10.7270/Q2NK3JNN
More data for this
Ligand-Target Pair
Ubiquitin carboxyl-terminal hydrolase 30


(Homo sapiens (Human))
BDBM445169
PNG
((S)-1-cyano-N-(4-(3- cyanophenyl)thiazol-2-yl)- N-...)
Show SMILES CN(C(=O)[C@@H]1CCCN1C#N)c1nc(cs1)-c1cccc(c1)C#N
Show InChI InChI=1S/C17H15N5OS/c1-21(16(23)15-6-3-7-22(15)11-19)17-20-14(10-24-17)13-5-2-4-12(8-13)9-18/h2,4-5,8,10,15H,3,6-7H2,1H3/t15-/m0/s1
PDB

UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a<100n/an/an/an/an/an/a


TBA

Assay Description
Inhibition of USP30 (unknown origin)


Citation and Details

Article DOI: 10.1016/j.bmcl.2018.05.013
BindingDB Entry DOI: 10.7270/Q2NK3JNN
More data for this
Ligand-Target Pair
Ubiquitin carboxyl-terminal hydrolase 30


(Homo sapiens (Human))
BDBM489727
PNG
((S)-N-(1-((5-(N-(tert- butyl)sulfamoyl)naphthalen-...)
Show SMILES CC(C)(C)NS(=O)(=O)c1cccc2c(NC(=O)[C@H](Cc3ccccc3)NC(=O)C3CCC(F)(F)CC3)cccc12 |r|
Show InChI InChI=1S/C30H35F2N3O4S/c1-29(2,3)35-40(38,39)26-14-8-11-22-23(26)12-7-13-24(22)33-28(37)25(19-20-9-5-4-6-10-20)34-27(36)21-15-17-30(31,32)18-16-21/h4-14,21,25,35H,15-19H2,1-3H3,(H,33,37)(H,34,36)/t25-/m0/s1
PDB

UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 100n/an/an/an/an/an/a


TBA

Assay Description
Inhibition of USP30 (unknown origin) using Ubiquitin-Rhodamine110-Glycine as substrate incubated for 15 mins followed by substrate addition and measu...


Citation and Details

Article DOI: 10.1016/j.bmcl.2018.05.013
BindingDB Entry DOI: 10.7270/Q2NK3JNN
More data for this
Ligand-Target Pair
Ubiquitin carboxyl-terminal hydrolase 30


(Homo sapiens (Human))
BDBM489704
PNG
((S)-N-(1-((5-(N-(tert- butyl)sulfamoyl)naphthalen-...)
Show SMILES CC(C)(C)NS(=O)(=O)c1cccc2c(NC(=O)[C@H](Cc3ccccc3)NC(=O)C3CCCCC3)cccc12 |r|
Show InChI InChI=1S/C30H37N3O4S/c1-30(2,3)33-38(36,37)27-19-11-16-23-24(27)17-10-18-25(23)31-29(35)26(20-21-12-6-4-7-13-21)32-28(34)22-14-8-5-9-15-22/h4,6-7,10-13,16-19,22,26,33H,5,8-9,14-15,20H2,1-3H3,(H,31,35)(H,32,34)/t26-/m0/s1
PDB

UniProtKB/SwissProt

GoogleScholar
AffyNet 
Purchase

MCE
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 120n/an/an/an/an/an/a


TBA

Assay Description
Inhibition of USP30 (unknown origin) using Ubiquitin-Rhodamine110-Glycine as substrate incubated for 15 mins followed by substrate addition and measu...


Citation and Details

Article DOI: 10.1016/j.bmcl.2018.05.013
BindingDB Entry DOI: 10.7270/Q2NK3JNN
More data for this
Ligand-Target Pair
Ubiquitin carboxyl-terminal hydrolase 30


(Homo sapiens (Human))
BDBM490044
PNG
((S)-N-(1-((4-(N-(tert- butyl)sulfamoyl)phenyl)amin...)
Show SMILES CC(C)(C)NS(=O)(=O)c1ccc(NC(=O)[C@H](CC2CCCCC2)NC(=O)c2ccccn2)cc1 |r|
Show InChI InChI=1S/C25H34N4O4S/c1-25(2,3)29-34(32,33)20-14-12-19(13-15-20)27-24(31)22(17-18-9-5-4-6-10-18)28-23(30)21-11-7-8-16-26-21/h7-8,11-16,18,22,29H,4-6,9-10,17H2,1-3H3,(H,27,31)(H,28,30)/t22-/m0/s1
PDB

UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 120n/an/an/an/an/an/a


TBA

Assay Description
Inhibition of USP30 (unknown origin) using Ubiquitin-Rhodamine110-Glycine as substrate incubated for 15 mins followed by substrate addition and measu...


