Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Glucose-dependent insulinotropic receptor (Homo sapiens (Human)) | BDBM50387888 (CHEMBL2058398) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 86 | n/a | n/a | n/a | n/a |
Sanwa Kagaku Kenkyusho Co., Ltd Curated by ChEMBL | Assay Description Agonist activity at human GPR119 receptor expressed in CHO-K1 cells assessed as cAMP accumulation after 30 mins by HTRF assay | Bioorg Med Chem Lett 22: 5123-8 (2012) Article DOI: 10.1016/j.bmcl.2012.05.117 BindingDB Entry DOI: 10.7270/Q2TD9ZC4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Homo sapiens (Human)) | BDBM50387901 (CHEMBL2058402) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.03E+3 | n/a | n/a | n/a | n/a |
Sanwa Kagaku Kenkyusho Co., Ltd Curated by ChEMBL | Assay Description Agonist activity at human GPR119 receptor expressed in CHO-K1 cells assessed as cAMP accumulation after 30 mins by HTRF assay | Bioorg Med Chem Lett 22: 5123-8 (2012) Article DOI: 10.1016/j.bmcl.2012.05.117 BindingDB Entry DOI: 10.7270/Q2TD9ZC4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Homo sapiens (Human)) | BDBM50387890 (CHEMBL2058388) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 2.61E+3 | n/a | n/a | n/a | n/a |
Sanwa Kagaku Kenkyusho Co., Ltd Curated by ChEMBL | Assay Description Agonist activity at human GPR119 receptor expressed in CHO-K1 cells assessed as cAMP accumulation after 30 mins by HTRF assay | Bioorg Med Chem Lett 22: 5123-8 (2012) Article DOI: 10.1016/j.bmcl.2012.05.117 BindingDB Entry DOI: 10.7270/Q2TD9ZC4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Homo sapiens (Human)) | BDBM50387891 (CHEMBL2058389) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 210 | n/a | n/a | n/a | n/a |
Sanwa Kagaku Kenkyusho Co., Ltd Curated by ChEMBL | Assay Description Agonist activity at human GPR119 receptor expressed in CHO-K1 cells assessed as cAMP accumulation after 30 mins by HTRF assay | Bioorg Med Chem Lett 22: 5123-8 (2012) Article DOI: 10.1016/j.bmcl.2012.05.117 BindingDB Entry DOI: 10.7270/Q2TD9ZC4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Homo sapiens (Human)) | BDBM50387892 (CHEMBL2058390) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 145 | n/a | n/a | n/a | n/a |
Sanwa Kagaku Kenkyusho Co., Ltd Curated by ChEMBL | Assay Description Agonist activity at human GPR119 receptor expressed in CHO-K1 cells assessed as cAMP accumulation after 30 mins by HTRF assay | Bioorg Med Chem Lett 22: 5123-8 (2012) Article DOI: 10.1016/j.bmcl.2012.05.117 BindingDB Entry DOI: 10.7270/Q2TD9ZC4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Homo sapiens (Human)) | BDBM50387893 (CHEMBL2058391) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 270 | n/a | n/a | n/a | n/a |
Sanwa Kagaku Kenkyusho Co., Ltd Curated by ChEMBL | Assay Description Agonist activity at human GPR119 receptor expressed in CHO-K1 cells assessed as cAMP accumulation after 30 mins by HTRF assay | Bioorg Med Chem Lett 22: 5123-8 (2012) Article DOI: 10.1016/j.bmcl.2012.05.117 BindingDB Entry DOI: 10.7270/Q2TD9ZC4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Homo sapiens (Human)) | BDBM50387894 (CHEMBL2058394) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 736 | n/a | n/a | n/a | n/a |
Sanwa Kagaku Kenkyusho Co., Ltd Curated by ChEMBL | Assay Description Agonist activity at human GPR119 receptor expressed in CHO-K1 cells assessed as cAMP accumulation after 30 mins by HTRF assay | Bioorg Med Chem Lett 22: 5123-8 (2012) Article DOI: 10.1016/j.bmcl.2012.05.117 BindingDB Entry DOI: 10.7270/Q2TD9ZC4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Homo sapiens (Human)) | BDBM50387895 (CHEMBL2058395) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 254 | n/a | n/a | n/a | n/a |
