Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Trace amine-associated receptor 1 (Mus musculus (Mouse)) | BDBM10758 (14C-phenylethylamine | 2-phenylethan-1-amine | CHE...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE KEGG MMDB PC cid PC sid PDB UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 138 | n/a | n/a | n/a | n/a |
University of Pisa Curated by ChEMBL | Assay Description Agonist activity at mouse TAAR1 expressed in HEK293 cells coexpressing cAMP BRET biosensor assessed as induction of CAMP production after 20 mins by ... | J Med Chem 58: 5096-107 (2015) Article DOI: 10.1021/acs.jmedchem.5b00526 BindingDB Entry DOI: 10.7270/Q2PC3446 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Trace amine-associated receptor 1 (Mus musculus (Mouse)) | BDBM50359505 (CHEMBL1182312) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid PDB UniChem Patents Similars | PDB Article PubMed | n/a | n/a | n/a | n/a | 189 | n/a | n/a | n/a | n/a |
University of Pisa Curated by ChEMBL | Assay Description Agonist activity at mouse TAAR1 expressed in HEK293 cells coexpressing cAMP BRET biosensor assessed as induction of CAMP production after 20 mins by ... | J Med Chem 58: 5096-107 (2015) Article DOI: 10.1021/acs.jmedchem.5b00526 BindingDB Entry DOI: 10.7270/Q2PC3446 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Trace amine-associated receptor 1 (Mus musculus (Mouse)) | BDBM50096963 (CHEMBL3580902) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 240 | n/a | n/a | n/a | n/a |
University of Pisa Curated by ChEMBL | Assay Description Agonist activity at mouse TAAR1 expressed in HEK293 cells coexpressing cAMP BRET biosensor assessed as induction of CAMP production after 20 mins by ... | J Med Chem 58: 5096-107 (2015) Article DOI: 10.1021/acs.jmedchem.5b00526 BindingDB Entry DOI: 10.7270/Q2PC3446 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Trace amine-associated receptor 1 (Mus musculus (Mouse)) | BDBM50096964 (CHEMBL3580901) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.70E+3 | n/a | n/a | n/a | n/a |
University of Pisa Curated by ChEMBL | Assay Description Agonist activity at mouse TAAR1 expressed in HEK293 cells coexpressing cAMP BRET biosensor assessed as induction of CAMP production after 20 mins by ... | J Med Chem 58: 5096-107 (2015) Article DOI: 10.1021/acs.jmedchem.5b00526 BindingDB Entry DOI: 10.7270/Q2PC3446 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Trace amine-associated receptor 1 (Mus musculus (Mouse)) | BDBM50096965 (CHEMBL3580905) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 800 | n/a | n/a | n/a | n/a |
University of Pisa Curated by ChEMBL | Assay Description Agonist activity at mouse TAAR1 expressed in HEK293 cells coexpressing cAMP BRET biosensor assessed as induction of CAMP production after 20 mins by ... | J Med Chem 58: 5096-107 (2015) Article DOI: 10.1021/acs.jmedchem.5b00526 BindingDB Entry DOI: 10.7270/Q2PC3446 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Trace amine-associated receptor 1 (Mus musculus (Mouse)) | BDBM50096966 (CHEMBL3580906) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 2.20E+3 | n/a | n/a | n/a | n/a |
University of Pisa Curated by ChEMBL | Assay Description Agonist activity at mouse TAAR1 expressed in HEK293 cells coexpressing cAMP BRET biosensor assessed as induction of CAMP production after 20 mins by ... | J Med Chem 58: 5096-107 (2015) Article DOI: 10.1021/acs.jmedchem.5b00526 BindingDB Entry DOI: 10.7270/Q2PC3446 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Trace amine-associated receptor 1 (Homo sapiens (Human)) | BDBM50359505 (CHEMBL1182312) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid PDB UniChem Patents Similars | PDB Article PubMed | n/a | n/a | n/a | n/a | 1.69E+3 | n/a | n/a | n/a | n/a |
