Found 719 hits with Last Name = 'barone' and Initial = 'd' Target/Host
(Institution) | Ligand | Target/Host
Links | Ligand
Links | Trg + Lig
Links | Ki
nM | ΔG°
kJ/mole | IC50
nM | Kd
nM | EC50/IC50
nM | koff
s-1 | kon
M-1s-1 | pH | Temp
°C |
|---|
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor
(Rattus norvegicus (rat)-Rattus norvegicus (Rat)) | BDBM50225657
(CHEMBL173570)Show SMILES CS(O)(=O)=O.CC(c1ccccc1)n1nc(c2CNCCc12)-c1ccc(F)cc1 Show InChI InChI=1S/C20H20FN3.CH4O3S/c1-14(15-5-3-2-4-6-15)24-19-11-12-22-13-18(19)20(23-24)16-7-9-17(21)10-8-16;1-5(2,3)4/h2-10,14,22H,11-13H2,1H3;1H3,(H,2,3,4) | PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
GoogleScholar
AffyNet 
| CHEMBL
PC cid
PC sid
UniChem
Patents
Similars
| PubMed
| 7.20 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
Curated by ChEMBL
| Assay Description
Ability to displace [3H]prazosin from postsynaptic alpha-1 adrenergic receptor of rat in vitro. |
J Med Chem 28: 934-40 (1985)
BindingDB Entry DOI: 10.7270/Q29C70NC |
More data for this
Ligand-Target Pair | |
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor
(Rattus norvegicus (rat)-Rattus norvegicus (Rat)) | BDBM50225567
(CHEMBL559369)Show SMILES Cl.CC(c1ccccc1)n1nc(c2CN(C)CCc12)-c1ccc(F)cc1 Show InChI InChI=1S/C21H22FN3.ClH/c1-15(16-6-4-3-5-7-16)25-20-12-13-24(2)14-19(20)21(23-25)17-8-10-18(22)11-9-17;/h3-11,15H,12-14H2,1-2H3;1H | PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Patents
| PubMed
| 8.10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
Curated by ChEMBL
| Assay Description
Ability to displace [3H]prazosin from postsynaptic alpha-1 adrenergic receptor of rat in vitro. |
J Med Chem 28: 934-40 (1985)
BindingDB Entry DOI: 10.7270/Q29C70NC |
More data for this
Ligand-Target Pair | |
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor
(Rattus norvegicus (rat)-Rattus norvegicus (Rat)) | BDBM50225661
(CHEMBL173988)Show SMILES CS(O)(=O)=O.CCCCCn1nc(c2CNCCc12)-c1ccc(F)cc1 Show InChI InChI=1S/C17H22FN3/c1-2-3-4-11-21-16-9-10-19-12-15(16)17(20-21)13-5-7-14(18)8-6-13/h5-8,19H,2-4,9-12H2,1H3 | PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Patents
Similars
| PubMed
| 8.70 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
Curated by ChEMBL
| Assay Description
Ability to displace [3H]prazosin from postsynaptic alpha-1 adrenergic receptor of rat in vitro. |
J Med Chem 28: 934-40 (1985)
BindingDB Entry DOI: 10.7270/Q29C70NC |
More data for this
Ligand-Target Pair | |
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor
(Rattus norvegicus (rat)-Rattus norvegicus (Rat)) | BDBM50225671
(CHEMBL369407)Show SMILES CS(O)(=O)=O.CCCCCCn1nc(c2CNCCc12)-c1ccc(F)cc1 Show InChI InChI=1S/C18H24FN3/c1-2-3-4-5-12-22-17-10-11-20-13-16(17)18(21-22)14-6-8-15(19)9-7-14/h6-9,20H,2-5,10-13H2,1H3 | PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Patents
Similars
| PubMed
| 13 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
Curated by ChEMBL
| Assay Description
Ability to displace [3H]prazosin from postsynaptic alpha-1 adrenergic receptor of rat in vitro. |
J Med Chem 28: 934-40 (1985)
BindingDB Entry DOI: 10.7270/Q29C70NC |
More data for this
Ligand-Target Pair | |
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor
(Rattus norvegicus (rat)-Rattus norvegicus (Rat)) | BDBM50225573
(CHEMBL173140)Show SMILES CS(O)(=O)=O.Fc1ccc(cc1)-c1nn(CCCc2ccccc2)c2CCNCc12 Show InChI InChI=1S/C21H22FN3/c22-18-10-8-17(9-11-18)21-19-15-23-13-12-20(19)25(24-21)14-4-7-16-5-2-1-3-6-16/h1-3,5-6,8-11,23H,4,7,12-15H2 | PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
| PubMed
| 13 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
Curated by ChEMBL
| Assay Description
Ability to displace [3H]prazosin from postsynaptic alpha-1 adrenergic receptor of rat in vitro. |
J Med Chem 28: 934-40 (1985)
BindingDB Entry DOI: 10.7270/Q29C70NC |
More data for this
Ligand-Target Pair | |
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor
(Rattus norvegicus (rat)-Rattus norvegicus (Rat)) | BDBM50225576
(CHEMBL535357)Show InChI InChI=1S/C19H18FN3/c20-16-8-6-15(7-9-16)19-17-12-21-11-10-18(17)23(22-19)13-14-4-2-1-3-5-14/h1-9,21H,10-13H2 | PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| PubMed