Sanwa Kagaku Kenkyusho Co., Ltd Curated by ChEMBL | Assay Description Agonist activity at human GPR119 receptor expressed in CHO-K1 cells assessed as cAMP accumulation after 30 mins by HTRF assay | Bioorg Med Chem Lett 22: 5123-8 (2012) Article DOI: 10.1016/j.bmcl.2012.05.117 BindingDB Entry DOI: 10.7270/Q2TD9ZC4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Homo sapiens (Human)) | BDBM50387896 (CHEMBL2058396) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 511 | n/a | n/a | n/a | n/a |
Sanwa Kagaku Kenkyusho Co., Ltd Curated by ChEMBL | Assay Description Agonist activity at human GPR119 receptor expressed in CHO-K1 cells assessed as cAMP accumulation after 30 mins by HTRF assay | Bioorg Med Chem Lett 22: 5123-8 (2012) Article DOI: 10.1016/j.bmcl.2012.05.117 BindingDB Entry DOI: 10.7270/Q2TD9ZC4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Homo sapiens (Human)) | BDBM50387897 (CHEMBL2058397) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 268 | n/a | n/a | n/a | n/a |
Sanwa Kagaku Kenkyusho Co., Ltd Curated by ChEMBL | Assay Description Agonist activity at human GPR119 receptor expressed in CHO-K1 cells assessed as cAMP accumulation after 30 mins by HTRF assay | Bioorg Med Chem Lett 22: 5123-8 (2012) Article DOI: 10.1016/j.bmcl.2012.05.117 BindingDB Entry DOI: 10.7270/Q2TD9ZC4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Homo sapiens (Human)) | BDBM50387898 (CHEMBL2058399) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 770 | n/a | n/a | n/a | n/a |
Sanwa Kagaku Kenkyusho Co., Ltd Curated by ChEMBL | Assay Description Agonist activity at human GPR119 receptor expressed in CHO-K1 cells assessed as cAMP accumulation after 30 mins by HTRF assay | Bioorg Med Chem Lett 22: 5123-8 (2012) Article DOI: 10.1016/j.bmcl.2012.05.117 BindingDB Entry DOI: 10.7270/Q2TD9ZC4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Homo sapiens (Human)) | BDBM50387899 (CHEMBL2058400) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 52 | n/a | n/a | n/a | n/a |
Sanwa Kagaku Kenkyusho Co., Ltd Curated by ChEMBL | Assay Description Agonist activity at human GPR119 receptor expressed in CHO-K1 cells assessed as cAMP accumulation after 30 mins by HTRF assay | Bioorg Med Chem Lett 22: 5123-8 (2012) Article DOI: 10.1016/j.bmcl.2012.05.117 BindingDB Entry DOI: 10.7270/Q2TD9ZC4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Homo sapiens (Human)) | BDBM50387902 (CHEMBL2058403) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 46 | n/a | n/a | n/a | n/a |
Sanwa Kagaku Kenkyusho Co., Ltd Curated by ChEMBL | Assay Description Agonist activity at human GPR119 receptor expressed in CHO-K1 cells assessed as cAMP accumulation after 30 mins by HTRF assay | Bioorg Med Chem Lett 22: 5123-8 (2012) Article DOI: 10.1016/j.bmcl.2012.05.117 BindingDB Entry DOI: 10.7270/Q2TD9ZC4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Homo sapiens (Human)) | BDBM50387903 (CHEMBL2058404) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 88 | n/a | n/a | n/a | n/a |
Sanwa Kagaku Kenkyusho Co., Ltd Curated by ChEMBL | Assay Description Agonist activity at human GPR119 receptor expressed in CHO-K1 cells assessed as cAMP accumulation after 30 mins by HTRF assay | Bioorg Med Chem Lett 22: 5123-8 (2012) Article DOI: 10.1016/j.bmcl.2012.05.117 BindingDB Entry DOI: 10.7270/Q2TD9ZC4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Homo sapiens (Human)) | BDBM50387904 (CHEMBL2058405) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 272 | n/a | n/a | n/a | n/a |