University of Genoa Curated by ChEMBL | Assay Description Inhibition of full length recombinant human N-terminal HA-tagged/C-terminal FLAG-tagged TAAR1 expressed in CHOK1 cells assessed as increase in cAMP a... | Eur J Med Chem 127: 781-792 (2017) Article DOI: 10.1016/j.ejmech.2016.10.058 BindingDB Entry DOI: 10.7270/Q2C24ZPS | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Trace amine-associated receptor 1 (Homo sapiens (Human)) | BDBM50053630 (4-Methyl-Phenyl biguanide | CHEMBL291064 | N-(4-me...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a |
University of Genoa Curated by ChEMBL | Assay Description Agonist activity at human TAAR1 expressed in HEK293 cells assessed as cAMP accumulation after 20 mins by BRET assay | Eur J Med Chem 127: 781-792 (2017) Article DOI: 10.1016/j.ejmech.2016.10.058 BindingDB Entry DOI: 10.7270/Q2C24ZPS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Trace amine-associated receptor 1 (Homo sapiens (Human)) | BDBM50227351 (CHEMBL3628706) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a |
University of Genoa Curated by ChEMBL | Assay Description Agonist activity at human TAAR1 expressed in HEK293 cells assessed as cAMP accumulation after 20 mins by BRET assay | Eur J Med Chem 127: 781-792 (2017) Article DOI: 10.1016/j.ejmech.2016.10.058 BindingDB Entry DOI: 10.7270/Q2C24ZPS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Trace amine-associated receptor 1 (Homo sapiens (Human)) | BDBM50227824 (CHEMBL4088689) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 7.00E+3 | n/a | n/a | n/a | n/a |
University of Genoa Curated by ChEMBL | Assay Description Agonist activity at human TAAR1 expressed in HEK293 cells assessed as cAMP accumulation after 20 mins by BRET assay | Eur J Med Chem 127: 781-792 (2017) Article DOI: 10.1016/j.ejmech.2016.10.058 BindingDB Entry DOI: 10.7270/Q2C24ZPS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Trace amine-associated receptor 1 (Homo sapiens (Human)) | BDBM50227825 (CHEMBL4060464) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.80E+3 | n/a | n/a | n/a | n/a |
University of Genoa Curated by ChEMBL | Assay Description Agonist activity at human TAAR1 expressed in HEK293 cells assessed as cAMP accumulation after 20 mins by BRET assay | Eur J Med Chem 127: 781-792 (2017) Article DOI: 10.1016/j.ejmech.2016.10.058 BindingDB Entry DOI: 10.7270/Q2C24ZPS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Trace amine-associated receptor 1 (Homo sapiens (Human)) | BDBM50227826 (CHEMBL4069147) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 1.60E+3 | n/a | n/a | n/a | n/a |
University of Genoa Curated by ChEMBL | Assay Description Agonist activity at human TAAR1 expressed in HEK293 cells assessed as cAMP accumulation after 20 mins by BRET assay | Eur J Med Chem 127: 781-792 (2017) Article DOI: 10.1016/j.ejmech.2016.10.058 BindingDB Entry DOI: 10.7270/Q2C24ZPS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Trace amine-associated receptor 1 (Homo sapiens (Human)) | BDBM50227828 (CHEMBL4068661) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 4.90E+3 | n/a | n/a | n/a | n/a |
University of Genoa Curated by ChEMBL | Assay Description Agonist activity at human TAAR1 expressed in HEK293 cells assessed as cAMP accumulation after 20 mins by BRET assay | Eur J Med Chem 127: 781-792 (2017) Article DOI: 10.1016/j.ejmech.2016.10.058 BindingDB Entry DOI: 10.7270/Q2C24ZPS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Trace amine-associated receptor 1 (Homo sapiens (Human)) | BDBM50227829 (CHEBI:8455 | CHLOROGUANIDE | Proguanil) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid PDB UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a |
