Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Diacylglycerol O-acyltransferase 1 (Homo sapiens (Human)) | BDBM50436848 (CHEMBL2403617) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 10 | n/a | n/a | n/a | n/a | n/a | n/a |
Piramal Enterprises Limited Curated by ChEMBL | Assay Description Inhibition of human DGAT1 using [14C]-oleoylCoA/diolein as substrate assessed as formation of [14C]triglyceride after 10 mins by scintillation counti... | Eur J Med Chem 65: 337-47 (2013) Article DOI: 10.1016/j.ejmech.2013.05.006 BindingDB Entry DOI: 10.7270/Q2QJ7JPW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Diacylglycerol O-acyltransferase 1 (Homo sapiens (Human)) | BDBM50354642 (CHEMBL1834204) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 14 | n/a | n/a | n/a | n/a | n/a | n/a |
Piramal Life Sciences Limited Curated by ChEMBL | Assay Description Inhibition of human DGAT1 assessed as formation of [14C]-triglyceride using [14C]oleoyl-CoA by liquid scintillation counting | Bioorg Med Chem Lett 21: 5812-7 (2011) Article DOI: 10.1016/j.bmcl.2011.07.109 BindingDB Entry DOI: 10.7270/Q28G8M29 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Diacylglycerol O-acyltransferase 1 (Homo sapiens (Human)) | BDBM50354637 (CHEMBL1834440) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 14 | n/a | n/a | n/a | n/a | n/a | n/a |
Piramal Life Sciences Limited Curated by ChEMBL | Assay Description Inhibition of human DGAT1 assessed as formation of [14C]-triglyceride using [14C]oleoyl-CoA by liquid scintillation counting | Bioorg Med Chem Lett 21: 5812-7 (2011) Article DOI: 10.1016/j.bmcl.2011.07.109 BindingDB Entry DOI: 10.7270/Q28G8M29 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Diacylglycerol O-acyltransferase 1 (Homo sapiens (Human)) | BDBM50436846 (CHEMBL2403620) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 16 | n/a | n/a | n/a | n/a | n/a | n/a |
Piramal Enterprises Limited Curated by ChEMBL | Assay Description Inhibition of human DGAT1 using [14C]-oleoylCoA/diolein as substrate assessed as formation of [14C]triglyceride after 10 mins by scintillation counti... | Eur J Med Chem 65: 337-47 (2013) Article DOI: 10.1016/j.ejmech.2013.05.006 BindingDB Entry DOI: 10.7270/Q2QJ7JPW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Diacylglycerol O-acyltransferase 1 (Homo sapiens (Human)) | BDBM50354639 (CHEMBL1834201) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 17 | n/a | n/a | n/a | n/a | n/a | n/a |
Piramal Life Sciences Limited Curated by ChEMBL | Assay Description Inhibition of human DGAT1 assessed as formation of [14C]-triglyceride using [14C]oleoyl-CoA by liquid scintillation counting | Bioorg Med Chem Lett 21: 5812-7 (2011) Article DOI: 10.1016/j.bmcl.2011.07.109 BindingDB Entry DOI: 10.7270/Q28G8M29 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Diacylglycerol O-acyltransferase 1 (Homo sapiens (Human)) | BDBM50354638 (CHEMBL1834200) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 18 | n/a | n/a | n/a | n/a | n/a | n/a |
Piramal Life Sciences Limited Curated by ChEMBL | Assay Description Inhibition of human DGAT1 assessed as formation of [14C]-triglyceride using [14C]oleoyl-CoA by liquid scintillation counting | Bioorg Med Chem Lett 21: 5812-7 (2011) Article DOI: 10.1016/j.bmcl.2011.07.109 BindingDB Entry DOI: 10.7270/Q28G8M29 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Xanthine dehydrogenase/oxidase (Homo sapiens (Human)) | BDBM50402272 (CHEMBL2205509) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 20 | n/a | n/a | n/a | n/a | n/a | n/a |
Piramal Healthcare Limited Curated by ChEMBL | Assay Description Inhibition of xanthine oxidase using xanthine as substrate at 30 mins by spectrophotometric analysis | Bioorg Med Chem Lett 22: 7543-6 (2012) Article DOI: 10.1016/j.bmcl.2012.10.029 BindingDB Entry DOI: 10.7270/Q2445NNH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Diacylglycerol O-acyltransferase 1 (Homo sapiens (Human)) | BDBM50436845 (CHEMBL2403621) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 20 | n/a | n/a | n/a | n/a | n/a | n/a |