| 15 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
Curated by ChEMBL
| Assay Description
Ability to displace [3H]prazosin from postsynaptic alpha-1 adrenergic receptor of rat in vitro. |
J Med Chem 28: 934-40 (1985)
BindingDB Entry DOI: 10.7270/Q29C70NC |
More data for this
Ligand-Target Pair | |
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor
(Rattus norvegicus (rat)-Rattus norvegicus (Rat)) | BDBM50225570
(CHEMBL171362)Show SMILES CS(O)(=O)=O.CCCCCCn1nc(c2CN(C)CCc12)-c1ccc(F)cc1 Show InChI InChI=1S/C19H26FN3/c1-3-4-5-6-12-23-18-11-13-22(2)14-17(18)19(21-23)15-7-9-16(20)10-8-15/h7-10H,3-6,11-14H2,1-2H3 | PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| PubMed
| 15 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
Curated by ChEMBL
| Assay Description
Ability to displace [3H]prazosin from postsynaptic alpha-1 adrenergic receptor of rat in vitro. |
J Med Chem 28: 934-40 (1985)
BindingDB Entry DOI: 10.7270/Q29C70NC |
More data for this
Ligand-Target Pair | |
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor
(Rattus norvegicus (rat)-Rattus norvegicus (Rat)) | BDBM50225673
(CHEMBL175271)Show SMILES CS(O)(=O)=O.CCCCn1nc(c2CNCCc12)-c1ccc(F)cc1 Show InChI InChI=1S/C16H20FN3/c1-2-3-10-20-15-8-9-18-11-14(15)16(19-20)12-4-6-13(17)7-5-12/h4-7,18H,2-3,8-11H2,1H3 | PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Patents
Similars
| PubMed
| 17 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
Curated by ChEMBL
| Assay Description
Ability to displace [3H]prazosin from postsynaptic alpha-1 adrenergic receptor of rat in vitro. |
J Med Chem 28: 934-40 (1985)
BindingDB Entry DOI: 10.7270/Q29C70NC |
More data for this
Ligand-Target Pair | |
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor
(Rattus norvegicus (rat)-Rattus norvegicus (Rat)) | BDBM50225575
(CHEMBL427474)Show SMILES CS(O)(=O)=O.CCCCCn1nc(c2CN(C)CCc12)-c1ccc(F)cc1 Show InChI InChI=1S/C18H24FN3/c1-3-4-5-11-22-17-10-12-21(2)13-16(17)18(20-22)14-6-8-15(19)9-7-14/h6-9H,3-5,10-13H2,1-2H3 | PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| PubMed
| 18 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
Curated by ChEMBL
| Assay Description
Ability to displace [3H]prazosin from postsynaptic alpha-1 adrenergic receptor of rat in vitro. |
J Med Chem 28: 934-40 (1985)
BindingDB Entry DOI: 10.7270/Q29C70NC |
More data for this
Ligand-Target Pair | |
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor
(Rattus norvegicus (rat)-Rattus norvegicus (Rat)) | BDBM50225574
(CHEMBL540615)Show SMILES Cl.CN1CCc2c(C1)c(nn2CCCc1ccccc1)-c1ccc(F)cc1 Show InChI InChI=1S/C22H24FN3/c1-25-15-13-21-20(16-25)22(18-9-11-19(23)12-10-18)24-26(21)14-5-8-17-6-3-2-4-7-17/h2-4,6-7,9-12H,5,8,13-16H2,1H3 | PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| PubMed
| 21 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
Curated by ChEMBL
| Assay Description
Ability to displace [3H]prazosin from postsynaptic alpha-1 adrenergic receptor of rat in vitro. |
J Med Chem 28: 934-40 (1985)
BindingDB Entry DOI: 10.7270/Q29C70NC |
More data for this
Ligand-Target Pair | |
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor
(Rattus norvegicus (rat)-Rattus norvegicus (Rat)) | BDBM50225554
(CHEMBL368408)Show SMILES CS(O)(=O)=O.CN1CCc2c(C1)c(nn2Cc1ccccc1)-c1ccc(F)cc1 Show InChI InChI=1S/C20H20FN3/c1-23-12-11-19-18(14-23)20(16-7-9-17(21)10-8-16)22-24(19)13-15-5-3-2-4-6-15/h2-10H,11-14H2,1H3 | PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| PubMed
| 21 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
Curated by ChEMBL
| Assay Description
Ability to displace [3H]prazosin from postsynaptic alpha-1 adrenergic receptor of rat in vitro. |
J Med Chem 28: 934-40 (1985)
BindingDB Entry DOI: 10.7270/Q29C70NC |
More data for this
Ligand-Target Pair | |
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor
(Rattus norvegicus (rat)-Rattus norvegicus (Rat)) | BDBM50225672
(CHEMBL171898)Show InChI InChI=1S/C15H18FN3/c1-2-9-19-14-7-8-17-10-13(14)15(18-19)11-3-5-12(16)6-4-11/h3-6,17H,2,7-10H2,1H3 | PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Patents
Similars
| PubMed
| 24 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
Curated by ChEMBL
| Assay Description