University of Genoa Curated by ChEMBL | Assay Description Agonist activity at human TAAR1 expressed in HEK293 cells assessed as cAMP accumulation after 20 mins by BRET assay | Eur J Med Chem 127: 781-792 (2017) Article DOI: 10.1016/j.ejmech.2016.10.058 BindingDB Entry DOI: 10.7270/Q2C24ZPS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Trace amine-associated receptor 5 (Mus musculus) | BDBM50053629 (2-Chloro-Phenyl biguanide | CHEMBL42752 | N-(2-chl...) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a |
University of Genoa Curated by ChEMBL | Assay Description Agonist activity at mouse TAAR5 expressed in HEK293 cells assessed as cAMP accumulation after 20 mins by BRET assay | Eur J Med Chem 127: 781-792 (2017) Article DOI: 10.1016/j.ejmech.2016.10.058 BindingDB Entry DOI: 10.7270/Q2C24ZPS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Trace amine-associated receptor 5 (Mus musculus) | BDBM50053615 (3-Chloro-Phenyl biguanide | CHEMBL13790 | N-(3-chl...) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a |
University of Genoa Curated by ChEMBL | Assay Description Agonist activity at mouse TAAR5 expressed in HEK293 cells assessed as cAMP accumulation after 20 mins by BRET assay | Eur J Med Chem 127: 781-792 (2017) Article DOI: 10.1016/j.ejmech.2016.10.058 BindingDB Entry DOI: 10.7270/Q2C24ZPS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Trace amine-associated receptor 5 (Mus musculus) | BDBM50100977 (3,4-dichloro-phenylbiguanide | CHEMBL41433 | N-(3,...) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a |
University of Genoa Curated by ChEMBL | Assay Description Agonist activity at mouse TAAR5 expressed in HEK293 cells assessed as cAMP accumulation after 20 mins by BRET assay | Eur J Med Chem 127: 781-792 (2017) Article DOI: 10.1016/j.ejmech.2016.10.058 BindingDB Entry DOI: 10.7270/Q2C24ZPS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Trace amine-associated receptor 5 (Mus musculus) | BDBM50227830 (CHEMBL4099661) | UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a |
University of Genoa Curated by ChEMBL | Assay Description Agonist activity at mouse TAAR5 expressed in HEK293 cells assessed as cAMP accumulation after 20 mins by BRET assay | Eur J Med Chem 127: 781-792 (2017) Article DOI: 10.1016/j.ejmech.2016.10.058 BindingDB Entry DOI: 10.7270/Q2C24ZPS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Trace amine-associated receptor 5 (Mus musculus) | BDBM50227833 (CHEMBL4088381) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a |
University of Genoa Curated by ChEMBL | Assay Description Agonist activity at mouse TAAR5 expressed in HEK293 cells assessed as cAMP accumulation after 20 mins by BRET assay | Eur J Med Chem 127: 781-792 (2017) Article DOI: 10.1016/j.ejmech.2016.10.058 BindingDB Entry DOI: 10.7270/Q2C24ZPS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Trace amine-associated receptor 5 (Mus musculus) | BDBM50227834 (CHEMBL4077681) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a |
University of Genoa Curated by ChEMBL | Assay Description Agonist activity at mouse TAAR5 expressed in HEK293 cells assessed as cAMP accumulation after 20 mins by BRET assay | Eur J Med Chem 127: 781-792 (2017) Article DOI: 10.1016/j.ejmech.2016.10.058 BindingDB Entry DOI: 10.7270/Q2C24ZPS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Trace amine-associated receptor 5 (Mus musculus) | BDBM50227351 (CHEMBL3628706) | UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a |
University of Genoa Curated by ChEMBL | Assay Description Agonist activity at mouse TAAR5 expressed in HEK293 cells assessed as cAMP accumulation after 20 mins by BRET assay | Eur J Med Chem 127: 781-792 (2017) Article DOI: 10.1016/j.ejmech.2016.10.058 BindingDB Entry DOI: 10.7270/Q2C24ZPS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Trace amine-associated receptor 5 (Mus musculus) | BDBM50227824 (CHEMBL4088689) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a |