Piramal Enterprises Limited Curated by ChEMBL | Assay Description Inhibition of human DGAT1 using [14C]-oleoylCoA/diolein as substrate assessed as formation of [14C]triglyceride after 10 mins by scintillation counti... | Eur J Med Chem 65: 337-47 (2013) Article DOI: 10.1016/j.ejmech.2013.05.006 BindingDB Entry DOI: 10.7270/Q2QJ7JPW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Diacylglycerol O-acyltransferase 1 (Homo sapiens (Human)) | BDBM20716 ((1R,2R)-2-[(4-{4-[(phenylcarbamoyl)amino]phenyl}ph...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 20 | n/a | n/a | n/a | n/a | n/a | n/a |
Piramal Life Sciences Limited Curated by ChEMBL | Assay Description Inhibition of human DGAT1 assessed as formation of [14C]-triglyceride using [14C]oleoyl-CoA by liquid scintillation counting | Bioorg Med Chem Lett 21: 5812-7 (2011) Article DOI: 10.1016/j.bmcl.2011.07.109 BindingDB Entry DOI: 10.7270/Q28G8M29 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Diacylglycerol O-acyltransferase 1 (Homo sapiens (Human)) | BDBM20716 ((1R,2R)-2-[(4-{4-[(phenylcarbamoyl)amino]phenyl}ph...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 20 | n/a | n/a | n/a | n/a | n/a | n/a |
Piramal Life Sciences Limited Curated by ChEMBL | Assay Description Inhibition of human DGAT1 expressed in Sf9 cells assessed as formation of didecanoylglycerol product after 1 hr using 14C-decanoyl-CoA by beta scinti... | Bioorg Med Chem Lett 21: 5812-7 (2011) Article DOI: 10.1016/j.bmcl.2011.07.109 BindingDB Entry DOI: 10.7270/Q28G8M29 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Diacylglycerol O-acyltransferase 1 (Homo sapiens (Human)) | BDBM50436847 (CHEMBL2403619) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 22 | n/a | n/a | n/a | n/a | n/a | n/a |
Piramal Enterprises Limited Curated by ChEMBL | Assay Description Inhibition of human DGAT1 using [14C]-oleoylCoA/diolein as substrate assessed as formation of [14C]triglyceride after 10 mins by scintillation counti... | Eur J Med Chem 65: 337-47 (2013) Article DOI: 10.1016/j.ejmech.2013.05.006 BindingDB Entry DOI: 10.7270/Q2QJ7JPW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Diacylglycerol O-acyltransferase 1 (Homo sapiens (Human)) | BDBM50436842 (CHEMBL2403624) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 23 | n/a | n/a | n/a | n/a | n/a | n/a |
Piramal Enterprises Limited Curated by ChEMBL | Assay Description Inhibition of human DGAT1 using [14C]-oleoylCoA/diolein as substrate assessed as formation of [14C]triglyceride after 10 mins by scintillation counti... | Eur J Med Chem 65: 337-47 (2013) Article DOI: 10.1016/j.ejmech.2013.05.006 BindingDB Entry DOI: 10.7270/Q2QJ7JPW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Diacylglycerol O-acyltransferase 1 (Homo sapiens (Human)) | BDBM50436844 (CHEMBL2403622) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 23 | n/a | n/a | n/a | n/a | n/a | n/a |
Piramal Enterprises Limited Curated by ChEMBL | Assay Description Inhibition of human DGAT1 using [14C]-oleoylCoA/diolein as substrate assessed as formation of [14C]triglyceride after 10 mins by scintillation counti... | Eur J Med Chem 65: 337-47 (2013) Article DOI: 10.1016/j.ejmech.2013.05.006 BindingDB Entry DOI: 10.7270/Q2QJ7JPW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Diacylglycerol O-acyltransferase 1 (Homo sapiens (Human)) | BDBM50354641 (CHEMBL1834203) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 25 | n/a | n/a | n/a | n/a | n/a | n/a |
Piramal Life Sciences Limited Curated by ChEMBL | Assay Description Inhibition of human DGAT1 assessed as formation of [14C]-triglyceride using [14C]oleoyl-CoA by liquid scintillation counting | Bioorg Med Chem Lett 21: 5812-7 (2011) Article DOI: 10.1016/j.bmcl.2011.07.109 BindingDB Entry DOI: 10.7270/Q28G8M29 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Diacylglycerol O-acyltransferase 1 (Homo sapiens (Human)) | BDBM50354631 (CHEMBL1834433) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 28 | n/a | n/a | n/a | n/a | n/a | n/a |
