Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
D(2) dopamine receptor (Homo sapiens (Human)) | BDBM21398 (4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG PC cid PC sid PDB UniChem Patents Similars | DrugBank PubMed | 0.160 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Uppsala University Curated by ChEMBL | Assay Description Displacement of [3H]-quinpirole from human dopamine D2A receptors expressed in LtK cells | Bioorg Med Chem Lett 9: 2167-72 (1999) BindingDB Entry DOI: 10.7270/Q2CF9P97 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(2) dopamine receptor (Homo sapiens (Human)) | BDBM21398 (4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG PC cid PC sid PDB UniChem Patents Similars | DrugBank PubMed | 0.440 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Uppsala University Curated by ChEMBL | Assay Description Displacement of [3H]-raclopride from human dopamine D2A receptors expressed in LtK cells | Bioorg Med Chem Lett 9: 2167-72 (1999) BindingDB Entry DOI: 10.7270/Q2CF9P97 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(2) dopamine receptor (Homo sapiens (Human)) | BDBM55121 (3-HYDROXYTYRAMINE HYDROCHLORIDE | 4-(2-aminoethyl)...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase DrugBank KEGG PC cid PC sid PDB UniChem Similars | DrugBank PubMed | 1.90 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Uppsala University Curated by ChEMBL | Assay Description Displacement of [3H]-quinpirole from human dopamine D2A receptors expressed in LtK cells | Bioorg Med Chem Lett 9: 2167-72 (1999) BindingDB Entry DOI: 10.7270/Q2CF9P97 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(2) dopamine receptor (Homo sapiens (Human)) | BDBM50080053 (((R)-5-Methoxy-1,2,3,4-tetrahydro-naphthalen-2-yl)...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | PubMed | 6.40 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Uppsala University Curated by ChEMBL | Assay Description Displacement of [3H]-quinpirole from human dopamine D2A receptors expressed in LtK cells | Bioorg Med Chem Lett 9: 2167-72 (1999) BindingDB Entry DOI: 10.7270/Q2CF9P97 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(2) dopamine receptor (Homo sapiens (Human)) | BDBM50080047 ((4-Methoxy-benzyl)-((R)-5-methoxy-1,2,3,4-tetrahyd...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 22 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Uppsala University Curated by ChEMBL | Assay Description Displacement of [3H]-raclopride from human dopamine D2A receptors expressed in LtK cells | Bioorg Med Chem Lett 9: 2167-72 (1999) BindingDB Entry DOI: 10.7270/Q2CF9P97 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(2) dopamine receptor (Homo sapiens (Human)) | BDBM50053670 (((R)-5-Fluoro-1,2,3,4-tetrahydro-naphthalen-2-yl)-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 26 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Uppsala University Curated by ChEMBL | Assay Description Displacement of [3H]-quinpirole from human dopamine D2A receptors expressed in LtK cells | Bioorg Med Chem Lett 9: 2167-72 (1999) BindingDB Entry DOI: 10.7270/Q2CF9P97 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(2) dopamine receptor (Homo sapiens (Human)) | BDBM50080048 ((4-Fluoro-benzyl)-((R)-5-methoxy-1,2,3,4-tetrahydr...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 43.8 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Uppsala University Curated by ChEMBL | Assay Description Displacement of [3H]-raclopride from human dopamine D2A receptors expressed in LtK cells | Bioorg Med Chem Lett 9: 2167-72 (1999) BindingDB Entry DOI: 10.7270/Q2CF9P97 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(2) dopamine receptor (Homo sapiens (Human)) | BDBM50080053 (((R)-5-Methoxy-1,2,3,4-tetrahydro-naphthalen-2-yl)...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | PubMed | 46 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Uppsala University Curated by ChEMBL | Assay Description Displacement of [3H]-raclopride from human dopamine D2A receptors expressed in LtK cells | Bioorg Med Chem Lett 9: 2167-72 (1999) BindingDB Entry DOI: 10.7270/Q2CF9P97 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(2) dopamine receptor (Homo sapiens (Human)) | BDBM50080050 (((R)-5-Methoxy-1,2,3,4-tetrahydro-naphthalen-2-yl)...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 59 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Uppsala University Curated by ChEMBL | Assay Description Displacement of [3H]-raclopride from human dopamine D2A receptors expressed in LtK cells | Bioorg Med Chem Lett 9: 2167-72 (1999) BindingDB Entry DOI: 10.7270/Q2CF9P97 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(2) dopamine receptor (Homo sapiens (Human)) | BDBM50080047 ((4-Methoxy-benzyl)-((R)-5-methoxy-1,2,3,4-tetrahyd...