University of Genoa Curated by ChEMBL | Assay Description Agonist activity at mouse TAAR5 expressed in HEK293 cells assessed as cAMP accumulation after 20 mins by BRET assay | Eur J Med Chem 127: 781-792 (2017) Article DOI: 10.1016/j.ejmech.2016.10.058 BindingDB Entry DOI: 10.7270/Q2C24ZPS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Trace amine-associated receptor 5 (Mus musculus) | BDBM50227825 (CHEMBL4060464) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a |
University of Genoa Curated by ChEMBL | Assay Description Agonist activity at mouse TAAR5 expressed in HEK293 cells assessed as cAMP accumulation after 20 mins by BRET assay | Eur J Med Chem 127: 781-792 (2017) Article DOI: 10.1016/j.ejmech.2016.10.058 BindingDB Entry DOI: 10.7270/Q2C24ZPS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Trace amine-associated receptor 5 (Mus musculus) | BDBM50227835 (CHEMBL4096403) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a |
University of Genoa Curated by ChEMBL | Assay Description Agonist activity at mouse TAAR5 expressed in HEK293 cells assessed as cAMP accumulation after 20 mins by BRET assay | Eur J Med Chem 127: 781-792 (2017) Article DOI: 10.1016/j.ejmech.2016.10.058 BindingDB Entry DOI: 10.7270/Q2C24ZPS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Trace amine-associated receptor 5 (Mus musculus) | BDBM50227828 (CHEMBL4068661) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a |
University of Genoa Curated by ChEMBL | Assay Description Agonist activity at mouse TAAR5 expressed in HEK293 cells assessed as cAMP accumulation after 20 mins by BRET assay | Eur J Med Chem 127: 781-792 (2017) Article DOI: 10.1016/j.ejmech.2016.10.058 BindingDB Entry DOI: 10.7270/Q2C24ZPS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Trace amine-associated receptor 5 (Mus musculus) | BDBM50227836 (CHEMBL4076103) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a |
University of Genoa Curated by ChEMBL | Assay Description Agonist activity at mouse TAAR5 expressed in HEK293 cells assessed as cAMP accumulation after 20 mins by BRET assay | Eur J Med Chem 127: 781-792 (2017) Article DOI: 10.1016/j.ejmech.2016.10.058 BindingDB Entry DOI: 10.7270/Q2C24ZPS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Trace amine-associated receptor 5 (Mus musculus) | BDBM50227838 (CHEMBL4102503) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a |
University of Genoa Curated by ChEMBL | Assay Description Agonist activity at mouse TAAR5 expressed in HEK293 cells assessed as cAMP accumulation after 20 mins by BRET assay | Eur J Med Chem 127: 781-792 (2017) Article DOI: 10.1016/j.ejmech.2016.10.058 BindingDB Entry DOI: 10.7270/Q2C24ZPS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Trace amine-associated receptor 5 (Mus musculus) | BDBM50227839 (CHEMBL4094764) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a |
University of Genoa Curated by ChEMBL | Assay Description Agonist activity at mouse TAAR5 expressed in HEK293 cells assessed as cAMP accumulation after 20 mins by BRET assay | Eur J Med Chem 127: 781-792 (2017) Article DOI: 10.1016/j.ejmech.2016.10.058 BindingDB Entry DOI: 10.7270/Q2C24ZPS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Trace amine-associated receptor 5 (Mus musculus) | BDBM50227840 (CHEMBL2079013) | UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a |