Piramal Life Sciences Limited Curated by ChEMBL | Assay Description Inhibition of human DGAT1 assessed as formation of [14C]-triglyceride using [14C]oleoyl-CoA by liquid scintillation counting | Bioorg Med Chem Lett 21: 5812-7 (2011) Article DOI: 10.1016/j.bmcl.2011.07.109 BindingDB Entry DOI: 10.7270/Q28G8M29 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Diacylglycerol O-acyltransferase 1 (Homo sapiens (Human)) | BDBM50354629 (CHEMBL1834431) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 30 | n/a | n/a | n/a | n/a | n/a | n/a |
Piramal Life Sciences Limited Curated by ChEMBL | Assay Description Inhibition of human DGAT1 assessed as formation of [14C]-triglyceride using [14C]oleoyl-CoA by liquid scintillation counting | Bioorg Med Chem Lett 21: 5812-7 (2011) Article DOI: 10.1016/j.bmcl.2011.07.109 BindingDB Entry DOI: 10.7270/Q28G8M29 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Xanthine dehydrogenase/oxidase (Homo sapiens (Human)) | BDBM50320491 (2-(3-CYANO-4-ISOBUTOXY-PHENYL)-4-METHYL-5-THIAZOLE...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE MMDB PC cid PC sid PDB UniChem Patents | MMDB PDB Article PubMed | n/a | n/a | 30 | n/a | n/a | n/a | n/a | n/a | n/a |
Piramal Healthcare Limited Curated by ChEMBL | Assay Description Inhibition of xanthine oxidase using xanthine as substrate at 30 mins by spectrophotometric analysis | Bioorg Med Chem Lett 22: 7543-6 (2012) Article DOI: 10.1016/j.bmcl.2012.10.029 BindingDB Entry DOI: 10.7270/Q2445NNH | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Diacylglycerol O-acyltransferase 1 (Homo sapiens (Human)) | BDBM50354634 (CHEMBL1834436) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 32 | n/a | n/a | n/a | n/a | n/a | n/a |
Piramal Life Sciences Limited Curated by ChEMBL | Assay Description Inhibition of human DGAT1 assessed as formation of [14C]-triglyceride using [14C]oleoyl-CoA by liquid scintillation counting | Bioorg Med Chem Lett 21: 5812-7 (2011) Article DOI: 10.1016/j.bmcl.2011.07.109 BindingDB Entry DOI: 10.7270/Q28G8M29 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Diacylglycerol O-acyltransferase 1 (Homo sapiens (Human)) | BDBM50386149 (CHEMBL2042351) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 35 | n/a | n/a | n/a | n/a | n/a | n/a |
Piramal Enterprises Limited Curated by ChEMBL | Assay Description Inhibition of human DGAT1 | Eur J Med Chem 65: 337-47 (2013) Article DOI: 10.1016/j.ejmech.2013.05.006 BindingDB Entry DOI: 10.7270/Q2QJ7JPW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Diacylglycerol O-acyltransferase 1 (Homo sapiens (Human)) | BDBM50436841 (CHEMBL2403625) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 37 | n/a | n/a | n/a | n/a | n/a | n/a |
Piramal Enterprises Limited Curated by ChEMBL | Assay Description Inhibition of human DGAT1 using [14C]-oleoylCoA/diolein as substrate assessed as formation of [14C]triglyceride after 10 mins by scintillation counti... | Eur J Med Chem 65: 337-47 (2013) Article DOI: 10.1016/j.ejmech.2013.05.006 BindingDB Entry DOI: 10.7270/Q2QJ7JPW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Diacylglycerol O-acyltransferase 1 (Homo sapiens (Human)) | BDBM50436839 (CHEMBL2403627) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 49 | n/a | n/a | n/a | n/a | n/a | n/a |
Piramal Enterprises Limited Curated by ChEMBL | Assay Description Inhibition of human DGAT1 using [14C]-oleoylCoA/diolein as substrate assessed as formation of [14C]triglyceride after 10 mins by scintillation counti... | Eur J Med Chem 65: 337-47 (2013) Article DOI: 10.1016/j.ejmech.2013.05.006 BindingDB Entry DOI: 10.7270/Q2QJ7JPW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Diacylglycerol O-acyltransferase 1 (Homo sapiens (Human)) | BDBM50354633 (CHEMBL1834435) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 51 | n/a | n/a | n/a | n/a | n/a | n/a |
