Found 87 hits with Last Name = 'hsu' and Initial = 'fl' Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
Alpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor
(RAT-NEONATAL RAT-Rattus norvegicus (rat)) | BDBM50471350
(CHEMBL102763)Show InChI InChI=1S/C13H14N2/c1-9-3-2-4-11-10(9)5-6-12(11)13-7-14-8-15-13/h2-4,7-8,12H,5-6H2,1H3,(H,14,15) | PDB
UniProtKB/SwissProt
GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 8.80 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Tennessee
Curated by ChEMBL
| Assay Description Displacement of [3H]rauwolscine from Alpha-2 adrenergic receptor of rat brain membranes |
J Med Chem 40: 3014-24 (1997)
Article DOI: 10.1021/jm960642q BindingDB Entry DOI: 10.7270/Q2ZG6VZ9 |
More data for this Ligand-Target Pair | |
Alpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor
(RAT-NEONATAL RAT-Rattus norvegicus (rat)) | BDBM50036910
(4-(1-Naphthalen-1-yl-ethyl)-1H-imidazole | CHEMBL3...)Show InChI InChI=1S/C15H14N2/c1-11(15-9-16-10-17-15)13-8-4-6-12-5-2-3-7-14(12)13/h2-11H,1H3,(H,16,17) | PDB
UniProtKB/SwissProt
GoogleScholar AffyNet
| Purchase
CHEMBL PC cid PC sid UniChem
Patents
Similars
| Article PubMed
| 13 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Ohio State University
Curated by ChEMBL
| Assay Description Alpha-2 adrenergic receptor binding affinity was tested against membrane preparations of rat brain using 0.2 nM [3H]rauwolscine as radioligand |
J Med Chem 39: 3001-13 (1996)
Article DOI: 10.1021/jm9506074 BindingDB Entry DOI: 10.7270/Q2BV7KBH |
More data for this Ligand-Target Pair | |
Alpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor
(RAT-NEONATAL RAT-Rattus norvegicus (rat)) | BDBM50036913
((+-)-4-(alpha,2,3-trimethylbenzyl)imidazole | 4-[1...)Show InChI InChI=1S/C13H16N2/c1-9-5-4-6-12(10(9)2)11(3)13-7-14-8-15-13/h4-8,11H,1-3H3,(H,14,15) | PDB
UniProtKB/SwissProt
GoogleScholar AffyNet
| Purchase
CHEMBL MCE PC cid PC sid UniChem
Patents
Similars
| Article PubMed
| 25 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Ohio State University
Curated by ChEMBL
| Assay Description Alpha-2 adrenergic receptor binding affinity was tested against membrane preparations of rat brain. |
J Med Chem 39: 3001-13 (1996)
Article DOI: 10.1021/jm9506074 BindingDB Entry DOI: 10.7270/Q2BV7KBH |
More data for this Ligand-Target Pair | |
Alpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor
(RAT-NEONATAL RAT-Rattus norvegicus (rat)) | BDBM50036913
((+-)-4-(alpha,2,3-trimethylbenzyl)imidazole | 4-[1...)Show InChI InChI=1S/C13H16N2/c1-9-5-4-6-12(10(9)2)11(3)13-7-14-8-15-13/h4-8,11H,1-3H3,(H,14,15) | PDB
UniProtKB/SwissProt
GoogleScholar AffyNet
| Purchase
CHEMBL MCE PC cid PC sid UniChem
Patents
Similars
| Article PubMed
| 25 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Tennessee
Curated by ChEMBL
| Assay Description Displacement of [3H]rauwolscine from Alpha-2 adrenergic receptor of rat brain membranes |
J Med Chem 40: 3014-24 (1997)
Article DOI: 10.1021/jm960642q BindingDB Entry DOI: 10.7270/Q2ZG6VZ9 |
More data for this Ligand-Target Pair | |
Alpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor
(RAT-NEONATAL RAT-Rattus norvegicus (rat)) | BDBM50471342
(CHEMBL322907)Show InChI InChI=1S/C14H14N2/c1-10-4-2-6-12-11(10)5-3-7-13(12)14-8-15-9-16-14/h2,4,6-9H,3,5H2,1H3,(H,15,16) | PDB
UniProtKB/SwissProt
GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 31 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Tennessee
Curated by ChEMBL
| Assay Description Displacement of [3H]rauwolscine from Alpha-2 adrenergic receptor of rat brain membranes |
J Med Chem 40: 3014-24 (1997)
Article DOI: 10.1021/jm960642q BindingDB Entry DOI: 10.7270/Q2ZG6VZ9 |
More data for this Ligand-Target Pair | |
Alpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor
(RAT-NEONATAL RAT-Rattus norvegicus (rat)) | BDBM50470860
(CHEMBL105328)Show InChI InChI=1S/C16H14N2/c1-3-11-5-2-6-14-13(15-9-17-10-18-15)8-7-12(4-1)16(11)14/h1-6,9-10,13H,7-8H2,(H,17,18) | PDB
UniProtKB/SwissProt
GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 33 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Ohio State University
Curated by ChEMBL
| Assay Description Alpha-2 adrenergic receptor binding affinity was tested against membrane preparations of rat brain using 0.2 nM [3H]rauwolscine as radioligand |