University of Genoa Curated by ChEMBL | Assay Description Agonist activity at mouse TAAR5 expressed in HEK293 cells assessed as cAMP accumulation after 20 mins by BRET assay | Eur J Med Chem 127: 781-792 (2017) Article DOI: 10.1016/j.ejmech.2016.10.058 BindingDB Entry DOI: 10.7270/Q2C24ZPS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Trace amine-associated receptor 5 (Mus musculus) | BDBM50227841 (ABOB | Moroxydine | SKF-8898A) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a |
University of Genoa Curated by ChEMBL | Assay Description Agonist activity at mouse TAAR5 expressed in HEK293 cells assessed as cAMP accumulation after 20 mins by BRET assay | Eur J Med Chem 127: 781-792 (2017) Article DOI: 10.1016/j.ejmech.2016.10.058 BindingDB Entry DOI: 10.7270/Q2C24ZPS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Trace amine-associated receptor 5 (Mus musculus) | BDBM18792 (1-(4-chlorophenyl)-6,6-dimethyl-1,6-dihydro-1,3,5-...) | UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE KEGG MMDB PC cid PC sid PDB UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a |
University of Genoa Curated by ChEMBL | Assay Description Agonist activity at mouse TAAR5 expressed in HEK293 cells assessed as cAMP accumulation after 20 mins by BRET assay | Eur J Med Chem 127: 781-792 (2017) Article DOI: 10.1016/j.ejmech.2016.10.058 BindingDB Entry DOI: 10.7270/Q2C24ZPS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Trace amine-associated receptor 5 (Mus musculus) | BDBM50378363 (CHEMBL574656) | UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a |
University of Genoa Curated by ChEMBL | Assay Description Agonist activity at mouse TAAR5 expressed in HEK293 cells assessed as cAMP accumulation after 20 mins by BRET assay | Eur J Med Chem 127: 781-792 (2017) Article DOI: 10.1016/j.ejmech.2016.10.058 BindingDB Entry DOI: 10.7270/Q2C24ZPS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Trace amine-associated receptor 5 (Mus musculus) | BDBM18069 (5-[(3,4,5-trimethoxyphenyl)methyl]pyrimidine-2,4-d...) | UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG MMDB PC cid PC sid PDB UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a |
University of Genoa Curated by ChEMBL | Assay Description Agonist activity at mouse TAAR5 expressed in HEK293 cells assessed as cAMP accumulation after 20 mins by BRET assay | Eur J Med Chem 127: 781-792 (2017) Article DOI: 10.1016/j.ejmech.2016.10.058 BindingDB Entry DOI: 10.7270/Q2C24ZPS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Trace amine-associated receptor 1 (Mus musculus (Mouse)) | BDBM50053629 (2-Chloro-Phenyl biguanide | CHEMBL42752 | N-(2-chl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 410 | n/a | n/a | n/a | n/a |
University of Genoa Curated by ChEMBL | Assay Description Agonist activity at mouse TAAR1 expressed in HEK293 cells assessed as cAMP accumulation after 20 mins by BRET assay | Eur J Med Chem 127: 781-792 (2017) Article DOI: 10.1016/j.ejmech.2016.10.058 BindingDB Entry DOI: 10.7270/Q2C24ZPS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Trace amine-associated receptor 1 (Mus musculus (Mouse)) | BDBM50053595 (4-Chloro-Phenyl biguanide | 4-Chlorophenylbiguanid...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 2.10E+3 | n/a | n/a | n/a | n/a |
University of Genoa Curated by ChEMBL | Assay Description Agonist activity at mouse TAAR1 expressed in HEK293 cells assessed as cAMP accumulation after 20 mins by BRET assay | Eur J Med Chem 127: 781-792 (2017) Article DOI: 10.1016/j.ejmech.2016.10.058 BindingDB Entry DOI: 10.7270/Q2C24ZPS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Trace amine-associated receptor 1 (Mus musculus (Mouse)) | BDBM50053630 (4-Methyl-Phenyl biguanide | CHEMBL291064 | N-(4-me...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.70E+3 | n/a | n/a | n/a | n/a |