Piramal Life Sciences Limited Curated by ChEMBL | Assay Description Inhibition of human DGAT1 assessed as formation of [14C]-triglyceride using [14C]oleoyl-CoA by liquid scintillation counting | Bioorg Med Chem Lett 21: 5812-7 (2011) Article DOI: 10.1016/j.bmcl.2011.07.109 BindingDB Entry DOI: 10.7270/Q28G8M29 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Diacylglycerol O-acyltransferase 1 (Homo sapiens (Human)) | BDBM50354636 (CHEMBL1834438) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 57 | n/a | n/a | n/a | n/a | n/a | n/a |
Piramal Life Sciences Limited Curated by ChEMBL | Assay Description Inhibition of human DGAT1 assessed as formation of [14C]-triglyceride using [14C]oleoyl-CoA by liquid scintillation counting | Bioorg Med Chem Lett 21: 5812-7 (2011) Article DOI: 10.1016/j.bmcl.2011.07.109 BindingDB Entry DOI: 10.7270/Q28G8M29 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Diacylglycerol O-acyltransferase 1 (Homo sapiens (Human)) | BDBM50436843 (CHEMBL2403623) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 58 | n/a | n/a | n/a | n/a | n/a | n/a |
Piramal Enterprises Limited Curated by ChEMBL | Assay Description Inhibition of human DGAT1 using [14C]-oleoylCoA/diolein as substrate assessed as formation of [14C]triglyceride after 10 mins by scintillation counti... | Eur J Med Chem 65: 337-47 (2013) Article DOI: 10.1016/j.ejmech.2013.05.006 BindingDB Entry DOI: 10.7270/Q2QJ7JPW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Diacylglycerol O-acyltransferase 1 (Homo sapiens (Human)) | BDBM50354640 (CHEMBL1834202) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 64 | n/a | n/a | n/a | n/a | n/a | n/a |
Piramal Life Sciences Limited Curated by ChEMBL | Assay Description Inhibition of human DGAT1 assessed as formation of [14C]-triglyceride using [14C]oleoyl-CoA by liquid scintillation counting | Bioorg Med Chem Lett 21: 5812-7 (2011) Article DOI: 10.1016/j.bmcl.2011.07.109 BindingDB Entry DOI: 10.7270/Q28G8M29 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Diacylglycerol O-acyltransferase 1 (Homo sapiens (Human)) | BDBM50354630 (CHEMBL1834432) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 72 | n/a | n/a | n/a | n/a | n/a | n/a |
Piramal Life Sciences Limited Curated by ChEMBL | Assay Description Inhibition of human DGAT1 assessed as formation of [14C]-triglyceride using [14C]oleoyl-CoA by liquid scintillation counting | Bioorg Med Chem Lett 21: 5812-7 (2011) Article DOI: 10.1016/j.bmcl.2011.07.109 BindingDB Entry DOI: 10.7270/Q28G8M29 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Diacylglycerol O-acyltransferase 1 (Homo sapiens (Human)) | BDBM50354643 (CHEMBL1834206) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 73 | n/a | n/a | n/a | n/a | n/a | n/a |
Piramal Life Sciences Limited Curated by ChEMBL | Assay Description Inhibition of human DGAT1 expressed in Sf9 cells assessed as formation of didecanoylglycerol product after 1 hr using 14C-decanoyl-CoA by beta scinti... | Bioorg Med Chem Lett 21: 5812-7 (2011) Article DOI: 10.1016/j.bmcl.2011.07.109 BindingDB Entry DOI: 10.7270/Q28G8M29 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Diacylglycerol O-acyltransferase 1 (Homo sapiens (Human)) | BDBM50436840 (CHEMBL2403626) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 82 | n/a | n/a | n/a | n/a | n/a | n/a |
Piramal Enterprises Limited Curated by ChEMBL | Assay Description Inhibition of human DGAT1 using [14C]-oleoylCoA/diolein as substrate assessed as formation of [14C]triglyceride after 10 mins by scintillation counti... | Eur J Med Chem 65: 337-47 (2013) Article DOI: 10.1016/j.ejmech.2013.05.006 BindingDB Entry DOI: 10.7270/Q2QJ7JPW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Diacylglycerol O-acyltransferase 1 (Homo sapiens (Human)) | BDBM50354632 (CHEMBL1834434) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 88 | n/a | n/a | n/a | n/a | n/a | n/a |