J Med Chem 39: 3001-13 (1996)
Article DOI: 10.1021/jm9506074 BindingDB Entry DOI: 10.7270/Q2BV7KBH |
More data for this Ligand-Target Pair | |
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor
(Rattus norvegicus (rat)-Rattus norvegicus (Rat)) | BDBM50470860
(CHEMBL105328)Show InChI InChI=1S/C16H14N2/c1-3-11-5-2-6-14-13(15-9-17-10-18-15)8-7-12(4-1)16(11)14/h1-6,9-10,13H,7-8H2,(H,17,18) | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 55 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Ohio State University
Curated by ChEMBL
| Assay Description Alpha-1 adrenergic receptor binding affinity in rat brain membranes |
J Med Chem 39: 3001-13 (1996)
Article DOI: 10.1021/jm9506074 BindingDB Entry DOI: 10.7270/Q2BV7KBH |
More data for this Ligand-Target Pair | |
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor
(Rattus norvegicus (rat)-Rattus norvegicus (Rat)) | BDBM50470861
(CHEMBL322844)Show InChI InChI=1S/C16H14N2/c1-2-13(16-10-17-11-18-16)15-9-5-7-12-6-3-4-8-14(12)15/h2-11H,1H3,(H,17,18)/b13-2- | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 57 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Ohio State University
Curated by ChEMBL
| Assay Description Alpha-1 adrenergic receptor binding affinity in rat brain membranes |
J Med Chem 39: 3001-13 (1996)
Article DOI: 10.1021/jm9506074 BindingDB Entry DOI: 10.7270/Q2BV7KBH |
More data for this Ligand-Target Pair | |
Alpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor
(RAT-NEONATAL RAT-Rattus norvegicus (rat)) | BDBM50471340
(CHEMBL317912)Show InChI InChI=1S/C13H14N2O/c16-13-6-2-3-9-10(4-1-5-11(9)13)12-7-14-8-15-12/h2-3,6-8,10,16H,1,4-5H2,(H,14,15) | PDB
UniProtKB/SwissProt
GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 63 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Tennessee
Curated by ChEMBL
| Assay Description Displacement of [3H]rauwolscine from Alpha-2 adrenergic receptor of rat brain membranes |
J Med Chem 40: 3014-24 (1997)
Article DOI: 10.1021/jm960642q BindingDB Entry DOI: 10.7270/Q2ZG6VZ9 |
More data for this Ligand-Target Pair | |
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor
(Rattus norvegicus (rat)-Rattus norvegicus (Rat)) | BDBM50471350
(CHEMBL102763)Show InChI InChI=1S/C13H14N2/c1-9-3-2-4-11-10(9)5-6-12(11)13-7-14-8-15-13/h2-4,7-8,12H,5-6H2,1H3,(H,14,15) | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 73 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Tennessee
Curated by ChEMBL
| Assay Description Displacement of [3H]-prazosin from Alpha-1 adrenergic receptor of rat brain membranes |
J Med Chem 40: 3014-24 (1997)
Article DOI: 10.1021/jm960642q BindingDB Entry DOI: 10.7270/Q2ZG6VZ9 |
More data for this Ligand-Target Pair | |
Alpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor
(RAT-NEONATAL RAT-Rattus norvegicus (rat)) | BDBM50471338
(CHEMBL105347)Show InChI InChI=1S/C14H16N2/c1-10-4-2-6-12-11(10)5-3-7-13(12)14-8-15-9-16-14/h2,4,6,8-9,13H,3,5,7H2,1H3,(H,15,16) | PDB
UniProtKB/SwissProt
GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 95 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Tennessee
Curated by ChEMBL
| Assay Description Displacement of [3H]rauwolscine from Alpha-2 adrenergic receptor of rat brain membranes |
J Med Chem 40: 3014-24 (1997)
Article DOI: 10.1021/jm960642q BindingDB Entry DOI: 10.7270/Q2ZG6VZ9 |
More data for this Ligand-Target Pair | |
Alpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor
(RAT-NEONATAL RAT-Rattus norvegicus (rat)) | BDBM50471346
(CHEMBL330185)Show InChI InChI=1S/C14H16N2O/c1-17-14-7-3-4-10-11(5-2-6-12(10)14)13-8-15-9-16-13/h3-4,7-9,11H,2,5-6H2,1H3,(H,15,16) | PDB
UniProtKB/SwissProt
GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 98 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Tennessee
Curated by ChEMBL
| Assay Description Displacement of [3H]rauwolscine from Alpha-2 adrenergic receptor of rat brain membranes |
J Med Chem 40: 3014-24 (1997)
Article DOI: 10.1021/jm960642q BindingDB Entry DOI: 10.7270/Q2ZG6VZ9 |
More data for this Ligand-Target Pair | |
Alpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor
(RAT-NEONATAL RAT-Rattus norvegicus (rat)) | BDBM50471343
(CHEMBL319221)Show InChI InChI=1S/C15H18N2/c1-10-6-11(2)12-4-3-5-13(14(12)7-10)15-8-16-9-17-15/h6-9,13H,3-5H2,1-2H3,(H,16,17) | PDB