Citation and Details

Article DOI: 10.1016/j.bmcl.2018.05.013
BindingDB Entry DOI: 10.7270/Q2NK3JNN
More data for this
Ligand-Target Pair
Ubiquitin carboxyl-terminal hydrolase 30


(Homo sapiens (Human))
BDBM489745
PNG
((S)-N-(1-((5-(N-(tert- butyl)sulfamoyl)naphthalen-...)
Show SMILES CC(C)(C)NS(=O)(=O)c1cccc2c(NC(=O)[C@H](Cc3ccccc3)NC(=O)c3ccccn3)cccc12 |r|
Show InChI InChI=1S/C29H30N4O4S/c1-29(2,3)33-38(36,37)26-17-10-13-21-22(26)14-9-16-23(21)31-28(35)25(19-20-11-5-4-6-12-20)32-27(34)24-15-7-8-18-30-24/h4-18,25,33H,19H2,1-3H3,(H,31,35)(H,32,34)/t25-/m0/s1
PDB

UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 160n/an/an/an/an/an/a


TBA

Assay Description
Inhibition of USP30 (unknown origin) using Ubiquitin-Rhodamine110-Glycine as substrate incubated for 15 mins followed by substrate addition and measu...


Citation and Details

Article DOI: 10.1016/j.bmcl.2018.05.013
BindingDB Entry DOI: 10.7270/Q2NK3JNN
More data for this
Ligand-Target Pair
Ubiquitin carboxyl-terminal hydrolase 30


(Homo sapiens (Human))
BDBM489738
PNG
((S)-N-(1-((5-(N-(tert- butyl)sulfamoyl)naphthalen-...)
Show SMILES CC(C)(C)NS(=O)(=O)c1cccc2c(NC(=O)[C@H](Cc3ccccc3)NC(=O)c3nccs3)cccc12 |r|
Show InChI InChI=1S/C27H28N4O4S2/c1-27(2,3)31-37(34,35)23-14-8-11-19-20(23)12-7-13-21(19)29-24(32)22(17-18-9-5-4-6-10-18)30-25(33)26-28-15-16-36-26/h4-16,22,31H,17H2,1-3H3,(H,29,32)(H,30,33)/t22-/m0/s1
PDB

UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 180n/an/an/an/an/an/a


TBA

Assay Description
Inhibition of USP30 (unknown origin) using Ubiquitin-Rhodamine110-Glycine as substrate incubated for 15 mins followed by substrate addition and measu...


Citation and Details

Article DOI: 10.1016/j.bmcl.2018.05.013
BindingDB Entry DOI: 10.7270/Q2NK3JNN
More data for this
Ligand-Target Pair
Ubiquitin carboxyl-terminal hydrolase 30


(Homo sapiens (Human))
BDBM490035
PNG
((S)-N-(1-((4-(N-(tert- butyl)sulfamoyl)phenyl)amin...)
Show SMILES CC(C)(C)NS(=O)(=O)c1ccc(NC(=O)[C@H](CC2CCCCC2)NC(=O)c2ccccc2)cc1 |r|
Show InChI InChI=1S/C26H35N3O4S/c1-26(2,3)29-34(32,33)22-16-14-21(15-17-22)27-25(31)23(18-19-10-6-4-7-11-19)28-24(30)20-12-8-5-9-13-20/h5,8-9,12-17,19,23,29H,4,6-7,10-11,18H2,1-3H3,(H,27,31)(H,28,30)/t23-/m0/s1
PDB

UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 230n/an/an/an/an/an/a


TBA

Assay Description
Inhibition of USP30 (unknown origin) using Ubiquitin-Rhodamine110-Glycine as substrate incubated for 15 mins followed by substrate addition and measu...


Citation and Details

Article DOI: 10.1016/j.bmcl.2018.05.013
BindingDB Entry DOI: 10.7270/Q2NK3JNN
More data for this
Ligand-Target Pair
Ubiquitin carboxyl-terminal hydrolase 30


(Homo sapiens (Human))
BDBM489702
PNG
((R)-N-(1-((5-(N-(tert- butyl)sulfamoyl)naphthalen-...)
Show SMILES CC(C)(C)NS(=O)(=O)c1cccc2c(NC(=O)[C@@H](Cc3ccccc3)NC(=O)c3ccccc3)cccc12 |r|
Show InChI InChI=1S/C30H31N3O4S/c1-30(2,3)33-38(36,37)27-19-11-16-23-24(27)17-10-18-25(23)31-29(35)26(20-21-12-6-4-7-13-21)32-28(34)22-14-8-5-9-15-22/h4-19,26,33H,20H2,1-3H3,(H,31,35)(H,32,34)/t26-/m1/s1
PDB

UniProtKB/SwissProt

GoogleScholar
AffyNet 
Purchase

PC cid
PC sid
UniChem
Article
PubMed
n/an/a 250n/an/an/an/an/an/a


TBA

Assay Description
Inhibition of USP30 (unknown origin) using Ubiquitin-Rhodamine110-Glycine as substrate incubated for 15 mins followed by substrate addition and measu...


Citation and Details

Article DOI: 10.1016/j.bmcl.2018.05.013
BindingDB Entry DOI: 10.7270/Q2NK3JNN
More data for this
Ligand-Target Pair
Ubiquitin carboxyl-terminal hydrolase 30


(Homo sapiens (Human))
BDBM490032
PNG
((S)-N-(1-((4-(N-(tert- butyl)sulfamoyl)phenyl)amin...)
Show SMILES CC(C)(C)NS(=O)(=O)c1ccc(NC(=O)[C@H](Cc2ccccc2)NC(=O)c2ccccn2)cc1 |r|
Show InChI InChI=1S/C25H28N4O4S/c1-25(2,3)29-34(32,33)20-14-12-19(13-15-20)27-24(31)22(17-18-9-5-4-6-10-18)28-23(30)21-11-7-8-16-26-21/h4-16,22,29H,17H2,1-3H3,(H,27,31)(H,28,30)/t22-/m0/s1
PDB

UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 250n/an/an/an/an/an/a


TBA

Assay Description
Inhibition of USP30 (unknown origin) using Ubiquitin-Rhodamine110-Glycine as substrate incubated for 15 mins followed by substrate addition and measu...