Piramal Life Sciences Limited Curated by ChEMBL | Assay Description Inhibition of human DGAT1 assessed as formation of [14C]-triglyceride using [14C]oleoyl-CoA by liquid scintillation counting | Bioorg Med Chem Lett 21: 5812-7 (2011) Article DOI: 10.1016/j.bmcl.2011.07.109 BindingDB Entry DOI: 10.7270/Q28G8M29 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Diacylglycerol O-acyltransferase 1 (Homo sapiens (Human)) | BDBM50436838 (CHEMBL2403628) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 97 | n/a | n/a | n/a | n/a | n/a | n/a |
Piramal Enterprises Limited Curated by ChEMBL | Assay Description Inhibition of human DGAT1 using [14C]-oleoylCoA/diolein as substrate assessed as formation of [14C]triglyceride after 10 mins by scintillation counti... | Eur J Med Chem 65: 337-47 (2013) Article DOI: 10.1016/j.ejmech.2013.05.006 BindingDB Entry DOI: 10.7270/Q2QJ7JPW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Diacylglycerol O-acyltransferase 1 (Homo sapiens (Human)) | BDBM50354635 (CHEMBL1834437) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 99 | n/a | n/a | n/a | n/a | n/a | n/a |
Piramal Life Sciences Limited Curated by ChEMBL | Assay Description Inhibition of human DGAT1 assessed as formation of [14C]-triglyceride using [14C]oleoyl-CoA by liquid scintillation counting | Bioorg Med Chem Lett 21: 5812-7 (2011) Article DOI: 10.1016/j.bmcl.2011.07.109 BindingDB Entry DOI: 10.7270/Q28G8M29 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Diacylglycerol O-acyltransferase 1 (Homo sapiens (Human)) | BDBM50436837 (CHEMBL2403629) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 101 | n/a | n/a | n/a | n/a | n/a | n/a |
Piramal Enterprises Limited Curated by ChEMBL | Assay Description Inhibition of human DGAT1 using [14C]-oleoylCoA/diolein as substrate assessed as formation of [14C]triglyceride after 10 mins by scintillation counti... | Eur J Med Chem 65: 337-47 (2013) Article DOI: 10.1016/j.ejmech.2013.05.006 BindingDB Entry DOI: 10.7270/Q2QJ7JPW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Xanthine dehydrogenase/oxidase (Homo sapiens (Human)) | BDBM50402273 (CHEMBL2205508) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 140 | n/a | n/a | n/a | n/a | n/a | n/a |
Piramal Healthcare Limited Curated by ChEMBL | Assay Description Inhibition of xanthine oxidase using xanthine as substrate at 30 mins by spectrophotometric analysis | Bioorg Med Chem Lett 22: 7543-6 (2012) Article DOI: 10.1016/j.bmcl.2012.10.029 BindingDB Entry DOI: 10.7270/Q2445NNH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Xanthine dehydrogenase/oxidase (Homo sapiens (Human)) | BDBM50402280 (CHEMBL2205501) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 310 | n/a | n/a | n/a | n/a | n/a | n/a |
Piramal Healthcare Limited Curated by ChEMBL | Assay Description Inhibition of xanthine oxidase using xanthine as substrate at 30 mins by spectrophotometric analysis | Bioorg Med Chem Lett 22: 7543-6 (2012) Article DOI: 10.1016/j.bmcl.2012.10.029 BindingDB Entry DOI: 10.7270/Q2445NNH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Xanthine dehydrogenase/oxidase (Homo sapiens (Human)) | BDBM50402288 (CHEMBL2205498) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 600 | n/a | n/a | n/a | n/a | n/a | n/a |
Piramal Healthcare Limited Curated by ChEMBL | Assay Description Inhibition of xanthine oxidase using xanthine as substrate at 30 mins by spectrophotometric analysis | Bioorg Med Chem Lett 22: 7543-6 (2012) Article DOI: 10.1016/j.bmcl.2012.10.029 BindingDB Entry DOI: 10.7270/Q2445NNH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Xanthine dehydrogenase/oxidase (Homo sapiens (Human)) | BDBM50402274 (CHEMBL2205507) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 950 | n/a | n/a | n/a | n/a | n/a | n/a |