UniProtKB/SwissProt
GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 103 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Tennessee
Curated by ChEMBL
| Assay Description Displacement of [3H]rauwolscine from Alpha-2 adrenergic receptor of rat brain membranes |
J Med Chem 40: 3014-24 (1997)
Article DOI: 10.1021/jm960642q BindingDB Entry DOI: 10.7270/Q2ZG6VZ9 |
More data for this Ligand-Target Pair | |
Alpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor
(RAT-NEONATAL RAT-Rattus norvegicus (rat)) | BDBM50470859
(CHEMBL105487)Show InChI InChI=1S/C15H12N2/c1-11(15-9-16-10-17-15)13-8-4-6-12-5-2-3-7-14(12)13/h2-10H,1H2,(H,16,17) | PDB
UniProtKB/SwissProt
GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 122 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Ohio State University
Curated by ChEMBL
| Assay Description Alpha-2 adrenergic receptor binding affinity was tested against membrane preparations of rat brain using 0.2 nM [3H]rauwolscine as radioligand |
J Med Chem 39: 3001-13 (1996)
Article DOI: 10.1021/jm9506074 BindingDB Entry DOI: 10.7270/Q2BV7KBH |
More data for this Ligand-Target Pair | |
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor
(Rattus norvegicus (rat)-Rattus norvegicus (Rat)) | BDBM50471340
(CHEMBL317912)Show InChI InChI=1S/C13H14N2O/c16-13-6-2-3-9-10(4-1-5-11(9)13)12-7-14-8-15-12/h2-3,6-8,10,16H,1,4-5H2,(H,14,15) | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 126 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Tennessee
Curated by ChEMBL
| Assay Description Displacement of [3H]-prazosin from Alpha-1 adrenergic receptor of rat brain membranes |
J Med Chem 40: 3014-24 (1997)
Article DOI: 10.1021/jm960642q BindingDB Entry DOI: 10.7270/Q2ZG6VZ9 |
More data for this Ligand-Target Pair | |
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor
(Rattus norvegicus (rat)-Rattus norvegicus (Rat)) | BDBM50471343
(CHEMBL319221)Show InChI InChI=1S/C15H18N2/c1-10-6-11(2)12-4-3-5-13(14(12)7-10)15-8-16-9-17-15/h6-9,13H,3-5H2,1-2H3,(H,16,17) | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 131 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Tennessee
Curated by ChEMBL
| Assay Description Displacement of [3H]-prazosin from Alpha-1 adrenergic receptor of rat brain membranes |
J Med Chem 40: 3014-24 (1997)
Article DOI: 10.1021/jm960642q BindingDB Entry DOI: 10.7270/Q2ZG6VZ9 |
More data for this Ligand-Target Pair | |
Alpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor
(RAT-NEONATAL RAT-Rattus norvegicus (rat)) | BDBM50470862
(CHEMBL102076)Show InChI InChI=1S/C16H16N2/c1-2-13(16-10-17-11-18-16)15-9-5-7-12-6-3-4-8-14(12)15/h3-11,13H,2H2,1H3,(H,17,18) | PDB
UniProtKB/SwissProt
GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 165 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Ohio State University
Curated by ChEMBL
| Assay Description Alpha-2 adrenergic receptor binding affinity was tested against membrane preparations of rat brain using 0.2 nM [3H]rauwolscine as radioligand |
J Med Chem 39: 3001-13 (1996)
Article DOI: 10.1021/jm9506074 BindingDB Entry DOI: 10.7270/Q2BV7KBH |
More data for this Ligand-Target Pair | |
Alpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor
(RAT-NEONATAL RAT-Rattus norvegicus (rat)) | BDBM50471347
(CHEMBL319984)Show InChI InChI=1S/C14H16N2O/c1-17-11-5-6-12-10(7-11)3-2-4-13(12)14-8-15-9-16-14/h5-9,13H,2-4H2,1H3,(H,15,16) | PDB
UniProtKB/SwissProt
GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 169 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Tennessee
Curated by ChEMBL
| Assay Description Displacement of [3H]rauwolscine from Alpha-2 adrenergic receptor of rat brain membranes |
J Med Chem 40: 3014-24 (1997)
Article DOI: 10.1021/jm960642q BindingDB Entry DOI: 10.7270/Q2ZG6VZ9 |
More data for this Ligand-Target Pair | |
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor
(Rattus norvegicus (rat)-Rattus norvegicus (Rat)) | BDBM50471338
(CHEMBL105347)Show InChI InChI=1S/C14H16N2/c1-10-4-2-6-12-11(10)5-3-7-13(12)14-8-15-9-16-14/h2,4,6,8-9,13H,3,5,7H2,1H3,(H,15,16) | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 191 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Tennessee
Curated by ChEMBL
| Assay Description Displacement of [3H]-prazosin from Alpha-1 adrenergic receptor of rat brain membranes |