Citation and Details

Article DOI: 10.1016/j.bmcl.2018.05.013
BindingDB Entry DOI: 10.7270/Q2NK3JNN
More data for this
Ligand-Target Pair
Ubiquitin carboxyl-terminal hydrolase 30


(Homo sapiens (Human))
BDBM489739
PNG
((S)-N-(1-((5-(N-(tert- butyl)sulfamoyl)naphthalen-...)
Show SMILES CC(C)(C)NS(=O)(=O)c1cccc2c(NC(=O)[C@H](Cc3ccccc3)NC(=O)c3ccc(cc3)C#N)cccc12 |r|
Show InChI InChI=1S/C31H30N4O4S/c1-31(2,3)35-40(38,39)28-14-8-11-24-25(28)12-7-13-26(24)33-30(37)27(19-21-9-5-4-6-10-21)34-29(36)23-17-15-22(20-32)16-18-23/h4-18,27,35H,19H2,1-3H3,(H,33,37)(H,34,36)/t27-/m0/s1
PDB

UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 270n/an/an/an/an/an/a


TBA

Assay Description
Inhibition of USP30 (unknown origin) using Ubiquitin-Rhodamine110-Glycine as substrate incubated for 15 mins followed by substrate addition and measu...


Citation and Details

Article DOI: 10.1016/j.bmcl.2018.05.013
BindingDB Entry DOI: 10.7270/Q2NK3JNN
More data for this
Ligand-Target Pair
Ubiquitin carboxyl-terminal hydrolase 30


(Homo sapiens (Human))
BDBM489703
PNG
((S)-N-(1-((5-(N-(tert- butyl)sulfamoyl)naphthalen-...)
Show SMILES CC(C)(C)NS(=O)(=O)c1cccc2c(NC(=O)[C@H](Cc3ccccc3)NC(=O)c3ccccc3)cccc12 |r|
Show InChI InChI=1S/C30H31N3O4S/c1-30(2,3)33-38(36,37)27-19-11-16-23-24(27)17-10-18-25(23)31-29(35)26(20-21-12-6-4-7-13-21)32-28(34)22-14-8-5-9-15-22/h4-19,26,33H,20H2,1-3H3,(H,31,35)(H,32,34)/t26-/m0/s1
PDB

UniProtKB/SwissProt

GoogleScholar
AffyNet 
Purchase

PC cid
PC sid
UniChem
Article
PubMed
n/an/a 270n/an/an/an/an/an/a


TBA

Assay Description
Inhibition of USP30 (unknown origin) using Ubiquitin-Rhodamine110-Glycine as substrate incubated for 15 mins followed by substrate addition and measu...


Citation and Details

Article DOI: 10.1016/j.bmcl.2018.05.013
BindingDB Entry DOI: 10.7270/Q2NK3JNN
More data for this
Ligand-Target Pair
Ubiquitin carboxyl-terminal hydrolase 30


(Homo sapiens (Human))
BDBM50548233
PNG
(CHEMBL4756029)
Show SMILES CC(C)(C)NS(=O)(=O)c1cccc2c(NC(=O)C(Cc3ccccc3)NC(=O)c3ccccc3)cccc12
PDB

UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 370n/an/an/an/an/an/a


TBA

Assay Description
Inhibition of USP30 (unknown origin)


Citation and Details

Article DOI: 10.1016/j.bmcl.2018.05.013
BindingDB Entry DOI: 10.7270/Q2NK3JNN
More data for this
Ligand-Target Pair
Ubiquitin carboxyl-terminal hydrolase 30


(Homo sapiens (Human))
BDBM489721
PNG
((S)-N-(1-((5-(N-(tert- butyl)sulfamoyl)naphthalen-...)
Show SMILES CC(C)(C)NS(=O)(=O)c1cccc2c(NC(=O)[C@H](Cc3ccccc3)NC(=O)C3CCCC3)cccc12 |r|
Show InChI InChI=1S/C29H35N3O4S/c1-29(2,3)32-37(35,36)26-18-10-15-22-23(26)16-9-17-24(22)30-28(34)25(19-20-11-5-4-6-12-20)31-27(33)21-13-7-8-14-21/h4-6,9-12,15-18,21,25,32H,7-8,13-14,19H2,1-3H3,(H,30,34)(H,31,33)/t25-/m0/s1
PDB

UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 370n/an/an/an/an/an/a


TBA

Assay Description
Inhibition of USP30 (unknown origin) using Ubiquitin-Rhodamine110-Glycine as substrate incubated for 15 mins followed by substrate addition and measu...