University of Genoa Curated by ChEMBL | Assay Description Agonist activity at mouse TAAR1 expressed in HEK293 cells assessed as cAMP accumulation after 20 mins by BRET assay | Eur J Med Chem 127: 781-792 (2017) Article DOI: 10.1016/j.ejmech.2016.10.058 BindingDB Entry DOI: 10.7270/Q2C24ZPS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Trace amine-associated receptor 1 (Mus musculus (Mouse)) | BDBM50227975 (CHEMBL4087775) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 410 | n/a | n/a | n/a | n/a |
University of Genoa Curated by ChEMBL | Assay Description Agonist activity at mouse TAAR1 expressed in HEK293 cells assessed as cAMP accumulation after 20 mins by BRET assay | Eur J Med Chem 127: 781-792 (2017) Article DOI: 10.1016/j.ejmech.2016.10.058 BindingDB Entry DOI: 10.7270/Q2C24ZPS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Trace amine-associated receptor 1 (Mus musculus (Mouse)) | BDBM50227824 (CHEMBL4088689) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 97 | n/a | n/a | n/a | n/a |
University of Genoa Curated by ChEMBL | Assay Description Agonist activity at mouse TAAR1 expressed in HEK293 cells assessed as cAMP accumulation after 20 mins by BRET assay | Eur J Med Chem 127: 781-792 (2017) Article DOI: 10.1016/j.ejmech.2016.10.058 BindingDB Entry DOI: 10.7270/Q2C24ZPS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Trace amine-associated receptor 1 (Mus musculus (Mouse)) | BDBM50227835 (CHEMBL4096403) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 36 | n/a | n/a | n/a | n/a |
University of Genoa Curated by ChEMBL | Assay Description Agonist activity at mouse TAAR1 expressed in HEK293 cells assessed as cAMP accumulation after 20 mins by BRET assay | Eur J Med Chem 127: 781-792 (2017) Article DOI: 10.1016/j.ejmech.2016.10.058 BindingDB Entry DOI: 10.7270/Q2C24ZPS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Trace amine-associated receptor 1 (Mus musculus (Mouse)) | BDBM50227826 (CHEMBL4069147) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 540 | n/a | n/a | n/a | n/a |
University of Genoa Curated by ChEMBL | Assay Description Agonist activity at mouse TAAR1 expressed in HEK293 cells assessed as cAMP accumulation after 20 mins by BRET assay | Eur J Med Chem 127: 781-792 (2017) Article DOI: 10.1016/j.ejmech.2016.10.058 BindingDB Entry DOI: 10.7270/Q2C24ZPS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Trace amine-associated receptor 1 (Mus musculus (Mouse)) | BDBM50227828 (CHEMBL4068661) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.80E+3 | n/a | n/a | n/a | n/a |
University of Genoa Curated by ChEMBL | Assay Description Agonist activity at mouse TAAR1 expressed in HEK293 cells assessed as cAMP accumulation after 20 mins by BRET assay | Eur J Med Chem 127: 781-792 (2017) Article DOI: 10.1016/j.ejmech.2016.10.058 BindingDB Entry DOI: 10.7270/Q2C24ZPS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Trace amine-associated receptor 1 (Homo sapiens (Human)) | BDBM50053595 (4-Chloro-Phenyl biguanide | 4-Chlorophenylbiguanid...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a |
University of Genoa Curated by ChEMBL | Assay Description Agonist activity at human TAAR1 expressed in HEK293 cells assessed as cAMP accumulation after 20 mins by BRET assay | Eur J Med Chem 127: 781-792 (2017) Article DOI: 10.1016/j.ejmech.2016.10.058 BindingDB Entry DOI: 10.7270/Q2C24ZPS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Trace amine-associated receptor 1 (Homo sapiens (Human)) | BDBM50227835 (CHEMBL4096403) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.20E+3 | n/a | n/a | n/a | n/a |
University of Genoa Curated by ChEMBL | Assay Description Agonist activity at human TAAR1 expressed in HEK293 cells assessed as cAMP accumulation after 20 mins by BRET assay | Eur J Med Chem 127: 781-792 (2017) Article DOI: 10.1016/j.ejmech.2016.10.058 BindingDB Entry DOI: 10.7270/Q2C24ZPS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Trace amine-associated receptor 5 (Mus musculus) | BDBM50053596 (1-phenylbiguanide | CHEMBL13791 | N-phenylimidodic...) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a |
University of Genoa Curated by ChEMBL | Assay Description Agonist activity at mouse TAAR5 expressed in HEK293 cells assessed as cAMP accumulation after 20 mins by BRET assay | Eur J Med Chem 127: 781-792 (2017) Article DOI: 10.1016/j.ejmech.2016.10.058 BindingDB Entry DOI: 10.7270/Q2C24ZPS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Trace amine-associated receptor 5 (Mus musculus) | BDBM50053595 (4-Chloro-Phenyl biguanide | 4-Chlorophenylbiguanid...) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a |
University of Genoa Curated by ChEMBL | Assay Description Agonist activity at mouse TAAR5 expressed in HEK293 cells assessed as cAMP accumulation after 20 mins by BRET assay | Eur J Med Chem 127: 781-792 (2017) Article DOI: 10.1016/j.ejmech.2016.10.058 BindingDB Entry DOI: 10.7270/Q2C24ZPS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Trace amine-associated receptor 5 (Mus musculus) | BDBM50053630 (4-Methyl-Phenyl biguanide | CHEMBL291064 | N-(4-me...) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a |
University of Genoa Curated by ChEMBL | Assay Description Agonist activity at mouse TAAR5 expressed in HEK293 cells assessed as cAMP accumulation after 20 mins by BRET assay | Eur J Med Chem 127: 781-792 (2017) Article DOI: 10.1016/j.ejmech.2016.10.058 BindingDB Entry DOI: 10.7270/Q2C24ZPS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Trace amine-associated receptor 5 (Mus musculus) | BDBM50227975 (CHEMBL4087775) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a |
University of Genoa Curated by ChEMBL | Assay Description Agonist activity at mouse TAAR5 expressed in HEK293 cells assessed as cAMP accumulation after 20 mins by BRET assay | Eur J Med Chem 127: 781-792 (2017) Article DOI: 10.1016/j.ejmech.2016.10.058 BindingDB Entry DOI: 10.7270/Q2C24ZPS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Trace amine-associated receptor 5 (Mus musculus) | BDBM50227826 (CHEMBL4069147) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a |
University of Genoa Curated by ChEMBL | Assay Description Agonist activity at mouse TAAR5 expressed in HEK293 cells assessed as cAMP accumulation after 20 mins by BRET assay | Eur J Med Chem 127: 781-792 (2017) Article DOI: 10.1016/j.ejmech.2016.10.058 BindingDB Entry DOI: 10.7270/Q2C24ZPS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Trace amine-associated receptor 5 (Mus musculus) | BDBM50227979 (CHEMBL4084561) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a |
University of Genoa Curated by ChEMBL | Assay Description Agonist activity at mouse TAAR5 expressed in HEK293 cells assessed as cAMP accumulation after 20 mins by BRET assay | Eur J Med Chem 127: 781-792 (2017) Article DOI: 10.1016/j.ejmech.2016.10.058 BindingDB Entry DOI: 10.7270/Q2C24ZPS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Trace amine-associated receptor 5 (Mus musculus) | BDBM50227829 (CHEBI:8455 | CHLOROGUANIDE | Proguanil) | UniProtKB/SwissProt GoogleScholar AffyNet | Purchase MCE PC cid PC sid PDB UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a |
University of Genoa Curated by ChEMBL | Assay Description Agonist activity at mouse TAAR5 expressed in HEK293 cells assessed as cAMP accumulation after 20 mins by BRET assay | Eur J Med Chem 127: 781-792 (2017) Article DOI: 10.1016/j.ejmech.2016.10.058 BindingDB Entry DOI: 10.7270/Q2C24ZPS | |||||||||||
More data for this Ligand-Target Pair |
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