J Med Chem 40: 3014-24 (1997)
Article DOI: 10.1021/jm960642q BindingDB Entry DOI: 10.7270/Q2ZG6VZ9 |
More data for this Ligand-Target Pair | |
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor
(Rattus norvegicus (rat)-Rattus norvegicus (Rat)) | BDBM50471347
(CHEMBL319984)Show InChI InChI=1S/C14H16N2O/c1-17-11-5-6-12-10(7-11)3-2-4-13(12)14-8-15-9-16-14/h5-9,13H,2-4H2,1H3,(H,15,16) | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 198 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Tennessee
Curated by ChEMBL
| Assay Description Displacement of [3H]-prazosin from Alpha-1 adrenergic receptor of rat brain membranes |
J Med Chem 40: 3014-24 (1997)
Article DOI: 10.1021/jm960642q BindingDB Entry DOI: 10.7270/Q2ZG6VZ9 |
More data for this Ligand-Target Pair | |
Alpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor
(RAT-NEONATAL RAT-Rattus norvegicus (rat)) | BDBM50471348
(CHEMBL103448)Show InChI InChI=1S/C14H16N2O/c1-17-11-6-5-10-3-2-4-12(13(10)7-11)14-8-15-9-16-14/h5-9,12H,2-4H2,1H3,(H,15,16) | PDB
UniProtKB/SwissProt
GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 201 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Tennessee
Curated by ChEMBL
| Assay Description Displacement of [3H]rauwolscine from Alpha-2 adrenergic receptor of rat brain membranes |
J Med Chem 40: 3014-24 (1997)
Article DOI: 10.1021/jm960642q BindingDB Entry DOI: 10.7270/Q2ZG6VZ9 |
More data for this Ligand-Target Pair | |
Alpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor
(RAT-NEONATAL RAT-Rattus norvegicus (rat)) | BDBM50223426
(CHEBI:10304 | Corbadrine | Levonordefrin | Neo-Cob...)Show SMILES [H][C@@](C)(N)[C@]([H])(O)c1ccc(O)c(O)c1 |r| Show InChI InChI=1S/C9H13NO3/c1-5(10)9(13)6-2-3-7(11)8(12)4-6/h2-5,9,11-13H,10H2,1H3/t5-,9-/m0/s1 | PDB
UniProtKB/SwissProt
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| Purchase
MCE KEGG PC cid PC sid UniChem
Similars
| Article PubMed
| 205 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Ohio State University
Curated by ChEMBL
| Assay Description Alpha-2 adrenergic receptor binding affinity was tested against membrane preparations of rat brain. |
J Med Chem 39: 3001-13 (1996)
Article DOI: 10.1021/jm9506074 BindingDB Entry DOI: 10.7270/Q2BV7KBH |
More data for this Ligand-Target Pair | |
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor
(Rattus norvegicus (rat)-Rattus norvegicus (Rat)) | BDBM50036910
(4-(1-Naphthalen-1-yl-ethyl)-1H-imidazole | CHEMBL3...)Show InChI InChI=1S/C15H14N2/c1-11(15-9-16-10-17-15)13-8-4-6-12-5-2-3-7-14(12)13/h2-11H,1H3,(H,16,17) | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank GoogleScholar AffyNet
| Purchase
CHEMBL PC cid PC sid UniChem
Patents
Similars
| Article PubMed
| 224 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Ohio State University
Curated by ChEMBL
| Assay Description Alpha-1 adrenergic receptor binding affinity in rat brain membranes |
J Med Chem 39: 3001-13 (1996)
Article DOI: 10.1021/jm9506074 BindingDB Entry DOI: 10.7270/Q2BV7KBH |
More data for this Ligand-Target Pair | |
Alpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor
(RAT-NEONATAL RAT-Rattus norvegicus (rat)) | BDBM50471344
(CHEMBL422247)Show InChI InChI=1S/C15H16N2/c1-10-6-11(2)12-4-3-5-13(14(12)7-10)15-8-16-9-17-15/h5-9H,3-4H2,1-2H3,(H,16,17) | PDB
UniProtKB/SwissProt
GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 232 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Tennessee
Curated by ChEMBL
| Assay Description Displacement of [3H]rauwolscine from Alpha-2 adrenergic receptor of rat brain membranes |
J Med Chem 40: 3014-24 (1997)
Article DOI: 10.1021/jm960642q BindingDB Entry DOI: 10.7270/Q2ZG6VZ9 |
More data for this Ligand-Target Pair | |
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor
(Rattus norvegicus (rat)-Rattus norvegicus (Rat)) | BDBM50471346
(CHEMBL330185)Show InChI InChI=1S/C14H16N2O/c1-17-14-7-3-4-10-11(5-2-6-12(10)14)13-8-15-9-16-13/h3-4,7-9,11H,2,5-6H2,1H3,(H,15,16) | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 243 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Tennessee
Curated by ChEMBL
| Assay Description Displacement of [3H]-prazosin from Alpha-1 adrenergic receptor of rat brain membranes |
J Med Chem 40: 3014-24 (1997)
Article DOI: 10.1021/jm960642q BindingDB Entry DOI: 10.7270/Q2ZG6VZ9 |