Citation and Details

Article DOI: 10.1016/j.bmcl.2018.05.013
BindingDB Entry DOI: 10.7270/Q2NK3JNN
More data for this
Ligand-Target Pair
Ubiquitin carboxyl-terminal hydrolase 30


(Homo sapiens (Human))
BDBM490040
PNG
((S)-N-(1-((4-(N-(tert- butyl)sulfamoyl)phenyl)amin...)
Show SMILES CC(C)(C)NS(=O)(=O)c1ccc(NC(=O)[C@H](CC2CCCCC2)NC(=O)c2ccccc2F)cc1 |r|
Show InChI InChI=1S/C26H34FN3O4S/c1-26(2,3)30-35(33,34)20-15-13-19(14-16-20)28-25(32)23(17-18-9-5-4-6-10-18)29-24(31)21-11-7-8-12-22(21)27/h7-8,11-16,18,23,30H,4-6,9-10,17H2,1-3H3,(H,28,32)(H,29,31)/t23-/m0/s1
PDB

UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 460n/an/an/an/an/an/a


TBA

Assay Description
Inhibition of USP30 (unknown origin) using Ubiquitin-Rhodamine110-Glycine as substrate incubated for 15 mins followed by substrate addition and measu...


Citation and Details

Article DOI: 10.1016/j.bmcl.2018.05.013
BindingDB Entry DOI: 10.7270/Q2NK3JNN
More data for this
Ligand-Target Pair
Ubiquitin carboxyl-terminal hydrolase 30


(Homo sapiens (Human))
BDBM490012
PNG
((S)-N-(1-((5-(N-(tert- butyl)sulfamoyl)naphthalen-...)
Show SMILES CC(C)(C)NS(=O)(=O)c1cccc2c(NC(=O)[C@H](Cc3ccc(O)cc3)NC(=O)c3ccccc3)cccc12 |r|
Show InChI InChI=1S/C30H31N3O5S/c1-30(2,3)33-39(37,38)27-14-8-11-23-24(27)12-7-13-25(23)31-29(36)26(19-20-15-17-22(34)18-16-20)32-28(35)21-9-5-4-6-10-21/h4-18,26,33-34H,19H2,1-3H3,(H,31,36)(H,32,35)/t26-/m0/s1
PDB

UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 470n/an/an/an/an/an/a


TBA

Assay Description
Inhibition of USP30 (unknown origin) using Ubiquitin-Rhodamine110-Glycine as substrate incubated for 15 mins followed by substrate addition and measu...


Citation and Details

Article DOI: 10.1016/j.bmcl.2018.05.013
BindingDB Entry DOI: 10.7270/Q2NK3JNN
More data for this
Ligand-Target Pair
Ubiquitin carboxyl-terminal hydrolase 30


(Homo sapiens (Human))
BDBM50548239
PNG
(CHEMBL4747607)
Show SMILES CC(C)NS(=O)(=O)c1cccc2c(NC(=O)C(Cc3ccccc3)NC(=O)c3ccccc3)cccc12
PDB

UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 510n/an/an/an/an/an/a


TBA

Assay Description
Inhibition of USP30 (unknown origin) using Ubiquitin-Rhodamine110-Glycine as substrate incubated for 15 mins followed by substrate addition and measu...


Citation and Details

Article DOI: 10.1016/j.bmcl.2018.05.013
BindingDB Entry DOI: 10.7270/Q2NK3JNN
More data for this
Ligand-Target Pair
Ubiquitin carboxyl-terminal hydrolase 30


(Homo sapiens (Human))
BDBM490013
PNG
((S)-N-(1-((5-(N-(tert- butyl)sulfamoyl)naphthalen-...)
Show SMILES CC(C)(C)NS(=O)(=O)c1cccc2c(NC(=O)[C@H](CC3CCCCC3)NC(=O)c3ccccc3)cccc12 |r|
Show InChI InChI=1S/C30H37N3O4S/c1-30(2,3)33-38(36,37)27-19-11-16-23-24(27)17-10-18-25(23)31-29(35)26(20-21-12-6-4-7-13-21)32-28(34)22-14-8-5-9-15-22/h5,8-11,14-19,21,26,33H,4,6-7,12-13,20H2,1-3H3,(H,31,35)(H,32,34)/t26-/m0/s1
PDB

UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 670n/an/an/an/an/an/a


TBA

Assay Description
Inhibition of USP30 (unknown origin) using Ubiquitin-Rhodamine110-Glycine as substrate incubated for 15 mins followed by substrate addition and measu...


Citation and Details

Article DOI: 10.1016/j.bmcl.2018.05.013
BindingDB Entry DOI: 10.7270/Q2NK3JNN
More data for this
Ligand-Target Pair
Ubiquitin carboxyl-terminal hydrolase 30


(Homo sapiens (Human))
BDBM489709
PNG
((S)-N-(1-((5-(N-(tert- butyl)sulfamoyl)naphthalen-...)
Show SMILES CC(C)(C)NS(=O)(=O)c1cccc2c(NC(=O)[C@H](Cc3ccccc3)NC(=O)c3ccc(Cl)cc3)cccc12 |r|
Show InChI InChI=1S/C30H30ClN3O4S/c1-30(2,3)34-39(37,38)27-14-8-11-23-24(27)12-7-13-25(23)32-29(36)26(19-20-9-5-4-6-10-20)33-28(35)21-15-17-22(31)18-16-21/h4-18,26,34H,19H2,1-3H3,(H,32,36)(H,33,35)/t26-/m0/s1
PDB

UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 830n/an/an/an/an/an/a


TBA

Assay Description
Inhibition of USP30 (unknown origin) using Ubiquitin-Rhodamine110-Glycine as substrate incubated for 15 mins followed by substrate addition and measu...