Sanwa Kagaku Kenkyusho Co., Ltd Curated by ChEMBL | Assay Description Agonist activity at human GPR119 receptor expressed in CHO-K1 cells assessed as cAMP accumulation after 30 mins by HTRF assay | Bioorg Med Chem Lett 22: 5123-8 (2012) Article DOI: 10.1016/j.bmcl.2012.05.117 BindingDB Entry DOI: 10.7270/Q2TD9ZC4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Homo sapiens (Human)) | BDBM50387905 (CHEMBL2058406) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 734 | n/a | n/a | n/a | n/a |
Sanwa Kagaku Kenkyusho Co., Ltd Curated by ChEMBL | Assay Description Agonist activity at human GPR119 receptor expressed in CHO-K1 cells assessed as cAMP accumulation after 30 mins by HTRF assay | Bioorg Med Chem Lett 22: 5123-8 (2012) Article DOI: 10.1016/j.bmcl.2012.05.117 BindingDB Entry DOI: 10.7270/Q2TD9ZC4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Homo sapiens (Human)) | BDBM50387889 (CHEMBL2058666) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 117 | n/a | n/a | n/a | n/a |
Sanwa Kagaku Kenkyusho Co., Ltd Curated by ChEMBL | Assay Description Agonist activity at human GPR119 receptor expressed in CHO-K1 cells assessed as cAMP accumulation after 30 mins by HTRF assay | Bioorg Med Chem Lett 22: 5123-8 (2012) Article DOI: 10.1016/j.bmcl.2012.05.117 BindingDB Entry DOI: 10.7270/Q2TD9ZC4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Homo sapiens (Human)) | BDBM50387906 (CHEMBL2058667) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 115 | n/a | n/a | n/a | n/a |
Sanwa Kagaku Kenkyusho Co., Ltd Curated by ChEMBL | Assay Description Agonist activity at human GPR119 receptor expressed in CHO-K1 cells assessed as cAMP accumulation after 30 mins by HTRF assay | Bioorg Med Chem Lett 22: 5123-8 (2012) Article DOI: 10.1016/j.bmcl.2012.05.117 BindingDB Entry DOI: 10.7270/Q2TD9ZC4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Homo sapiens (Human)) | BDBM50387907 (CHEMBL2058668) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 149 | n/a | n/a | n/a | n/a |
Sanwa Kagaku Kenkyusho Co., Ltd Curated by ChEMBL | Assay Description Agonist activity at human GPR119 receptor expressed in CHO-K1 cells assessed as cAMP accumulation after 30 mins by HTRF assay | Bioorg Med Chem Lett 22: 5123-8 (2012) Article DOI: 10.1016/j.bmcl.2012.05.117 BindingDB Entry DOI: 10.7270/Q2TD9ZC4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Homo sapiens (Human)) | BDBM50387908 (CHEMBL2058669) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 73 | n/a | n/a | n/a | n/a |
Sanwa Kagaku Kenkyusho Co., Ltd Curated by ChEMBL | Assay Description Agonist activity at human GPR119 receptor expressed in CHO-K1 cells assessed as cAMP accumulation after 30 mins by HTRF assay | Bioorg Med Chem Lett 22: 5123-8 (2012) Article DOI: 10.1016/j.bmcl.2012.05.117 BindingDB Entry DOI: 10.7270/Q2TD9ZC4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Homo sapiens (Human)) | BDBM50387909 (CHEMBL2058670) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 161 | n/a | n/a | n/a | n/a |
Sanwa Kagaku Kenkyusho Co., Ltd Curated by ChEMBL | Assay Description Agonist activity at human GPR119 receptor expressed in CHO-K1 cells assessed as cAMP accumulation after 30 mins by HTRF assay | Bioorg Med Chem Lett 22: 5123-8 (2012) Article DOI: 10.1016/j.bmcl.2012.05.117 BindingDB Entry DOI: 10.7270/Q2TD9ZC4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Homo sapiens (Human)) | BDBM50387910 (CHEMBL2058671) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 704 | n/a | n/a | n/a | n/a |