More data for this Ligand-Target Pair | |
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor
(Rattus norvegicus (rat)-Rattus norvegicus (Rat)) | BDBM50470863
(CHEMBL102669)Show InChI InChI=1S/C16H14N2/c1-2-13(16-10-17-11-18-16)15-9-5-7-12-6-3-4-8-14(12)15/h2-11H,1H3,(H,17,18)/b13-2+ | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 387 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Ohio State University
Curated by ChEMBL
| Assay Description Alpha-1 adrenergic receptor binding affinity in rat brain membranes |
J Med Chem 39: 3001-13 (1996)
Article DOI: 10.1021/jm9506074 BindingDB Entry DOI: 10.7270/Q2BV7KBH |
More data for this Ligand-Target Pair | |
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor
(Rattus norvegicus (rat)-Rattus norvegicus (Rat)) | BDBM50470862
(CHEMBL102076)Show InChI InChI=1S/C16H16N2/c1-2-13(16-10-17-11-18-16)15-9-5-7-12-6-3-4-8-14(12)15/h3-11,13H,2H2,1H3,(H,17,18) | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 574 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Ohio State University
Curated by ChEMBL
| Assay Description Alpha-1 adrenergic receptor binding affinity in rat brain membranes |
J Med Chem 39: 3001-13 (1996)
Article DOI: 10.1021/jm9506074 BindingDB Entry DOI: 10.7270/Q2BV7KBH |
More data for this Ligand-Target Pair | |
Alpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor
(RAT-NEONATAL RAT-Rattus norvegicus (rat)) | BDBM50471339
(CHEMBL103500)Show InChI InChI=1S/C14H14N2O/c1-17-11-5-6-12-10(7-11)3-2-4-13(12)14-8-15-9-16-14/h4-9H,2-3H2,1H3,(H,15,16) | PDB
UniProtKB/SwissProt
GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 580 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Tennessee
Curated by ChEMBL
| Assay Description Displacement of [3H]rauwolscine from Alpha-2 adrenergic receptor of rat brain membranes |
J Med Chem 40: 3014-24 (1997)
Article DOI: 10.1021/jm960642q BindingDB Entry DOI: 10.7270/Q2ZG6VZ9 |
More data for this Ligand-Target Pair | |
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor
(Rattus norvegicus (rat)-Rattus norvegicus (Rat)) | BDBM50470864
(CHEMBL420652)Show InChI InChI=1S/C17H16N2/c1-2-6-14-12(4-1)8-9-13-5-3-7-15(17(13)14)16-10-18-11-19-16/h1-2,4,6,8-11,15H,3,5,7H2,(H,18,19) | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 655 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Ohio State University
Curated by ChEMBL
| Assay Description Alpha-1 adrenergic receptor binding affinity in rat brain membranes |
J Med Chem 39: 3001-13 (1996)
Article DOI: 10.1021/jm9506074 BindingDB Entry DOI: 10.7270/Q2BV7KBH |
More data for this Ligand-Target Pair | |
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor
(Rattus norvegicus (rat)-Rattus norvegicus (Rat)) | BDBM50471342
(CHEMBL322907)Show InChI InChI=1S/C14H14N2/c1-10-4-2-6-12-11(10)5-3-7-13(12)14-8-15-9-16-14/h2,4,6-9H,3,5H2,1H3,(H,15,16) | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 992 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Tennessee
Curated by ChEMBL
| Assay Description Displacement of [3H]-prazosin from Alpha-1 adrenergic receptor of rat brain membranes |
J Med Chem 40: 3014-24 (1997)
Article DOI: 10.1021/jm960642q BindingDB Entry DOI: 10.7270/Q2ZG6VZ9 |
More data for this Ligand-Target Pair | |
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor
(Rattus norvegicus (rat)-Rattus norvegicus (Rat)) | BDBM50036913
((+-)-4-(alpha,2,3-trimethylbenzyl)imidazole | 4-[1...)Show InChI InChI=1S/C13H16N2/c1-9-5-4-6-12(10(9)2)11(3)13-7-14-8-15-13/h4-8,11H,1-3H3,(H,14,15) | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank GoogleScholar AffyNet
| Purchase
CHEMBL MCE PC cid PC sid UniChem
Patents
Similars
| Article PubMed
| 1.11E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Ohio State University
Curated by ChEMBL
| Assay Description Alpha-1 adrenergic receptor binding affinity in rat brain membranes |
J Med Chem 39: 3001-13 (1996)
Article DOI: 10.1021/jm9506074 BindingDB Entry DOI: 10.7270/Q2BV7KBH |
More data for this Ligand-Target Pair | |
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor
(Rattus norvegicus (rat)-Rattus norvegicus (Rat)) | BDBM50036913
((+-)-4-(alpha,2,3-trimethylbenzyl)imidazole | 4-[1...)Show InChI InChI=1S/C13H16N2/c1-9-5-4-6-12(10(9)2)11(3)13-7-14-8-15-13/h4-8,11H,1-3H3,(H,14,15) | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank GoogleScholar AffyNet