Citation and Details

Article DOI: 10.1016/j.bmcl.2018.05.013
BindingDB Entry DOI: 10.7270/Q2NK3JNN
More data for this
Ligand-Target Pair
Ubiquitin carboxyl-terminal hydrolase 30


(Homo sapiens (Human))
BDBM490017
PNG
((S)-N-(1-((5-(N-(tert- butyl)sulfamoyl)naphthalen-...)
Show SMILES CC(C)(C)NS(=O)(=O)c1cccc2c(NC(=O)[C@H](CCc3ccccc3)NC(=O)c3ccccc3)cccc12 |r|
Show InChI InChI=1S/C31H33N3O4S/c1-31(2,3)34-39(37,38)28-19-11-16-24-25(28)17-10-18-26(24)32-30(36)27(21-20-22-12-6-4-7-13-22)33-29(35)23-14-8-5-9-15-23/h4-19,27,34H,20-21H2,1-3H3,(H,32,36)(H,33,35)/t27-/m0/s1
PDB

UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 2.27E+3n/an/an/an/an/an/a


TBA

Assay Description
Inhibition of USP30 (unknown origin) using Ubiquitin-Rhodamine110-Glycine as substrate incubated for 15 mins followed by substrate addition and measu...


Citation and Details

Article DOI: 10.1016/j.bmcl.2018.05.013
BindingDB Entry DOI: 10.7270/Q2NK3JNN
More data for this
Ligand-Target Pair
Ubiquitin carboxyl-terminal hydrolase 30


(Homo sapiens (Human))
BDBM489715
PNG
((S)-N-(1-((5-(N-(tert- butyl)sulfamoyl)naphthalen-...)
Show SMILES Cc1ccc(cc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)Nc1cccc2c(cccc12)S(=O)(=O)NC(C)(C)C |r|
Show InChI InChI=1S/C31H33N3O4S/c1-21-16-18-23(19-17-21)29(35)33-27(20-22-10-6-5-7-11-22)30(36)32-26-14-8-13-25-24(26)12-9-15-28(25)39(37,38)34-31(2,3)4/h5-19,27,34H,20H2,1-4H3,(H,32,36)(H,33,35)/t27-/m0/s1
PDB

UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 2.50E+3n/an/an/an/an/an/a


TBA

Assay Description
Inhibition of USP30 (unknown origin) using Ubiquitin-Rhodamine110-Glycine as substrate incubated for 15 mins followed by substrate addition and measu...


Citation and Details

Article DOI: 10.1016/j.bmcl.2018.05.013
BindingDB Entry DOI: 10.7270/Q2NK3JNN
More data for this
Ligand-Target Pair
Ubiquitin carboxyl-terminal hydrolase 30


(Homo sapiens (Human))
BDBM489730
PNG
((S)-N-(1-((5-(N-(tert- butyl)sulfamoyl)naphthalen-...)
Show SMILES CC(C)(C)NS(=O)(=O)c1cccc2c(NC(=O)[C@H](Cc3ccccc3)NC(=O)C3CCCCCC3)cccc12 |r|
Show InChI InChI=1S/C31H39N3O4S/c1-31(2,3)34-39(37,38)28-20-12-17-24-25(28)18-11-19-26(24)32-30(36)27(21-22-13-7-6-8-14-22)33-29(35)23-15-9-4-5-10-16-23/h6-8,11-14,17-20,23,27,34H,4-5,9-10,15-16,21H2,1-3H3,(H,32,36)(H,33,35)/t27-/m0/s1
PDB

UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 4.30E+3n/an/an/an/an/an/a


TBA

Assay Description
Inhibition of USP30 (unknown origin) using Ubiquitin-Rhodamine110-Glycine as substrate incubated for 15 mins followed by substrate addition and measu...


Citation and Details

Article DOI: 10.1016/j.bmcl.2018.05.013
BindingDB Entry DOI: 10.7270/Q2NK3JNN
More data for this
Ligand-Target Pair
Ubiquitin carboxyl-terminal hydrolase 30


(Homo sapiens (Human))
BDBM489743
PNG
((S)-N-(1-((5-(N-(tert- butyl)sulfamoyl)naphthalen-...)
Show SMILES COc1ccc(cc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)Nc1cccc2c(cccc12)S(=O)(=O)NC(C)(C)C |r|
Show InChI InChI=1S/C31H33N3O5S/c1-31(2,3)34-40(37,38)28-15-9-12-24-25(28)13-8-14-26(24)32-30(36)27(20-21-10-6-5-7-11-21)33-29(35)22-16-18-23(39-4)19-17-22/h5-19,27,34H,20H2,1-4H3,(H,32,36)(H,33,35)/t27-/m0/s1
PDB

UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 9.00E+3n/an/an/an/an/an/a


TBA

Assay Description
Inhibition of USP30 (unknown origin) using Ubiquitin-Rhodamine110-Glycine as substrate incubated for 15 mins followed by substrate addition and measu...