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 64 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Uppsala University Curated by ChEMBL | Assay Description Displacement of [3H]-quinpirole from human dopamine D2A receptors expressed in LtK cells | Bioorg Med Chem Lett 9: 2167-72 (1999) BindingDB Entry DOI: 10.7270/Q2CF9P97 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(2) dopamine receptor (Homo sapiens (Human)) | BDBM50080051 (Benzyl-((R)-5-methoxy-1,2,3,4-tetrahydro-naphthale...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 65.6 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Uppsala University Curated by ChEMBL | Assay Description Displacement of [3H]-raclopride from human dopamine D2A receptors expressed in LtK cells | Bioorg Med Chem Lett 9: 2167-72 (1999) BindingDB Entry DOI: 10.7270/Q2CF9P97 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(2) dopamine receptor (Homo sapiens (Human)) | BDBM50080048 ((4-Fluoro-benzyl)-((R)-5-methoxy-1,2,3,4-tetrahydr...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 70 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Uppsala University Curated by ChEMBL | Assay Description Displacement of [3H]-quinpirole from human dopamine D2A receptors expressed in LtK cells | Bioorg Med Chem Lett 9: 2167-72 (1999) BindingDB Entry DOI: 10.7270/Q2CF9P97 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(2) dopamine receptor (Homo sapiens (Human)) | BDBM50080051 (Benzyl-((R)-5-methoxy-1,2,3,4-tetrahydro-naphthale...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 75 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Uppsala University Curated by ChEMBL | Assay Description Displacement of [3H]-quinpirole from human dopamine D2A receptors expressed in LtK cells | Bioorg Med Chem Lett 9: 2167-72 (1999) BindingDB Entry DOI: 10.7270/Q2CF9P97 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(2) dopamine receptor (Homo sapiens (Human)) | BDBM50080055 (((R)-5-Methoxy-1,2,3,4-tetrahydro-naphthalen-2-yl)...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | PubMed | 82.3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Uppsala University Curated by ChEMBL | Assay Description Displacement of [3H]-quinpirole from human dopamine D2A receptors expressed in LtK cells | Bioorg Med Chem Lett 9: 2167-72 (1999) BindingDB Entry DOI: 10.7270/Q2CF9P97 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(2) dopamine receptor (Homo sapiens (Human)) | BDBM50080055 (((R)-5-Methoxy-1,2,3,4-tetrahydro-naphthalen-2-yl)...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | PubMed | 114 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Uppsala University Curated by ChEMBL | Assay Description Displacement of [3H]-raclopride from human dopamine D2A receptors expressed in LtK cells | Bioorg Med Chem Lett 9: 2167-72 (1999) BindingDB Entry DOI: 10.7270/Q2CF9P97 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(2) dopamine receptor (Homo sapiens (Human)) | BDBM50080052 (CHEMBL303502 | Furan-2-ylmethyl-((R)-5-methoxy-1,2...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | PubMed | 118 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Uppsala University Curated by ChEMBL | Assay Description Displacement of [3H]-quinpirole from human dopamine D2A receptors expressed in LtK cells | Bioorg Med Chem Lett 9: 2167-72 (1999) BindingDB Entry DOI: 10.7270/Q2CF9P97 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(2) dopamine receptor (Homo sapiens (Human)) | BDBM50080052 (CHEMBL303502 | Furan-2-ylmethyl-((R)-5-methoxy-1,2...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | PubMed | 125 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Uppsala University Curated by ChEMBL | Assay Description Displacement of [3H]-raclopride from human dopamine D2A receptors expressed in LtK cells | Bioorg Med Chem Lett 9: 2167-72 (1999) BindingDB Entry DOI: 10.7270/Q2CF9P97 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(2) dopamine receptor (Homo sapiens (Human)) | BDBM50080049 (((R)-5-Methoxy-1,2,3,4-tetrahydro-naphthalen-2-yl)...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | PubMed | 152 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Uppsala University Curated by ChEMBL | Assay Description Displacement of [3H]-raclopride from human dopamine D2A receptors expressed in LtK cells | Bioorg Med Chem Lett 9: 2167-72 (1999) BindingDB Entry DOI: 10.7270/Q2CF9P97 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(2) dopamine receptor (Homo sapiens (Human)) | BDBM50054337 (Benzyl-((R)-5-fluoro-1,2,3,4-tetrahydro-naphthalen...