| Purchase
CHEMBL MCE PC cid PC sid UniChem
Patents
Similars
| Article PubMed
| 1.11E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Tennessee
Curated by ChEMBL
| Assay Description Displacement of [3H]-prazosin from Alpha-1 adrenergic receptor of rat brain membranes |
J Med Chem 40: 3014-24 (1997)
Article DOI: 10.1021/jm960642q BindingDB Entry DOI: 10.7270/Q2ZG6VZ9 |
More data for this Ligand-Target Pair | |
Alpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor
(RAT-NEONATAL RAT-Rattus norvegicus (rat)) | BDBM50471349
(CHEMBL321964)Show InChI InChI=1S/C14H14N2O/c1-17-14-7-3-4-10-11(5-2-6-12(10)14)13-8-15-9-16-13/h3-5,7-9H,2,6H2,1H3,(H,15,16) | PDB
UniProtKB/SwissProt
GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 1.42E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Tennessee
Curated by ChEMBL
| Assay Description Displacement of [3H]rauwolscine from Alpha-2 adrenergic receptor of rat brain membranes |
J Med Chem 40: 3014-24 (1997)
Article DOI: 10.1021/jm960642q BindingDB Entry DOI: 10.7270/Q2ZG6VZ9 |
More data for this Ligand-Target Pair | |
Alpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor
(RAT-NEONATAL RAT-Rattus norvegicus (rat)) | BDBM50470864
(CHEMBL420652)Show InChI InChI=1S/C17H16N2/c1-2-6-14-12(4-1)8-9-13-5-3-7-15(17(13)14)16-10-18-11-19-16/h1-2,4,6,8-11,15H,3,5,7H2,(H,18,19) | PDB
UniProtKB/SwissProt
GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 1.45E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Ohio State University
Curated by ChEMBL
| Assay Description Alpha-2 adrenergic receptor binding affinity was tested against membrane preparations of rat brain. |
J Med Chem 39: 3001-13 (1996)
Article DOI: 10.1021/jm9506074 BindingDB Entry DOI: 10.7270/Q2BV7KBH |
More data for this Ligand-Target Pair | |
Alpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor
(RAT-NEONATAL RAT-Rattus norvegicus (rat)) | BDBM50470863
(CHEMBL102669)Show InChI InChI=1S/C16H14N2/c1-2-13(16-10-17-11-18-16)15-9-5-7-12-6-3-4-8-14(12)15/h2-11H,1H3,(H,17,18)/b13-2+ | PDB
UniProtKB/SwissProt
GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 1.47E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Ohio State University
Curated by ChEMBL
| Assay Description Alpha-2 adrenergic receptor binding affinity was tested against membrane preparations of rat brain using 0.2 nM [3H]rauwolscine as radioligand |
J Med Chem 39: 3001-13 (1996)
Article DOI: 10.1021/jm9506074 BindingDB Entry DOI: 10.7270/Q2BV7KBH |
More data for this Ligand-Target Pair | |
Alpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor
(RAT-NEONATAL RAT-Rattus norvegicus (rat)) | BDBM50471345
(CHEMBL102538)Show InChI InChI=1S/C14H14N2O/c1-17-11-6-5-10-3-2-4-12(13(10)7-11)14-8-15-9-16-14/h4-9H,2-3H2,1H3,(H,15,16) | PDB
UniProtKB/SwissProt
GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 1.57E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Tennessee
Curated by ChEMBL
| Assay Description Displacement of [3H]rauwolscine from Alpha-2 adrenergic receptor of rat brain membranes |
J Med Chem 40: 3014-24 (1997)
Article DOI: 10.1021/jm960642q BindingDB Entry DOI: 10.7270/Q2ZG6VZ9 |
More data for this Ligand-Target Pair | |
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor
(Rattus norvegicus (rat)-Rattus norvegicus (Rat)) | BDBM50471339
(CHEMBL103500)Show InChI InChI=1S/C14H14N2O/c1-17-11-5-6-12-10(7-11)3-2-4-13(12)14-8-15-9-16-14/h4-9H,2-3H2,1H3,(H,15,16) | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 1.63E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Tennessee
Curated by ChEMBL
| Assay Description Displacement of [3H]-prazosin from Alpha-1 adrenergic receptor of rat brain membranes |
J Med Chem 40: 3014-24 (1997)
Article DOI: 10.1021/jm960642q BindingDB Entry DOI: 10.7270/Q2ZG6VZ9 |
More data for this Ligand-Target Pair | |
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor
(Rattus norvegicus (rat)-Rattus norvegicus (Rat)) | BDBM50470859
(CHEMBL105487)Show InChI InChI=1S/C15H12N2/c1-11(15-9-16-10-17-15)13-8-4-6-12-5-2-3-7-14(12)13/h2-10H,1H2,(H,16,17) | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 1.73E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Ohio State University
Curated by ChEMBL