Ability to displace [3H]prazosin from postsynaptic alpha-1 adrenergic receptor of rat in vitro. |
J Med Chem 28: 934-40 (1985)
BindingDB Entry DOI: 10.7270/Q29C70NC |
More data for this
Ligand-Target Pair | |
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor
(Rattus norvegicus (rat)-Rattus norvegicus (Rat)) | BDBM50225577
(CHEMBL353160)Show SMILES CS(O)(=O)=O.CCCCn1nc(c2CN(C)CCc12)-c1ccc(F)cc1 Show InChI InChI=1S/C17H22FN3/c1-3-4-10-21-16-9-11-20(2)12-15(16)17(19-21)13-5-7-14(18)8-6-13/h5-8H,3-4,9-12H2,1-2H3 | PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| PubMed
| 33 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
Curated by ChEMBL
| Assay Description
Ability to displace [3H]prazosin from postsynaptic alpha-1 adrenergic receptor of rat in vitro. |
J Med Chem 28: 934-40 (1985)
BindingDB Entry DOI: 10.7270/Q29C70NC |
More data for this
Ligand-Target Pair | |
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor
(Rattus norvegicus (rat)-Rattus norvegicus (Rat)) | BDBM50225555
(CHEMBL174512)Show InChI InChI=1S/C14H16FN3/c1-2-18-13-7-8-16-9-12(13)14(17-18)10-3-5-11(15)6-4-10/h3-6,16H,2,7-9H2,1H3 | PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
| PubMed
| 33 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
Curated by ChEMBL
| Assay Description
Ability to displace [3H]prazosin from postsynaptic alpha-1 adrenergic receptor of rat in vitro. |
J Med Chem 28: 934-40 (1985)
BindingDB Entry DOI: 10.7270/Q29C70NC |
More data for this
Ligand-Target Pair | |
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor
(Rattus norvegicus (rat)-Rattus norvegicus (Rat)) | BDBM50225568
(CHEMBL171296)Show InChI InChI=1S/C21H22FN3/c1-24-13-12-20-19(15-24)21(17-7-9-18(22)10-8-17)23-25(20)14-11-16-5-3-2-4-6-16/h2-10H,11-15H2,1H3 | PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Patents
Similars
| PubMed
| 40 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
Curated by ChEMBL
| Assay Description
Ability to displace [3H]prazosin from postsynaptic alpha-1 adrenergic receptor of rat in vitro. |
J Med Chem 28: 934-40 (1985)
BindingDB Entry DOI: 10.7270/Q29C70NC |
More data for this
Ligand-Target Pair | |
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor
(Rattus norvegicus (rat)-Rattus norvegicus (Rat)) | BDBM50225658
(CHEMBL176567)Show SMILES CS(O)(=O)=O.Fc1ccc(cc1)-c1nn(CCc2ccccc2)c2CCNCc12 Show InChI InChI=1S/C20H20FN3/c21-17-8-6-16(7-9-17)20-18-14-22-12-10-19(18)24(23-20)13-11-15-4-2-1-3-5-15/h1-9,22H,10-14H2 | PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| PubMed
| 40 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
Curated by ChEMBL
| Assay Description
Ability to displace [3H]prazosin from postsynaptic alpha-1 adrenergic receptor of rat in vitro. |
J Med Chem 28: 934-40 (1985)
BindingDB Entry DOI: 10.7270/Q29C70NC |
More data for this
Ligand-Target Pair | |
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor
(Rattus norvegicus (rat)-Rattus norvegicus (Rat)) | BDBM50225564
(CHEMBL536715)Show SMILES Cl.Fc1ccc(cc1)-c1nn(Cc2ccccc2)c2CCN(Cc12)C1CCCC1 Show InChI InChI=1S/C24H26FN3/c25-20-12-10-19(11-13-20)24-22-17-27(21-8-4-5-9-21)15-14-23(22)28(26-24)16-18-6-2-1-3-7-18/h1-3,6-7,10-13,21H,4-5,8-9,14-17H2 | PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Patents
Similars
| PubMed
| 42 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
Curated by ChEMBL
| Assay Description
Ability to displace [3H]prazosin from postsynaptic alpha-1 adrenergic receptor of rat in vitro. |
J Med Chem 28: 934-40 (1985)
BindingDB Entry DOI: 10.7270/Q29C70NC |
More data for this
Ligand-Target Pair | |
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor
(Rattus norvegicus (rat)-Rattus norvegicus (Rat)) | BDBM50225579
(CHEMBL355447)Show InChI InChI=1S/C12H12FN3/c13-9-3-1-8(2-4-9)12-10-7-14-6-5-11(10)15-16-12/h1-4,14H,5-7H2,(H,15,16) | PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
GoogleScholar
AffyNet
| Purchase
CHEMBL
PC cid
PC sid
UniChem
| PubMed
| 69 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
Curated by ChEMBL
| Assay Description
Ability to displace [3H]prazosin from postsynaptic alpha-1 adrenergic receptor of rat in vitro. |
J Med Chem 28: 934-40 (1985)
BindingDB Entry DOI: 10.7270/Q29C70NC |