Citation and Details

Article DOI: 10.1016/j.bmcl.2018.05.013
BindingDB Entry DOI: 10.7270/Q2NK3JNN
More data for this
Ligand-Target Pair
Ubiquitin carboxyl-terminal hydrolase 30


(Homo sapiens (Human))
BDBM50548236
PNG
(CHEMBL4790811)
Show SMILES CN(C(C)(C)C)S(=O)(=O)c1cccc2c(NC(=O)C(Cc3ccccc3)NC(=O)c3ccccc3)cccc12
PDB

UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a>1.00E+4n/an/an/an/an/an/a


TBA

Assay Description
Inhibition of USP30 (unknown origin) using Ubiquitin-Rhodamine110-Glycine as substrate incubated for 15 mins followed by substrate addition and measu...


Citation and Details

Article DOI: 10.1016/j.bmcl.2018.05.013
BindingDB Entry DOI: 10.7270/Q2NK3JNN
More data for this
Ligand-Target Pair
Ubiquitin carboxyl-terminal hydrolase 30


(Homo sapiens (Human))
BDBM50548235
PNG
(CHEMBL4793428)
Show SMILES CN(C(=O)C(Cc1ccccc1)NC(=O)c1ccccc1)c1cccc2c(cccc12)S(=O)(=O)NC(C)(C)C
PDB

UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a>1.00E+4n/an/an/an/an/an/a


TBA

Assay Description
Inhibition of USP30 (unknown origin) using Ubiquitin-Rhodamine110-Glycine as substrate incubated for 15 mins followed by substrate addition and measu...


Citation and Details

Article DOI: 10.1016/j.bmcl.2018.05.013
BindingDB Entry DOI: 10.7270/Q2NK3JNN
More data for this
Ligand-Target Pair
Ubiquitin carboxyl-terminal hydrolase 30


(Homo sapiens (Human))
BDBM50548234
PNG
(CHEMBL4745470)
Show SMILES CN(C(Cc1ccccc1)C(=O)Nc1cccc2c(cccc12)S(=O)(=O)NC(C)(C)C)C(=O)c1ccccc1
PDB

UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a>1.00E+4n/an/an/an/an/an/a


TBA

Assay Description
Inhibition of USP30 (unknown origin) using Ubiquitin-Rhodamine110-Glycine as substrate incubated for 15 mins followed by substrate addition and measu...


Citation and Details

Article DOI: 10.1016/j.bmcl.2018.05.013
BindingDB Entry DOI: 10.7270/Q2NK3JNN
More data for this
Ligand-Target Pair
Probable ubiquitin carboxyl-terminal hydrolase FAF-X


(Homo sapiens (Human))
BDBM50548233
PNG
(CHEMBL4756029)
Show SMILES CC(C)(C)NS(=O)(=O)c1cccc2c(NC(=O)C(Cc3ccccc3)NC(=O)c3ccccc3)cccc12
PDB

Reactome pathway
KEGG

UniProtKB/SwissProt

antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a>1.00E+4n/an/an/an/an/an/a


TBA

Assay Description
Inhibition of USP9 (unknown origin)


Citation and Details

Article DOI: 10.1016/j.bmcl.2018.05.013
BindingDB Entry DOI: 10.7270/Q2NK3JNN
More data for this
Ligand-Target Pair
Ubiquitin carboxyl-terminal hydrolase 8


(Homo sapiens (Human))
BDBM50548233
PNG
(CHEMBL4756029)
Show SMILES CC(C)(C)NS(=O)(=O)c1cccc2c(NC(=O)C(Cc3ccccc3)NC(=O)c3ccccc3)cccc12
PDB
MMDB

Reactome pathway
KEGG

UniProtKB/SwissProt

B.MOAD
antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a>1.00E+4n/an/an/an/an/an/a


TBA

Assay Description
Inhibition of USP8 (unknown origin)


Citation and Details

Article DOI: 10.1016/j.bmcl.2018.05.013
BindingDB Entry DOI: 10.7270/Q2NK3JNN
More data for this
Ligand-Target Pair
Ubiquitin carboxyl-terminal hydrolase 1


(Homo sapiens (Human))
BDBM50548233
PNG
(CHEMBL4756029)
Show SMILES CC(C)(C)NS(=O)(=O)c1cccc2c(NC(=O)C(Cc3ccccc3)NC(=O)c3ccccc3)cccc12
PDB

UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a>1.00E+4n/an/an/an/an/an/a


TBA

Assay Description
Inhibition of USP1 (unknown origin)


Citation and Details

Article DOI: 10.1016/j.bmcl.2018.05.013
BindingDB Entry DOI: 10.7270/Q2NK3JNN
More data for this
Ligand-Target Pair
Ubiquitin carboxyl-terminal hydrolase 30


(Homo sapiens (Human))
BDBM50548237
PNG
(CHEMBL4758731)
Show SMILES CC(C)(C)NS(=O)(=O)Cc1cccc2c(NC(=O)C(Cc3ccccc3)NC(=O)c3ccccc3)cccc12
PDB

UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a>1.00E+4n/an/an/an/an/an/a


TBA

Assay Description
Inhibition of USP30 (unknown origin) using Ubiquitin-Rhodamine110-Glycine as substrate incubated for 15 mins followed by substrate addition and measu...