Piramal Healthcare Limited Curated by ChEMBL | Assay Description Inhibition of xanthine oxidase using xanthine as substrate at 30 mins by spectrophotometric analysis | Bioorg Med Chem Lett 22: 7543-6 (2012) Article DOI: 10.1016/j.bmcl.2012.10.029 BindingDB Entry DOI: 10.7270/Q2445NNH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Xanthine dehydrogenase/oxidase (Bos taurus (Bovine)) | BDBM50381872 (CHEMBL2022883) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.40E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Piramal Healthcare Limited Curated by ChEMBL | Assay Description Inhibition of bovine xanthine oxidase assessed as uric acid formation using xanthine as substrate after 30 mins by spectrophotometric analysis | Bioorg Med Chem 20: 2930-9 (2012) Article DOI: 10.1016/j.bmc.2012.03.019 BindingDB Entry DOI: 10.7270/Q2Z320NM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Xanthine dehydrogenase/oxidase (Homo sapiens (Human)) | BDBM50402284 (CHEMBL2205495) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.63E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Piramal Healthcare Limited Curated by ChEMBL | Assay Description Inhibition of xanthine oxidase using xanthine as substrate at 30 mins by spectrophotometric analysis | Bioorg Med Chem Lett 22: 7543-6 (2012) Article DOI: 10.1016/j.bmcl.2012.10.029 BindingDB Entry DOI: 10.7270/Q2445NNH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Xanthine dehydrogenase/oxidase (Homo sapiens (Human)) | BDBM50402275 (CHEMBL2205506) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.92E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Piramal Healthcare Limited Curated by ChEMBL | Assay Description Inhibition of xanthine oxidase using xanthine as substrate at 30 mins by spectrophotometric analysis | Bioorg Med Chem Lett 22: 7543-6 (2012) Article DOI: 10.1016/j.bmcl.2012.10.029 BindingDB Entry DOI: 10.7270/Q2445NNH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Xanthine dehydrogenase/oxidase (Homo sapiens (Human)) | BDBM50402287 (CHEMBL2205497) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Piramal Healthcare Limited Curated by ChEMBL | Assay Description Inhibition of xanthine oxidase using xanthine as substrate at 30 mins by spectrophotometric analysis | Bioorg Med Chem Lett 22: 7543-6 (2012) Article DOI: 10.1016/j.bmcl.2012.10.029 BindingDB Entry DOI: 10.7270/Q2445NNH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Xanthine dehydrogenase/oxidase (Homo sapiens (Human)) | BDBM50402286 (CHEMBL2205496) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.44E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Piramal Healthcare Limited Curated by ChEMBL | Assay Description Inhibition of xanthine oxidase using xanthine as substrate at 30 mins by spectrophotometric analysis | Bioorg Med Chem Lett 22: 7543-6 (2012) Article DOI: 10.1016/j.bmcl.2012.10.029 BindingDB Entry DOI: 10.7270/Q2445NNH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Xanthine dehydrogenase/oxidase (Homo sapiens (Human)) | BDBM50402278 (CHEMBL2205503) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.47E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Piramal Healthcare Limited Curated by ChEMBL | Assay Description Inhibition of xanthine oxidase using xanthine as substrate at 30 mins by spectrophotometric analysis | Bioorg Med Chem Lett 22: 7543-6 (2012) Article DOI: 10.1016/j.bmcl.2012.10.029 BindingDB Entry DOI: 10.7270/Q2445NNH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Xanthine dehydrogenase/oxidase (Homo sapiens (Human)) | BDBM50402281 (CHEMBL2205502) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.65E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Piramal Healthcare Limited Curated by ChEMBL | Assay Description Inhibition of xanthine oxidase using xanthine as substrate at 30 mins by spectrophotometric analysis | Bioorg Med Chem Lett 22: 7543-6 (2012) Article DOI: 10.1016/j.bmcl.2012.10.029 BindingDB Entry DOI: 10.7270/Q2445NNH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Xanthine dehydrogenase/oxidase (Homo sapiens (Human)) | BDBM35440 (ALLOPURINOL | MLS000069453 | SMR000059083 | cid_20...