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 179 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Uppsala University Curated by ChEMBL | Assay Description Inhibition of [3H]-quinpirole binding to human dopamine D2A receptor expressed in LtK cells | Bioorg Med Chem Lett 9: 2167-72 (1999) BindingDB Entry DOI: 10.7270/Q2CF9P97 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(2) dopamine receptor (Homo sapiens (Human)) | BDBM50053670 (((R)-5-Fluoro-1,2,3,4-tetrahydro-naphthalen-2-yl)-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 201 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Uppsala University Curated by ChEMBL | Assay Description Displacement of [3H]-raclopride from human dopamine D2A receptors expressed in LtK cells | Bioorg Med Chem Lett 9: 2167-72 (1999) BindingDB Entry DOI: 10.7270/Q2CF9P97 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(2) dopamine receptor (Homo sapiens (Human)) | BDBM50080050 (((R)-5-Methoxy-1,2,3,4-tetrahydro-naphthalen-2-yl)...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 215 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Uppsala University Curated by ChEMBL | Assay Description Displacement of [3H]-quinpirole from human dopamine D2A receptors expressed in LtK cells | Bioorg Med Chem Lett 9: 2167-72 (1999) BindingDB Entry DOI: 10.7270/Q2CF9P97 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(2) dopamine receptor (Homo sapiens (Human)) | BDBM50080049 (((R)-5-Methoxy-1,2,3,4-tetrahydro-naphthalen-2-yl)...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | PubMed | 339 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Uppsala University Curated by ChEMBL | Assay Description Displacement of [3H]-quinpirole from human dopamine D2A receptors expressed in LtK cells | Bioorg Med Chem Lett 9: 2167-72 (1999) BindingDB Entry DOI: 10.7270/Q2CF9P97 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(2) dopamine receptor (Homo sapiens (Human)) | BDBM50054337 (Benzyl-((R)-5-fluoro-1,2,3,4-tetrahydro-naphthalen...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 415 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Uppsala University Curated by ChEMBL | Assay Description Inhibition of [3H]-raclopride binding to human dopamine D2A receptor expressed in LtK cells | Bioorg Med Chem Lett 9: 2167-72 (1999) BindingDB Entry DOI: 10.7270/Q2CF9P97 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(2) dopamine receptor (Homo sapiens (Human)) | BDBM55121 (3-HYDROXYTYRAMINE HYDROCHLORIDE | 4-(2-aminoethyl)...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase DrugBank KEGG PC cid PC sid PDB UniChem Similars | DrugBank PubMed | 759 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Uppsala University Curated by ChEMBL | Assay Description Displacement of [3H]-raclopride from human dopamine D2A receptors expressed in LtK cells | Bioorg Med Chem Lett 9: 2167-72 (1999) BindingDB Entry DOI: 10.7270/Q2CF9P97 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(2) dopamine receptor (Homo sapiens (Human)) | BDBM50080056 (Benzyl-((R)-5-methoxy-1,2,3,4-tetrahydro-naphthale...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | 1.01E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Uppsala University Curated by ChEMBL | Assay Description Displacement of [3H]-raclopride from human dopamine D2A receptors expressed in LtK cells | Bioorg Med Chem Lett 9: 2167-72 (1999) BindingDB Entry DOI: 10.7270/Q2CF9P97 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(2) dopamine receptor (Homo sapiens (Human)) | BDBM50080056 (Benzyl-((R)-5-methoxy-1,2,3,4-tetrahydro-naphthale...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | 1.31E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Uppsala University Curated by ChEMBL | Assay Description Displacement of [3H]-quinpirole from human dopamine D2A receptors expressed in LtK cells | Bioorg Med Chem Lett 9: 2167-72 (1999) BindingDB Entry DOI: 10.7270/Q2CF9P97 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(2) dopamine receptor (Homo sapiens (Human)) | BDBM50080054 (CHEMBL69705 | Dibenzyl-((R)-5-methoxy-1,2,3,4-tetr...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | >5.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Uppsala University Curated by ChEMBL | Assay Description Displacement of [3H]-quinpirole from human dopamine D2A receptors expressed in LtK cells | Bioorg Med Chem Lett 9: 2167-72 (1999) BindingDB Entry DOI: 10.7270/Q2CF9P97 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(2) dopamine receptor (Homo sapiens (Human)) | BDBM50080054 (CHEMBL69705 | Dibenzyl-((R)-5-methoxy-1,2,3,4-tetr...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | >5.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Uppsala University Curated by ChEMBL | Assay Description Displacement of [3H]-raclopride from human dopamine D2A receptors expressed in LtK cells | Bioorg Med Chem Lett 9: 2167-72 (1999) BindingDB Entry DOI: 10.7270/Q2CF9P97 | |||||||||||
More data for this Ligand-Target Pair |