Sanwa Kagaku Kenkyusho Co., Ltd Curated by ChEMBL | Assay Description Agonist activity at human GPR119 receptor expressed in CHO-K1 cells assessed as cAMP accumulation after 30 mins by HTRF assay | Bioorg Med Chem Lett 22: 5123-8 (2012) Article DOI: 10.1016/j.bmcl.2012.05.117 BindingDB Entry DOI: 10.7270/Q2TD9ZC4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Homo sapiens (Human)) | BDBM50387911 (CHEMBL2058672) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 121 | n/a | n/a | n/a | n/a |
Sanwa Kagaku Kenkyusho Co., Ltd Curated by ChEMBL | Assay Description Agonist activity at human GPR119 receptor expressed in CHO-K1 cells assessed as cAMP accumulation after 30 mins by HTRF assay | Bioorg Med Chem Lett 22: 5123-8 (2012) Article DOI: 10.1016/j.bmcl.2012.05.117 BindingDB Entry DOI: 10.7270/Q2TD9ZC4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Homo sapiens (Human)) | BDBM50387912 (CHEMBL2058673) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 51 | n/a | n/a | n/a | n/a |
Sanwa Kagaku Kenkyusho Co., Ltd Curated by ChEMBL | Assay Description Agonist activity at human GPR119 receptor expressed in CHO-K1 cells assessed as cAMP accumulation after 30 mins by HTRF assay | Bioorg Med Chem Lett 22: 5123-8 (2012) Article DOI: 10.1016/j.bmcl.2012.05.117 BindingDB Entry DOI: 10.7270/Q2TD9ZC4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Homo sapiens (Human)) | BDBM50387913 (CHEMBL2058674) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 58 | n/a | n/a | n/a | n/a |
Sanwa Kagaku Kenkyusho Co., Ltd Curated by ChEMBL | Assay Description Agonist activity at human GPR119 receptor expressed in CHO-K1 cells assessed as cAMP accumulation after 30 mins by HTRF assay | Bioorg Med Chem Lett 22: 5123-8 (2012) Article DOI: 10.1016/j.bmcl.2012.05.117 BindingDB Entry DOI: 10.7270/Q2TD9ZC4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Mus musculus) | BDBM50387893 (CHEMBL2058391) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 224 | n/a | n/a | n/a | n/a |
Sanwa Kagaku Kenkyusho Co., Ltd Curated by ChEMBL | Assay Description Agonist activity at mouse GPR119 receptor expressed in CHO-K1 cells assessed as cAMP accumulation after 30 mins by HTRF assay | Bioorg Med Chem Lett 22: 5123-8 (2012) Article DOI: 10.1016/j.bmcl.2012.05.117 BindingDB Entry DOI: 10.7270/Q2TD9ZC4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Mus musculus) | BDBM50387895 (CHEMBL2058395) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 266 | n/a | n/a | n/a | n/a |
Sanwa Kagaku Kenkyusho Co., Ltd Curated by ChEMBL | Assay Description Agonist activity at mouse GPR119 receptor expressed in CHO-K1 cells assessed as cAMP accumulation after 30 mins by HTRF assay | Bioorg Med Chem Lett 22: 5123-8 (2012) Article DOI: 10.1016/j.bmcl.2012.05.117 BindingDB Entry DOI: 10.7270/Q2TD9ZC4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Mus musculus) | BDBM50387897 (CHEMBL2058397) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 331 | n/a | n/a | n/a | n/a |
Sanwa Kagaku Kenkyusho Co., Ltd Curated by ChEMBL | Assay Description Agonist activity at mouse GPR119 receptor expressed in CHO-K1 cells assessed as cAMP accumulation after 30 mins by HTRF assay | Bioorg Med Chem Lett 22: 5123-8 (2012) Article DOI: 10.1016/j.bmcl.2012.05.117 BindingDB Entry DOI: 10.7270/Q2TD9ZC4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Mus musculus) | BDBM50387888 (CHEMBL2058398) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 87 | n/a | n/a | n/a | n/a |