More data for this
Ligand-Target Pair | |
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor
(Rattus norvegicus (rat)-Rattus norvegicus (Rat)) | BDBM50225569
(CHEMBL353329)Show SMILES CS(O)(=O)=O.CCCn1nc(c2CN(C)CCc12)-c1ccc(F)cc1 Show InChI InChI=1S/C16H20FN3/c1-3-9-20-15-8-10-19(2)11-14(15)16(18-20)12-4-6-13(17)7-5-12/h4-7H,3,8-11H2,1-2H3 | PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| PubMed
| 74 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
Curated by ChEMBL
| Assay Description
Ability to displace [3H]prazosin from postsynaptic alpha-1 adrenergic receptor of rat in vitro. |
J Med Chem 28: 934-40 (1985)
BindingDB Entry DOI: 10.7270/Q29C70NC |
More data for this
Ligand-Target Pair | |
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor
(Rattus norvegicus (rat)-Rattus norvegicus (Rat)) | BDBM50225676
(CHEMBL3216631)Show InChI InChI=1S/C13H15N3/c1-9-2-4-10(5-3-9)13-11-8-14-7-6-12(11)15-16-13/h2-5,14H,6-8H2,1H3,(H,15,16) | PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Patents
Similars
| PubMed
| 92 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
Curated by ChEMBL
| Assay Description
Ability to displace [3H]prazosin from postsynaptic alpha-1 adrenergic receptor of rat in vitro. |
J Med Chem 28: 934-40 (1985)
BindingDB Entry DOI: 10.7270/Q29C70NC |
More data for this
Ligand-Target Pair | |
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor
(Rattus norvegicus (rat)-Rattus norvegicus (Rat)) | BDBM50225660
(CHEMBL174934)Show SMILES CC(C)N1CCc2c(C1)c(nn2Cc1ccccc1)-c1ccc(F)cc1 Show InChI InChI=1S/C22H24FN3/c1-16(2)25-13-12-21-20(15-25)22(18-8-10-19(23)11-9-18)24-26(21)14-17-6-4-3-5-7-17/h3-11,16H,12-15H2,1-2H3 | PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Patents
Similars
| PubMed
| 98 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
Curated by ChEMBL
| Assay Description
Ability to displace [3H]prazosin from postsynaptic alpha-1 adrenergic receptor of rat in vitro. |
J Med Chem 28: 934-40 (1985)
BindingDB Entry DOI: 10.7270/Q29C70NC |
More data for this
Ligand-Target Pair | |
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor
(Rattus norvegicus (rat)-Rattus norvegicus (Rat)) | BDBM50225557
(CHEMBL534693)Show SMILES Cl.CCCCN1CCc2c(C1)c(nn2Cc1ccccc1)-c1ccc(F)cc1 Show InChI InChI=1S/C23H26FN3/c1-2-3-14-26-15-13-22-21(17-26)23(19-9-11-20(24)12-10-19)25-27(22)16-18-7-5-4-6-8-18/h4-12H,2-3,13-17H2,1H3 | PDB
Reactome pathway
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| 119 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
Curated by ChEMBL
| Assay Description
Ability to displace [3H]prazosin from postsynaptic alpha-1 adrenergic receptor of rat in vitro. |
J Med Chem 28: 934-40 (1985)
BindingDB Entry DOI: 10.7270/Q29C70NC |
More data for this
Ligand-Target Pair | |
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor
(Rattus norvegicus (rat)-Rattus norvegicus (Rat)) | BDBM50225558
(CHEMBL553465)Show InChI InChI=1S/C12H12ClN3/c13-9-3-1-8(2-4-9)12-10-7-14-6-5-11(10)15-16-12/h1-4,14H,5-7H2,(H,15,16) | PDB
Reactome pathway
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| 145 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
Curated by ChEMBL
| Assay Description
Ability to displace [3H]prazosin from postsynaptic alpha-1 adrenergic receptor of rat in vitro. |
J Med Chem 28: 934-40 (1985)
BindingDB Entry DOI: 10.7270/Q29C70NC |
More data for this
Ligand-Target Pair | |
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor
(Rattus norvegicus (rat)-Rattus norvegicus (Rat)) | BDBM50225678
(CHEMBL539332)Show InChI InChI=1S/C18H15F2N3/c19-13-3-1-12(2-4-13)18-16-11-21-10-9-17(16)23(22-18)15-7-5-14(20)6-8-15/h1-8,21H,9-11H2 | PDB
Reactome pathway
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| 161 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
Curated by ChEMBL
| Assay Description
Ability to displace [3H]prazosin from postsynaptic alpha-1 adrenergic receptor of rat in vitro. |
J Med Chem 28: 934-40 (1985)
BindingDB Entry DOI: 10.7270/Q29C70NC |
More data for this
Ligand-Target Pair | |
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor
(Rattus norvegicus (rat)-Rattus norvegicus (Rat)) | BDBM50225668