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 4.19E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Piramal Healthcare Limited Curated by ChEMBL | Assay Description Inhibition of xanthine oxidase using xanthine as substrate at 30 mins by spectrophotometric analysis | Bioorg Med Chem Lett 22: 7543-6 (2012) Article DOI: 10.1016/j.bmcl.2012.10.029 BindingDB Entry DOI: 10.7270/Q2445NNH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Xanthine dehydrogenase/oxidase (Homo sapiens (Human)) | BDBM50402283 (CHEMBL2205494) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 4.95E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Piramal Healthcare Limited Curated by ChEMBL | Assay Description Inhibition of xanthine oxidase using xanthine as substrate at 30 mins by spectrophotometric analysis | Bioorg Med Chem Lett 22: 7543-6 (2012) Article DOI: 10.1016/j.bmcl.2012.10.029 BindingDB Entry DOI: 10.7270/Q2445NNH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Xanthine dehydrogenase/oxidase (Bos taurus (Bovine)) | BDBM35440 (ALLOPURINOL | MLS000069453 | SMR000059083 | cid_20...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 5.70E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Piramal Healthcare Limited Curated by ChEMBL | Assay Description Inhibition of bovine xanthine oxidase assessed as uric acid formation using xanthine as substrate after 30 mins by spectrophotometric analysis | Bioorg Med Chem 20: 2930-9 (2012) Article DOI: 10.1016/j.bmc.2012.03.019 BindingDB Entry DOI: 10.7270/Q2Z320NM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Xanthine dehydrogenase/oxidase (Homo sapiens (Human)) | BDBM50402276 (CHEMBL2205505) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 6.72E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Piramal Healthcare Limited Curated by ChEMBL | Assay Description Inhibition of xanthine oxidase using xanthine as substrate at 30 mins by spectrophotometric analysis | Bioorg Med Chem Lett 22: 7543-6 (2012) Article DOI: 10.1016/j.bmcl.2012.10.029 BindingDB Entry DOI: 10.7270/Q2445NNH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Xanthine dehydrogenase/oxidase (Homo sapiens (Human)) | BDBM50402285 (CHEMBL2205499) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 9.24E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Piramal Healthcare Limited Curated by ChEMBL | Assay Description Inhibition of xanthine oxidase using xanthine as substrate at 30 mins by spectrophotometric analysis | Bioorg Med Chem Lett 22: 7543-6 (2012) Article DOI: 10.1016/j.bmcl.2012.10.029 BindingDB Entry DOI: 10.7270/Q2445NNH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Xanthine dehydrogenase/oxidase (Bos taurus (Bovine)) | BDBM50381870 (CHEMBL2022881) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 9.40E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Piramal Healthcare Limited Curated by ChEMBL | Assay Description Inhibition of bovine xanthine oxidase assessed as uric acid formation using xanthine as substrate after 30 mins by spectrophotometric analysis | Bioorg Med Chem 20: 2930-9 (2012) Article DOI: 10.1016/j.bmc.2012.03.019 BindingDB Entry DOI: 10.7270/Q2Z320NM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Xanthine dehydrogenase/oxidase (Homo sapiens (Human)) | BDBM50402279 (CHEMBL2205500) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.65E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Piramal Healthcare Limited Curated by ChEMBL | Assay Description Inhibition of xanthine oxidase using xanthine as substrate at 30 mins by spectrophotometric analysis | Bioorg Med Chem Lett 22: 7543-6 (2012) Article DOI: 10.1016/j.bmcl.2012.10.029 BindingDB Entry DOI: 10.7270/Q2445NNH | |||||||||||
More data for this Ligand-Target Pair |
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