Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Type-1 angiotensin II receptor (RABBIT) | BDBM50038189 (4'-(2-Ethyl-5,7-dimethyl-imidazo[4,5-b]pyridin-3-y...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 0.200 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description In vitro binding affinity of the compound for angiotensin II AT1 receptor in rabbit aorta | J Med Chem 37: 4068-72 (1995) BindingDB Entry DOI: 10.7270/Q2DV1HZ3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Type-1 angiotensin II receptor (RABBIT) | BDBM50038190 (4'-(2-Ethyl-5,7-dimethyl-imidazo[4,5-b]pyridin-3-y...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 0.210 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description In vitro binding affinity of the compound for angiotensin II AT1 receptor in rabbit aorta | J Med Chem 37: 4068-72 (1995) BindingDB Entry DOI: 10.7270/Q2DV1HZ3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Type-1 angiotensin II receptor (RABBIT) | BDBM50038192 (4'-(2-Ethyl-5,7-dimethyl-imidazo[4,5-b]pyridin-3-y...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 0.270 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description In vitro binding affinity of the compound for angiotensin II AT1 receptor in rabbit aorta | J Med Chem 37: 4068-72 (1995) BindingDB Entry DOI: 10.7270/Q2DV1HZ3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Type-1 angiotensin II receptor (RABBIT) | BDBM50009718 (2-Ethyl-5,7-dimethyl-3-[2'-(1H-tetrazol-5-yl)-biph...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 0.300 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description In vitro binding affinity of the compound for angiotensin II AT1 receptor in rabbit aorta | J Med Chem 37: 4068-72 (1995) BindingDB Entry DOI: 10.7270/Q2DV1HZ3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Type-1 angiotensin II receptor (RABBIT) | BDBM50038193 (4'-(2-Ethyl-5,7-dimethyl-imidazo[4,5-b]pyridin-3-y...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 0.680 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description In vitro binding affinity of the compound for angiotensin II AT1 receptor in rabbit aorta | J Med Chem 37: 4068-72 (1995) BindingDB Entry DOI: 10.7270/Q2DV1HZ3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Type-1 angiotensin II receptor (RABBIT) | BDBM50038191 (4'-(2-Ethyl-5,7-dimethyl-imidazo[4,5-b]pyridin-3-y...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 2.20 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description In vitro binding affinity of the compound for angiotensin II AT1 receptor in rabbit aorta | J Med Chem 37: 4068-72 (1995) BindingDB Entry DOI: 10.7270/Q2DV1HZ3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Type-1 angiotensin II receptor (RABBIT) | BDBM50006909 (2-Butyl-5-chloro-3-[2'-(1H-tetrazol-5-yl)-biphenyl...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE KEGG PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 6 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description In vitro binding affinity of the compound for angiotensin II AT1 receptor in rabbit aorta | J Med Chem 37: 4068-72 (1995) BindingDB Entry DOI: 10.7270/Q2DV1HZ3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Type-1 angiotensin II receptor (RABBIT) | BDBM50009714 (CHEMBL191 | {2-Butyl-5-chloro-3-[2'-(2H-tetrazol-5...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 50 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description In vitro binding affinity of the compound for angiotensin II AT1 receptor in rabbit aorta | J Med Chem 37: 4068-72 (1995) BindingDB Entry DOI: 10.7270/Q2DV1HZ3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Type-2 angiotensin II receptor (RAT) | BDBM50038190 (4'-(2-Ethyl-5,7-dimethyl-imidazo[4,5-b]pyridin-3-y...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 1.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description In vitro binding affinity of the compound for angiotensin II AT2 receptor in rat midbrain | J Med Chem 37: 4068-72 (1995) BindingDB Entry DOI: 10.7270/Q2DV1HZ3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Type-2 angiotensin II receptor (RAT) | BDBM50038193 (4'-(2-Ethyl-5,7-dimethyl-imidazo[4,5-b]pyridin-3-y...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 2.40E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description In vitro binding affinity of the compound for angiotensin II AT2 receptor in rat midbrain | J Med Chem 37: 4068-72 (1995) BindingDB Entry DOI: 10.7270/Q2DV1HZ3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Type-2 angiotensin II receptor (RAT) | BDBM50038189 (4'-(2-Ethyl-5,7-dimethyl-imidazo[4,5-b]pyridin-3-y...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 2.90E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description In vitro binding affinity of the compound for angiotensin II AT2 receptor in rat midbrain | J Med Chem 37: 4068-72 (1995) BindingDB Entry DOI: 10.7270/Q2DV1HZ3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Type-2 angiotensin II receptor (RAT) | BDBM50038192 (4'-(2-Ethyl-5,7-dimethyl-imidazo[4,5-b]pyridin-3-y...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 3.60E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description In vitro binding affinity of the compound for angiotensin II AT2 receptor in rat midbrain | J Med Chem 37: 4068-72 (1995) BindingDB Entry DOI: 10.7270/Q2DV1HZ3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Type-2 angiotensin II receptor (RAT) | BDBM50038191 (4'-(2-Ethyl-5,7-dimethyl-imidazo[4,5-b]pyridin-3-y...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description In vitro binding affinity of the compound for angiotensin II AT2 receptor in rat midbrain | J Med Chem 37: 4068-72 (1995) BindingDB Entry DOI: 10.7270/Q2DV1HZ3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Type-2 angiotensin II receptor (RAT) | BDBM50009718 (2-Ethyl-5,7-dimethyl-3-[2'-(1H-tetrazol-5-yl)-biph...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 5.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description In vitro binding affinity of the compound for angiotensin II AT2 receptor in rat midbrain | J Med Chem 37: 4068-72 (1995) BindingDB Entry DOI: 10.7270/Q2DV1HZ3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Type-2 angiotensin II receptor (RAT) | BDBM50006909 (2-Butyl-5-chloro-3-[2'-(1H-tetrazol-5-yl)-biphenyl...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE KEGG PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 5.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description In vitro binding affinity of the compound for angiotensin II AT2 receptor in rat midbrain | J Med Chem 37: 4068-72 (1995) BindingDB Entry DOI: 10.7270/Q2DV1HZ3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Type-2 angiotensin II receptor (RAT) | BDBM50009714 (CHEMBL191 | {2-Butyl-5-chloro-3-[2'-(2H-tetrazol-5...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 5.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description In vitro binding affinity of the compound for angiotensin II AT2 receptor in rat midbrain | J Med Chem 37: 4068-72 (1995) BindingDB Entry DOI: 10.7270/Q2DV1HZ3 | |||||||||||
More data for this Ligand-Target Pair |