Citation and Details

Article DOI: 10.1016/j.bmcl.2018.05.013
BindingDB Entry DOI: 10.7270/Q2NK3JNN
More data for this
Ligand-Target Pair
Ubiquitin carboxyl-terminal hydrolase 30


(Homo sapiens (Human))
BDBM50548238
PNG
(CHEMBL4788134)
Show SMILES CCNS(=O)(=O)c1cccc2c(NC(=O)C(Cc3ccccc3)NC(=O)c3ccccc3)cccc12
PDB

UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a>1.00E+4n/an/an/an/an/an/a


TBA

Assay Description
Inhibition of USP30 (unknown origin) using Ubiquitin-Rhodamine110-Glycine as substrate incubated for 15 mins followed by substrate addition and measu...


Citation and Details

Article DOI: 10.1016/j.bmcl.2018.05.013
BindingDB Entry DOI: 10.7270/Q2NK3JNN
More data for this
Ligand-Target Pair
Ubiquitin carboxyl-terminal hydrolase 30


(Homo sapiens (Human))
BDBM490025
PNG
((S)-N-(1-((4-(N-(tert- butyl)sulfamoyl)phenyl)amin...)
Show SMILES CC(C)(C)NS(=O)(=O)c1ccc(NC(=O)[C@H](Cc2ccccc2)NC(=O)c2ccccc2)cc1 |r|
Show InChI InChI=1S/C26H29N3O4S/c1-26(2,3)29-34(32,33)22-16-14-21(15-17-22)27-25(31)23(18-19-10-6-4-7-11-19)28-24(30)20-12-8-5-9-13-20/h4-17,23,29H,18H2,1-3H3,(H,27,31)(H,28,30)/t23-/m0/s1
PDB

UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a>1.00E+4n/an/an/an/an/an/a


TBA

Assay Description
Inhibition of USP30 (unknown origin) using Ubiquitin-Rhodamine110-Glycine as substrate incubated for 15 mins followed by substrate addition and measu...


Citation and Details

Article DOI: 10.1016/j.bmcl.2018.05.013
BindingDB Entry DOI: 10.7270/Q2NK3JNN
More data for this
Ligand-Target Pair
Ubiquitin carboxyl-terminal hydrolase 30


(Homo sapiens (Human))
BDBM50548240
PNG
(CHEMBL4784059)
Show SMILES CC(C)(C)NC(=O)c1cccc2c(NC(=O)[C@H](Cc3ccccc3)NC(=O)c3ccccc3)cccc12 |r|
PDB

UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a>1.00E+4n/an/an/an/an/an/a


TBA

Assay Description
Inhibition of USP30 (unknown origin) using Ubiquitin-Rhodamine110-Glycine as substrate incubated for 15 mins followed by substrate addition and measu...


Citation and Details

Article DOI: 10.1016/j.bmcl.2018.05.013
BindingDB Entry DOI: 10.7270/Q2NK3JNN
More data for this
Ligand-Target Pair
Ubiquitin carboxyl-terminal hydrolase 30


(Homo sapiens (Human))
BDBM489705
PNG
((S)-N-(1-((5-(N-(tert- butyl)sulfamoyl)naphthalen-...)
Show SMILES CC(C)(C)NS(=O)(=O)c1cccc2c(NC(=O)[C@H](Cc3ccccc3)NC(=O)C3CC3)cccc12 |r|
Show InChI InChI=1S/C27H31N3O4S/c1-27(2,3)30-35(33,34)24-14-8-11-20-21(24)12-7-13-22(20)28-26(32)23(29-25(31)19-15-16-19)17-18-9-5-4-6-10-18/h4-14,19,23,30H,15-17H2,1-3H3,(H,28,32)(H,29,31)/t23-/m0/s1
PDB

UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a>1.00E+4n/an/an/an/an/an/a


TBA

Assay Description
Inhibition of USP30 (unknown origin) using Ubiquitin-Rhodamine110-Glycine as substrate incubated for 15 mins followed by substrate addition and measu...


Citation and Details

Article DOI: 10.1016/j.bmcl.2018.05.013
BindingDB Entry DOI: 10.7270/Q2NK3JNN
More data for this
Ligand-Target Pair
Ubiquitin carboxyl-terminal hydrolase 30


(Homo sapiens (Human))
BDBM50548245
PNG
(CHEMBL4752106)
Show SMILES CC(C)(C)NS(=O)(=O)c1cccc2c(NC(=O)[C@H](Cc3ccccc3)NC(=O)OCc3ccccc3)cccc12 |r|
PDB

UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a>1.00E+4n/an/an/an/an/an/a


TBA

Assay Description
Inhibition of USP30 (unknown origin) using Ubiquitin-Rhodamine110-Glycine as substrate incubated for 15 mins followed by substrate addition and measu...


Citation and Details

Article DOI: 10.1016/j.bmcl.2018.05.013
BindingDB Entry DOI: 10.7270/Q2NK3JNN
More data for this
Ligand-Target Pair
Ubiquitin carboxyl-terminal hydrolase 30


(Homo sapiens (Human))
BDBM489708
PNG
((S)-N-(5-(N-(tert- butyl)sulfamoyl)naphthalen-1-yl...)
Show SMILES CC(C)(C)NS(=O)(=O)c1cccc2c(NC(=O)[C@H](Cc3ccccc3)NC(=O)CCc3ccccc3)cccc12 |r|
Show InChI InChI=1S/C32H35N3O4S/c1-32(2,3)35-40(38,39)29-19-11-16-25-26(29)17-10-18-27(25)34-31(37)28(22-24-14-8-5-9-15-24)33-30(36)21-20-23-12-6-4-7-13-23/h4-19,28,35H,20-22H2,1-3H3,(H,33,36)(H,34,37)/t28-/m0/s1
PDB

UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a>1.00E+4n/an/an/an/an/an/a


TBA

Assay Description
Inhibition of USP30 (unknown origin) using Ubiquitin-Rhodamine110-Glycine as substrate incubated for 15 mins followed by substrate addition and measu...