| Assay Description Alpha-1 adrenergic receptor binding affinity in rat brain membranes |
J Med Chem 39: 3001-13 (1996)
Article DOI: 10.1021/jm9506074 BindingDB Entry DOI: 10.7270/Q2BV7KBH |
More data for this Ligand-Target Pair | |
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor
(Rattus norvegicus (rat)-Rattus norvegicus (Rat)) | BDBM50471348
(CHEMBL103448)Show InChI InChI=1S/C14H16N2O/c1-17-11-6-5-10-3-2-4-12(13(10)7-11)14-8-15-9-16-14/h5-9,12H,2-4H2,1H3,(H,15,16) | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 1.77E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Tennessee
Curated by ChEMBL
| Assay Description Displacement of [3H]-prazosin from Alpha-1 adrenergic receptor of rat brain membranes |
J Med Chem 40: 3014-24 (1997)
Article DOI: 10.1021/jm960642q BindingDB Entry DOI: 10.7270/Q2ZG6VZ9 |
More data for this Ligand-Target Pair | |
Alpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor
(RAT-NEONATAL RAT-Rattus norvegicus (rat)) | BDBM50470861
(CHEMBL322844)Show InChI InChI=1S/C16H14N2/c1-2-13(16-10-17-11-18-16)15-9-5-7-12-6-3-4-8-14(12)15/h2-11H,1H3,(H,17,18)/b13-2- | PDB
UniProtKB/SwissProt
GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 1.89E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Ohio State University
Curated by ChEMBL
| Assay Description Alpha-2 adrenergic receptor binding affinity was tested against membrane preparations of rat brain using 0.2 nM [3H]rauwolscine as radioligand |
J Med Chem 39: 3001-13 (1996)
Article DOI: 10.1021/jm9506074 BindingDB Entry DOI: 10.7270/Q2BV7KBH |
More data for this Ligand-Target Pair | |
Alpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor
(RAT-NEONATAL RAT-Rattus norvegicus (rat)) | BDBM50471341
(CHEMBL103438)Show SMILES C(Oc1cccc2C(=CCCc12)c1c[nH]cn1)c1ccccc1 |c:7| Show InChI InChI=1S/C20H18N2O/c1-2-6-15(7-3-1)13-23-20-11-5-8-16-17(9-4-10-18(16)20)19-12-21-14-22-19/h1-3,5-9,11-12,14H,4,10,13H2,(H,21,22) | PDB
UniProtKB/SwissProt
GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 2.67E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Tennessee
Curated by ChEMBL
| Assay Description Displacement of [3H]rauwolscine from Alpha-2 adrenergic receptor of rat brain membranes |
J Med Chem 40: 3014-24 (1997)
Article DOI: 10.1021/jm960642q BindingDB Entry DOI: 10.7270/Q2ZG6VZ9 |
More data for this Ligand-Target Pair | |
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor
(Rattus norvegicus (rat)-Rattus norvegicus (Rat)) | BDBM50471344
(CHEMBL422247)Show InChI InChI=1S/C15H16N2/c1-10-6-11(2)12-4-3-5-13(14(12)7-10)15-8-16-9-17-15/h5-9H,3-4H2,1-2H3,(H,16,17) | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 2.96E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Tennessee
Curated by ChEMBL
| Assay Description Displacement of [3H]-prazosin from Alpha-1 adrenergic receptor of rat brain membranes |
J Med Chem 40: 3014-24 (1997)
Article DOI: 10.1021/jm960642q BindingDB Entry DOI: 10.7270/Q2ZG6VZ9 |
More data for this Ligand-Target Pair | |
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor
(Rattus norvegicus (rat)-Rattus norvegicus (Rat)) | BDBM50471349
(CHEMBL321964)Show InChI InChI=1S/C14H14N2O/c1-17-14-7-3-4-10-11(5-2-6-12(10)14)13-8-15-9-16-13/h3-5,7-9H,2,6H2,1H3,(H,15,16) | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 2.97E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Tennessee
Curated by ChEMBL
| Assay Description Displacement of [3H]-prazosin from Alpha-1 adrenergic receptor of rat brain membranes |
J Med Chem 40: 3014-24 (1997)
Article DOI: 10.1021/jm960642q BindingDB Entry DOI: 10.7270/Q2ZG6VZ9 |
More data for this Ligand-Target Pair | |
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor
(Rattus norvegicus (rat)-Rattus norvegicus (Rat)) | BDBM50471341
(CHEMBL103438)Show SMILES C(Oc1cccc2C(=CCCc12)c1c[nH]cn1)c1ccccc1 |c:7| Show InChI InChI=1S/C20H18N2O/c1-2-6-15(7-3-1)13-23-20-11-5-8-16-17(9-4-10-18(16)20)19-12-21-14-22-19/h1-3,5-9,11-12,14H,4,10,13H2,(H,21,22) | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 8.25E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Tennessee
Curated by ChEMBL
| Assay Description Displacement of [3H]-prazosin from Alpha-1 adrenergic receptor of rat brain membranes |
J Med Chem 40: 3014-24 (1997)
Article DOI: 10.1021/jm960642q BindingDB Entry DOI: 10.7270/Q2ZG6VZ9 |