(CHEMBL552522)Show InChI InChI=1S/C13H14ClN3/c1-17-12-6-7-15-8-11(12)13(16-17)9-2-4-10(14)5-3-9/h2-5,15H,6-8H2,1H3 | PDB
Reactome pathway
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| 190 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
Curated by ChEMBL
| Assay Description
Ability to displace [3H]prazosin from postsynaptic alpha-1 adrenergic receptor of rat in vitro. |
J Med Chem 28: 934-40 (1985)
BindingDB Entry DOI: 10.7270/Q29C70NC |
More data for this
Ligand-Target Pair | |
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor
(Rattus norvegicus (rat)-Rattus norvegicus (Rat)) | BDBM50225556
(CHEMBL174027)Show SMILES CS(O)(=O)=O.CN1CCc2c(C1)c(nn2-c1ccc(F)cc1)-c1ccc(F)cc1 Show InChI InChI=1S/C19H17F2N3/c1-23-11-10-18-17(12-23)19(13-2-4-14(20)5-3-13)22-24(18)16-8-6-15(21)7-9-16/h2-9H,10-12H2,1H3 | PDB
Reactome pathway
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| 206 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
Curated by ChEMBL
| Assay Description
Ability to displace [3H]prazosin from postsynaptic alpha-1 adrenergic receptor of rat in vitro. |
J Med Chem 28: 934-40 (1985)
BindingDB Entry DOI: 10.7270/Q29C70NC |
More data for this
Ligand-Target Pair | |
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor
(Rattus norvegicus (rat)-Rattus norvegicus (Rat)) | BDBM50225560
(CHEMBL177092)Show SMILES Cc1ccc(cc1)S(O)(=O)=O.CN1CCc2n[nH]c(c2C1)-c1ccc(C)cc1 Show InChI InChI=1S/C14H17N3/c1-10-3-5-11(6-4-10)14-12-9-17(2)8-7-13(12)15-16-14/h3-6H,7-9H2,1-2H3,(H,15,16) | PDB
Reactome pathway
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| 249 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
Curated by ChEMBL
| Assay Description
Ability to displace [3H]prazosin from postsynaptic alpha-1 adrenergic receptor of rat in vitro. |
J Med Chem 28: 934-40 (1985)
BindingDB Entry DOI: 10.7270/Q29C70NC |
More data for this
Ligand-Target Pair | |
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor
(Rattus norvegicus (rat)-Rattus norvegicus (Rat)) | BDBM50225654
(CHEMBL172121)Show SMILES OC(=O)CC(O)=O.CCN1CCc2n[nH]c(c2C1)-c1ccc(C)cc1 Show InChI InChI=1S/C15H19N3/c1-3-18-9-8-14-13(10-18)15(17-16-14)12-6-4-11(2)5-7-12/h4-7H,3,8-10H2,1-2H3,(H,16,17) | PDB
Reactome pathway
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| 350 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
Curated by ChEMBL
| Assay Description
Ability to displace [3H]prazosin from postsynaptic alpha-1 adrenergic receptor of rat in vitro. |
J Med Chem 28: 934-40 (1985)
BindingDB Entry DOI: 10.7270/Q29C70NC |
More data for this
Ligand-Target Pair | |
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor
(Rattus norvegicus (rat)-Rattus norvegicus (Rat)) | BDBM50225666
(CHEMBL173504)Show SMILES CS(O)(=O)=O.CCn1nc(c2CN(C)CCc12)-c1ccc(F)cc1 Show InChI InChI=1S/C15H18FN3/c1-3-19-14-8-9-18(2)10-13(14)15(17-19)11-4-6-12(16)7-5-11/h4-7H,3,8-10H2,1-2H3 | PDB
Reactome pathway
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| 362 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
Curated by ChEMBL
| Assay Description
Ability to displace [3H]prazosin from postsynaptic alpha-1 adrenergic receptor of rat in vitro. |
J Med Chem 28: 934-40 (1985)
BindingDB Entry DOI: 10.7270/Q29C70NC |
More data for this
Ligand-Target Pair | |
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor
(Rattus norvegicus (rat)-Rattus norvegicus (Rat)) | BDBM50225655
(CHEMBL175218)Show InChI InChI=1S/C13H15N3O/c1-17-10-4-2-9(3-5-10)13-11-8-14-7-6-12(11)15-16-13/h2-5,14H,6-8H2,1H3,(H,15,16) | PDB
Reactome pathway
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| 448 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
Curated by ChEMBL
| Assay Description
Ability to displace [3H]prazosin from postsynaptic alpha-1 adrenergic receptor of rat in vitro. |
J Med Chem 28: 934-40 (1985)
BindingDB Entry DOI: 10.7270/Q29C70NC |
More data for this
Ligand-Target Pair | |
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor
(Rattus norvegicus (rat)-Rattus norvegicus (Rat)) | BDBM50225549
(CHEMBL3216881)Show InChI InChI=1S/C12H13N3/c1-2-4-9(5-3-1)12-10-8-13-7-6-11(10)14-15-12/h1-5,13H,6-8H2,(H,14,15) | PDB
Reactome pathway
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| 490 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