Citation and Details

Article DOI: 10.1016/j.bmcl.2018.05.013
BindingDB Entry DOI: 10.7270/Q2NK3JNN
More data for this
Ligand-Target Pair
Ubiquitin carboxyl-terminal hydrolase 30


(Homo sapiens (Human))
BDBM489707
PNG
((S)-N-(5-(N-(tert- butyl)sulfamoyl)naphthalen-1-yl...)
Show SMILES CC(C)(C)NS(=O)(=O)c1cccc2c(NC(=O)[C@H](Cc3ccccc3)NC(=O)Cc3ccccc3)cccc12 |r|
Show InChI InChI=1S/C31H33N3O4S/c1-31(2,3)34-39(37,38)28-19-11-16-24-25(28)17-10-18-26(24)33-30(36)27(20-22-12-6-4-7-13-22)32-29(35)21-23-14-8-5-9-15-23/h4-19,27,34H,20-21H2,1-3H3,(H,32,35)(H,33,36)/t27-/m0/s1
PDB

UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a>1.00E+4n/an/an/an/an/an/a


TBA

Assay Description
Inhibition of USP30 (unknown origin) using Ubiquitin-Rhodamine110-Glycine as substrate incubated for 15 mins followed by substrate addition and measu...


Citation and Details

Article DOI: 10.1016/j.bmcl.2018.05.013
BindingDB Entry DOI: 10.7270/Q2NK3JNN
More data for this
Ligand-Target Pair
Ubiquitin carboxyl-terminal hydrolase 30


(Homo sapiens (Human))
BDBM490023
PNG
((S)-N-(1-((5-(N-(tert- butyl)sulfamoyl)naphthalen-...)
Show SMILES Cc1ccc(C[C@H](NC(=O)c2ccccc2)C(=O)Nc2cccc3c(cccc23)S(=O)(=O)NC(C)(C)C)cc1 |r|
Show InChI InChI=1S/C31H33N3O4S/c1-21-16-18-22(19-17-21)20-27(33-29(35)23-10-6-5-7-11-23)30(36)32-26-14-8-13-25-24(26)12-9-15-28(25)39(37,38)34-31(2,3)4/h5-19,27,34H,20H2,1-4H3,(H,32,36)(H,33,35)/t27-/m0/s1
PDB

UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a>1.00E+4n/an/an/an/an/an/a


TBA

Assay Description
Inhibition of USP30 (unknown origin) using Ubiquitin-Rhodamine110-Glycine as substrate incubated for 15 mins followed by substrate addition and measu...


Citation and Details

Article DOI: 10.1016/j.bmcl.2018.05.013
BindingDB Entry DOI: 10.7270/Q2NK3JNN
More data for this
Ligand-Target Pair
Ubiquitin carboxyl-terminal hydrolase 30


(Homo sapiens (Human))
BDBM489744
PNG
((S)-N-(1-((5-(N-(tert- butyl)sulfamoyl)naphthalen-...)
Show SMILES CC(C)(C)NS(=O)(=O)c1cccc2c(NC(=O)[C@H](Cc3ccccc3)NC(=O)c3ccc(O)cc3)cccc12 |r|
Show InChI InChI=1S/C30H31N3O5S/c1-30(2,3)33-39(37,38)27-14-8-11-23-24(27)12-7-13-25(23)31-29(36)26(19-20-9-5-4-6-10-20)32-28(35)21-15-17-22(34)18-16-21/h4-18,26,33-34H,19H2,1-3H3,(H,31,36)(H,32,35)/t26-/m0/s1
PDB

UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a>1.00E+4n/an/an/an/an/an/a


TBA

Assay Description
Inhibition of USP30 (unknown origin) using Ubiquitin-Rhodamine110-Glycine as substrate incubated for 15 mins followed by substrate addition and measu...


Citation and Details

Article DOI: 10.1016/j.bmcl.2018.05.013
BindingDB Entry DOI: 10.7270/Q2NK3JNN
More data for this
Ligand-Target Pair
Ubiquitin carboxyl-terminal hydrolase 30


(Homo sapiens (Human))
BDBM50548241
PNG
(CHEMBL4743014)
Show SMILES CC(C)(C)NS(=O)(=O)c1cccc2c(NC(=O)CNC(=O)c3ccccc3)cccc12
PDB

UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a>1.00E+4n/an/an/an/an/an/a


TBA

Assay Description
Inhibition of USP30 (unknown origin) using Ubiquitin-Rhodamine110-Glycine as substrate incubated for 15 mins followed by substrate addition and measu...


Citation and Details

Article DOI: 10.1016/j.bmcl.2018.05.013
BindingDB Entry DOI: 10.7270/Q2NK3JNN
More data for this
Ligand-Target Pair
Displayed 1 to 50 (of 53 total )  |  Next  |  Last  >>
Jump to: