Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
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Peroxisome proliferator-activated receptor gamma (Homo sapiens (Human)) | BDBM50428826 (CHEMBL2337127) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid PDB UniChem Similars | PDB Article PubMed | n/a | n/a | n/a | n/a | 73 | n/a | n/a | n/a | n/a |
Max Planck Institute for Molecular Genetics Curated by ChEMBL | Assay Description Agonist at human PPARgamma LBD expressed in human HEK293 cells cotransfected with GAL4-Luc assessed as transcriptional activation by luciferase repor... | J Nat Prod 78: 1160-4 (2015) Article DOI: 10.1021/np500747y BindingDB Entry DOI: 10.7270/Q24T6M4N | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) |