Curated by ChEMBL
| Assay Description
Ability to displace [3H]prazosin from postsynaptic alpha-1 adrenergic receptor of rat in vitro. |
J Med Chem 28: 934-40 (1985)
BindingDB Entry DOI: 10.7270/Q29C70NC |
More data for this
Ligand-Target Pair | |
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor
(Rattus norvegicus (rat)-Rattus norvegicus (Rat)) | BDBM50225659
(CHEMBL177161)Show InChI InChI=1S/C13H14FN3/c1-17-7-6-12-11(8-17)13(16-15-12)9-2-4-10(14)5-3-9/h2-5H,6-8H2,1H3,(H,15,16) | PDB
Reactome pathway
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| 507 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
Curated by ChEMBL
| Assay Description
Ability to displace [3H]prazosin from postsynaptic alpha-1 adrenergic receptor of rat in vitro. |
J Med Chem 28: 934-40 (1985)
BindingDB Entry DOI: 10.7270/Q29C70NC |
More data for this
Ligand-Target Pair | |
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor
(Rattus norvegicus (rat)-Rattus norvegicus (Rat)) | BDBM50225675
(CHEMBL174513)Show InChI InChI=1S/C13H14FN3/c1-17-12-6-7-15-8-11(12)13(16-17)9-2-4-10(14)5-3-9/h2-5,15H,6-8H2,1H3 | PDB
Reactome pathway
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| 1.06E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
Curated by ChEMBL
| Assay Description
Ability to displace [3H]prazosin from postsynaptic alpha-1 adrenergic receptor of rat in vitro. |
J Med Chem 28: 934-40 (1985)
BindingDB Entry DOI: 10.7270/Q29C70NC |
More data for this
Ligand-Target Pair | |
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor
(Rattus norvegicus (rat)-Rattus norvegicus (Rat)) | BDBM50225656
(CHEMBL174126)Show InChI InChI=1S/C15H19N3/c1-11(2)18-14-8-9-16-10-13(14)15(17-18)12-6-4-3-5-7-12/h3-7,11,16H,8-10H2,1-2H3 | PDB
Reactome pathway
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| 1.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
Curated by ChEMBL
| Assay Description
Ability to displace [3H]prazosin from postsynaptic alpha-1 adrenergic receptor of rat in vitro. |
J Med Chem 28: 934-40 (1985)
BindingDB Entry DOI: 10.7270/Q29C70NC |
More data for this
Ligand-Target Pair | |
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor
(Rattus norvegicus (rat)-Rattus norvegicus (Rat)) | BDBM50225566
(CHEMBL172130)Show SMILES OC(=O)CC(O)(CC(O)=O)C(O)=O.CN1CCc2n[nH]c(c2C1)-c1ccccc1 Show InChI InChI=1S/C13H15N3/c1-16-8-7-12-11(9-16)13(15-14-12)10-5-3-2-4-6-10/h2-6H,7-9H2,1H3,(H,14,15) | PDB
Reactome pathway
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| 1.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
Curated by ChEMBL
| Assay Description
Ability to displace [3H]prazosin from postsynaptic alpha-1 adrenergic receptor of rat in vitro. |
J Med Chem 28: 934-40 (1985)
BindingDB Entry DOI: 10.7270/Q29C70NC |
More data for this
Ligand-Target Pair | |
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor
(Rattus norvegicus (rat)-Rattus norvegicus (Rat)) | BDBM50225669
(CHEMBL538812)Show InChI InChI=1S/C14H17N3/c1-2-17-9-8-13-12(10-17)14(16-15-13)11-6-4-3-5-7-11/h3-7H,2,8-10H2,1H3,(H,15,16) | PDB
Reactome pathway
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| 1.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
Curated by ChEMBL
| Assay Description
Ability to displace [3H]prazosin from postsynaptic alpha-1 adrenergic receptor of rat in vitro. |
J Med Chem 28: 934-40 (1985)
BindingDB Entry DOI: 10.7270/Q29C70NC |
More data for this
Ligand-Target Pair | |
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor
(Rattus norvegicus (rat)-Rattus norvegicus (Rat)) | BDBM50225561
(CHEMBL177160)Show SMILES OC(=O)CC(O)(CC(O)=O)C(O)=O.CN1CCc2n[nH]c(c2C1)-c1ccc(Cl)cc1 Show InChI InChI=1S/C13H14ClN3/c1-17-7-6-12-11(8-17)13(16-15-12)9-2-4-10(14)5-3-9/h2-5H,6-8H2,1H3,(H,15,16) | PDB
Reactome pathway
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| 2.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
Curated by ChEMBL
| Assay Description
Ability to displace [3H]prazosin from postsynaptic alpha-1 adrenergic receptor of rat in vitro. |
J Med Chem 28: 934-40 (1985)
BindingDB Entry DOI: 10.7270/Q29C70NC |
More data for this
Ligand-Target Pair | |
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor
(Rattus norvegicus (rat)-Rattus norvegicus (Rat)) | BDBM50225670
(CHEMBL174346)Show SMILES CS(O)(=O)=O.CCn1nc(c2CN(Cc3ccccc3)CCc12)-c1ccc(F)cc1 Show InChI InChI=1S/C21H22FN3/c1-2-25-20-12-13-24(14-16-6-4-3-5-7-16)15-19(20)21(23-25)17-8-10-18(22)11-9-17/h3-11H,2,12-15H2,1H3 | PDB
Reactome pathway
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| 2.02E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
Curated by ChEMBL
| Assay Description
Ability to displace [3H]prazosin from postsynaptic alpha-1 adrenergic receptor of rat in vitro. |
J Med Chem 28: 934-40 (1985)
BindingDB Entry DOI: 10.7270/Q29C70NC |
More data for this
Ligand-Target Pair | |
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor
(Rattus norvegicus (rat)-Rattus norvegicus (Rat)) | BDBM50225662
(CHEMBL368299)Show SMILES CS(O)(=O)=O.CC(C)n1nc(c2CN(C)CCc12)-c1ccccc1 Show InChI InChI=1S/C16H21N3/c1-12(2)19-15-9-10-18(3)11-14(15)16(17-19)13-7-5-4-6-8-13/h4-8,12H,9-11H2,1-3H3 | PDB
Reactome pathway
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| 2.87E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
Curated by ChEMBL
| Assay Description
Ability to displace [3H]prazosin from postsynaptic alpha-1 adrenergic receptor of rat in vitro. |
J Med Chem 28: 934-40 (1985)
BindingDB Entry DOI: 10.7270/Q29C70NC |
More data for this
Ligand-Target Pair | |
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor
(Rattus norvegicus (rat)-Rattus norvegicus (Rat)) | BDBM50225674
(CHEMBL174204)Show InChI InChI=1S/C12H12FN3/c13-9-3-1-2-8(6-9)12-10-7-14-5-4-11(10)15-16-12/h1-3,6,14H,4-5,7H2,(H,15,16) | PDB
Reactome pathway
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| >3.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
Curated by ChEMBL
| Assay Description
Ability to displace [3H]prazosin from postsynaptic alpha-1 adrenergic receptor of rat in vitro. |
J Med Chem 28: 934-40 (1985)
BindingDB Entry DOI: 10.7270/Q29C70NC |
More data for this
Ligand-Target Pair | |
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor
(Rattus norvegicus (rat)-Rattus norvegicus (Rat)) | BDBM50225667
(CHEMBL172357)Show InChI InChI=1S/C12H12ClN3/c13-9-3-1-2-8(6-9)12-10-7-14-5-4-11(10)15-16-12/h1-3,6,14H,4-5,7H2,(H,15,16) | PDB
Reactome pathway
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| >3.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
Curated by ChEMBL
| Assay Description
Ability to displace [3H]prazosin from postsynaptic alpha-1 adrenergic receptor of rat in vitro. |
J Med Chem 28: 934-40 (1985)
BindingDB Entry DOI: 10.7270/Q29C70NC |
More data for this
Ligand-Target Pair | |
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor
(Rattus norvegicus (rat)-Rattus norvegicus (Rat)) | BDBM50225665
(CHEMBL368369)Show InChI InChI=1S/C13H14FN3/c1-17-12-5-6-15-8-11(12)13(16-17)9-3-2-4-10(14)7-9/h2-4,7,15H,5-6,8H2,1H3 | PDB
Reactome pathway
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| >3.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
Curated by ChEMBL
| Assay Description
Ability to displace [3H]prazosin from postsynaptic alpha-1 adrenergic receptor of rat in vitro. |
J Med Chem 28: 934-40 (1985)
BindingDB Entry DOI: 10.7270/Q29C70NC |
More data for this
Ligand-Target Pair | |
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor
(Rattus norvegicus (rat)-Rattus norvegicus (Rat)) | BDBM50225664
(CHEMBL175219)Show InChI InChI=1S/C13H12N4/c14-7-9-1-3-10(4-2-9)13-11-8-15-6-5-12(11)16-17-13/h1-4,15H,5-6,8H2,(H,16,17) | PDB
Reactome pathway
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| >3.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
Curated by ChEMBL
| Assay Description
Ability to displace [3H]prazosin from postsynaptic alpha-1 adrenergic receptor of rat in vitro. |
J Med Chem 28: 934-40 (1985)
BindingDB Entry DOI: 10.7270/Q29C70NC |
More data for this
Ligand-Target Pair | |
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor
(Rattus norvegicus (rat)-Rattus norvegicus (Rat)) | BDBM50225578
(CHEMBL368541)Show SMILES Cc1ccc(cc1)S(O)(=O)=O.Cn1nc(c2CNCCc12)-c1ccccc1F Show InChI InChI=1S/C13H14FN3/c1-17-12-6-7-15-8-10(12)13(16-17)9-4-2-3-5-11(9)14/h2-5,15H,6-8H2,1H3 | PDB
Reactome pathway
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Similars
| PubMed
| >3.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
Curated by ChEMBL
| Assay Description
Ability to displace [3H]prazosin from postsynaptic alpha-1 adrenergic receptor of rat in vitro. |
J Med Chem 28: 934-40 (1985)
BindingDB Entry DOI: 10.7270/Q29C70NC |
More data for this
Ligand-Target Pair | |
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor
(Rattus norvegicus (rat)-Rattus norvegicus (Rat)) | BDBM50225565
(CHEMBL557186)Show InChI InChI=1S/C12H12N4O2/c17-16(18)9-3-1-8(2-4-9)12-10-7-13-6-5-11(10)14-15-12/h1-4,13H,5-7H2,(H,14,15) | PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
| PubMed
| >3.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
Curated by ChEMBL
| Assay Description
Ability to displace [3H]prazosin from postsynaptic alpha-1 adrenergic receptor of rat in vitro. |
J Med Chem 28: 934-40 (1985)
BindingDB Entry DOI: 10.7270/Q29C70NC |
More data for this
Ligand-Target Pair | |
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor
(Rattus norvegicus (rat)-Rattus norvegicus (Rat)) | BDBM50225548
(CHEMBL174178)Show InChI InChI=1S/C14H17N3O2/c1-18-12-4-3-9(7-13(12)19-2)14-10-8-15-6-5-11(10)16-17-14/h3-4,7,15H,5-6,8H2,1-2H3,(H,16,17) | PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
GoogleScholar
AffyNet
| Purchase
CHEMBL
PC cid
PC sid
UniChem
Similars
| PubMed
| >3.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
Curated by ChEMBL
| Assay Description
Ability to displace [3H]prazosin from postsynaptic alpha-1 adrenergic receptor of rat in vitro. |
J Med Chem 28: 934-40 (1985)
BindingDB Entry DOI: 10.7270/Q29C70NC |
More data for this
Ligand-Target Pair | |
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor
(Rattus norvegicus (rat)-Rattus norvegicus (Rat)) | BDBM50225680
(CHEMBL367848)Show InChI InChI=1S/C13H14ClN3/c1-17-12-5-6-15-8-11(12)13(16-17)9-3-2-4-10(14)7-9/h2-4,7,15H,5-6,8H2,1H3 | PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| PubMed
| >3.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
Curated by ChEMBL
| Assay Description
Ability to displace [3H]prazosin from postsynaptic alpha-1 adrenergic receptor of rat in vitro. |
J Med Chem 28: 934-40 (1985)
BindingDB Entry DOI: 10.7270/Q29C70NC |
More data for this
Ligand-Target Pair | |
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor
(Rattus norvegicus (rat)-Rattus norvegicus (Rat)) | BDBM50225580
(CHEMBL171410)Show InChI InChI=1S/C15H19N3O/c1-3-18-9-8-14-13(10-18)15(17-16-14)11-4-6-12(19-2)7-5-11/h4-7H,3,8-10H2,1-2H3,(H,16,17) | PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| PubMed
| >3.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
Curated by ChEMBL
| Assay Description
Ability to displace [3H]prazosin from postsynaptic alpha-1 adrenergic receptor of rat in vitro. |
J Med Chem 28: 934-40 (1985)
BindingDB Entry DOI: 10.7270/Q29C70NC |
More data for this
Ligand-Target Pair | |
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor
(Rattus norvegicus (rat)-Rattus norvegicus (Rat)) | BDBM50225679
(CHEMBL170483)Show InChI InChI=1S/C12H12FN3/c13-10-4-2-1-3-8(10)12-9-7-14-6-5-11(9)15-16-12/h1-4,14H,5-7H2,(H,15,16) | PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
GoogleScholar
AffyNet
| Purchase
CHEMBL
PC cid
PC sid
UniChem
| PubMed
| >3.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
Curated by ChEMBL
| Assay Description
Ability to displace [3H]prazosin from postsynaptic alpha-1 adrenergic receptor of rat in vitro. |
J Med Chem 28: 934-40 (1985)
BindingDB Entry DOI: 10.7270/Q29C70NC |
More data for this
Ligand-Target Pair | |
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor
(Rattus norvegicus (rat)-Rattus norvegicus (Rat)) | BDBM50225677
(CHEMBL367555)Show InChI InChI=1S/C13H15N3/c1-16-12-7-8-14-9-11(12)13(15-16)10-5-3-2-4-6-10/h2-6,14H,7-9H2,1H3 | PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Patents
Similars
| PubMed
| 3.29E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
Curated by ChEMBL
| Assay Description
Ability to displace [3H]prazosin from postsynaptic alpha-1 adrenergic receptor of rat in vitro. |
J Med Chem 28: 934-40 (1985)
BindingDB Entry DOI: 10.7270/Q29C70NC |
More data for this
Ligand-Target Pair | |
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