More data for this Ligand-Target Pair | |
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor
(Rattus norvegicus (rat)-Rattus norvegicus (Rat)) | BDBM50223426
(CHEBI:10304 | Corbadrine | Levonordefrin | Neo-Cob...)Show SMILES [H][C@@](C)(N)[C@]([H])(O)c1ccc(O)c(O)c1 |r| Show InChI InChI=1S/C9H13NO3/c1-5(10)9(13)6-2-3-7(11)8(12)4-6/h2-5,9,11-13H,10H2,1H3/t5-,9-/m0/s1 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank GoogleScholar AffyNet
| Purchase
MCE KEGG PC cid PC sid UniChem
Similars
| Article PubMed
| 9.22E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Ohio State University
Curated by ChEMBL
| Assay Description Alpha-1 adrenergic receptor binding affinity in rat brain membranes |
J Med Chem 39: 3001-13 (1996)
Article DOI: 10.1021/jm9506074 BindingDB Entry DOI: 10.7270/Q2BV7KBH |
More data for this Ligand-Target Pair | |
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor
(Rattus norvegicus (rat)-Rattus norvegicus (Rat)) | BDBM50471345
(CHEMBL102538)Show InChI InChI=1S/C14H14N2O/c1-17-11-6-5-10-3-2-4-12(13(10)7-11)14-8-15-9-16-14/h4-9H,2-3H2,1H3,(H,15,16) | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 1.42E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Tennessee
Curated by ChEMBL
| Assay Description Displacement of [3H]-prazosin from Alpha-1 adrenergic receptor of rat brain membranes |
J Med Chem 40: 3014-24 (1997)
Article DOI: 10.1021/jm960642q BindingDB Entry DOI: 10.7270/Q2ZG6VZ9 |
More data for this Ligand-Target Pair | |
Alpha-2A/Alpha-2B/Alpha-2C adrenergic receptor
(Homo sapiens (Human)) | BDBM50001922
(2-Naphthalen-1-ylmethyl-4,5-dihydro-1H-imidazole; ...)Show InChI InChI=1S/C14H14N2/c1-2-7-13-11(4-1)5-3-6-12(13)10-14-15-8-9-16-14/h1-7H,8-10H2,(H,15,16) | PDB
KEGG
UniProtKB/SwissProt
DrugBank antibodypedia antibodypedia GoogleScholar AffyNet
| Purchase
CHEMBL DrugBank MCE KEGG PC cid PC sid UniChem
Similars
| DrugBank PubMed
| n/a | n/a | 0.00110 | n/a | n/a | n/a | n/a | n/a | n/a |
Ohio State University
Curated by ChEMBL
| Assay Description Compound was evaluated for Adrenergic activity against Alpha-2 adrenergic receptor in human platelets |
J Med Chem 35: 750-5 (1992)
BindingDB Entry DOI: 10.7270/Q27H1MTJ |
More data for this Ligand-Target Pair | |
Alpha-2A/Alpha-2B/Alpha-2C adrenergic receptor
(Homo sapiens (Human)) | BDBM50230389
(CHEMBL541105)Show InChI InChI=1S/C15H14N2.ClH/c1-11(15-9-16-10-17-15)13-8-4-6-12-5-2-3-7-14(12)13;/h2-11H,1H3,(H,16,17);1H | PDB
KEGG
UniProtKB/SwissProt
DrugBank antibodypedia antibodypedia GoogleScholar AffyNet
| Purchase
CHEMBL PC cid PC sid UniChem
Similars
| PubMed
| n/a | n/a | 0.00340 | n/a | n/a | n/a | n/a | n/a | n/a |
Ohio State University
Curated by ChEMBL
| Assay Description Compound was tested for Adrenergic activity against Alpha-2 adrenergic receptor from rat aorta |
J Med Chem 35: 750-5 (1992)
BindingDB Entry DOI: 10.7270/Q27H1MTJ |
More data for this Ligand-Target Pair | |
Alpha-2A/Alpha-2B/Alpha-2C adrenergic receptor
(Homo sapiens (Human)) | BDBM50230393
(CHEMBL553231)Show InChI InChI=1S/C15H16N2.ClH/c1-11(15-16-9-10-17-15)13-8-4-6-12-5-2-3-7-14(12)13;/h2-8,11H,9-10H2,1H3,(H,16,17);1H | PDB
KEGG
UniProtKB/SwissProt
DrugBank antibodypedia antibodypedia GoogleScholar AffyNet
| CHEMBL PC cid PC sid UniChem
Similars
| PubMed
| n/a | n/a | 0.0140 | n/a | n/a | n/a | n/a | n/a | n/a |
Ohio State University
Curated by ChEMBL
| Assay Description Compound was evaluated for Adrenergic activity against Alpha-2 adrenergic receptor in human platelets |
J Med Chem 35: 750-5 (1992)
BindingDB Entry DOI: 10.7270/Q27H1MTJ |
More data for this Ligand-Target Pair | |
Alpha-2A/Alpha-2B/Alpha-2C adrenergic receptor
(Homo sapiens (Human)) | BDBM50230395
(CHEMBL557985)Show InChI InChI=1S/C15H16N2.ClH/c1-11(15-16-8-9-17-15)13-7-6-12-4-2-3-5-14(12)10-13;/h2-7,10-11H,8-9H2,1H3,(H,16,17);1H | PDB
KEGG
UniProtKB/SwissProt
DrugBank antibodypedia antibodypedia GoogleScholar AffyNet
| CHEMBL PC cid PC sid UniChem
| PubMed
| n/a | n/a | 0.0160 | n/a | n/a | n/a | n/a | n/a | n/a |
Ohio State University
Curated by ChEMBL
| Assay Description Compound was evaluated for Adrenergic activity against Alpha-2 adrenergic receptor in human platelets |
J Med Chem 35: 750-5 (1992)
BindingDB Entry DOI: 10.7270/Q27H1MTJ |
More data for this Ligand-Target Pair | |