Sanwa Kagaku Kenkyusho Co., Ltd Curated by ChEMBL | Assay Description Agonist activity at mouse GPR119 receptor expressed in CHO-K1 cells assessed as cAMP accumulation after 30 mins by HTRF assay | Bioorg Med Chem Lett 22: 5123-8 (2012) Article DOI: 10.1016/j.bmcl.2012.05.117 BindingDB Entry DOI: 10.7270/Q2TD9ZC4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Mus musculus) | BDBM50387899 (CHEMBL2058400) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 66 | n/a | n/a | n/a | n/a |
Sanwa Kagaku Kenkyusho Co., Ltd Curated by ChEMBL | Assay Description Agonist activity at mouse GPR119 receptor expressed in CHO-K1 cells assessed as cAMP accumulation after 30 mins by HTRF assay | Bioorg Med Chem Lett 22: 5123-8 (2012) Article DOI: 10.1016/j.bmcl.2012.05.117 BindingDB Entry DOI: 10.7270/Q2TD9ZC4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Mus musculus) | BDBM50387900 (CHEMBL2058401) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 515 | n/a | n/a | n/a | n/a |
Sanwa Kagaku Kenkyusho Co., Ltd Curated by ChEMBL | Assay Description Agonist activity at mouse GPR119 receptor expressed in CHO-K1 cells assessed as cAMP accumulation after 30 mins by HTRF assay | Bioorg Med Chem Lett 22: 5123-8 (2012) Article DOI: 10.1016/j.bmcl.2012.05.117 BindingDB Entry DOI: 10.7270/Q2TD9ZC4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Mus musculus) | BDBM50387902 (CHEMBL2058403) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 123 | n/a | n/a | n/a | n/a |
Sanwa Kagaku Kenkyusho Co., Ltd Curated by ChEMBL | Assay Description Agonist activity at mouse GPR119 receptor expressed in CHO-K1 cells assessed as cAMP accumulation after 30 mins by HTRF assay | Bioorg Med Chem Lett 22: 5123-8 (2012) Article DOI: 10.1016/j.bmcl.2012.05.117 BindingDB Entry DOI: 10.7270/Q2TD9ZC4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Mus musculus) | BDBM50387903 (CHEMBL2058404) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 262 | n/a | n/a | n/a | n/a |
Sanwa Kagaku Kenkyusho Co., Ltd Curated by ChEMBL | Assay Description Agonist activity at mouse GPR119 receptor expressed in CHO-K1 cells assessed as cAMP accumulation after 30 mins by HTRF assay | Bioorg Med Chem Lett 22: 5123-8 (2012) Article DOI: 10.1016/j.bmcl.2012.05.117 BindingDB Entry DOI: 10.7270/Q2TD9ZC4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Mus musculus) | BDBM50387904 (CHEMBL2058405) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 351 | n/a | n/a | n/a | n/a |
Sanwa Kagaku Kenkyusho Co., Ltd Curated by ChEMBL | Assay Description Agonist activity at mouse GPR119 receptor expressed in CHO-K1 cells assessed as cAMP accumulation after 30 mins by HTRF assay | Bioorg Med Chem Lett 22: 5123-8 (2012) Article DOI: 10.1016/j.bmcl.2012.05.117 BindingDB Entry DOI: 10.7270/Q2TD9ZC4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Mus musculus) | BDBM50387905 (CHEMBL2058406) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 892 | n/a | n/a | n/a | n/a |
Sanwa Kagaku Kenkyusho Co., Ltd Curated by ChEMBL | Assay Description Agonist activity at mouse GPR119 receptor expressed in CHO-K1 cells assessed as cAMP accumulation after 30 mins by HTRF assay | Bioorg Med Chem Lett 22: 5123-8 (2012) Article DOI: 10.1016/j.bmcl.2012.05.117 BindingDB Entry DOI: 10.7270/Q2TD9ZC4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Mus musculus) | BDBM50387906 (CHEMBL2058667) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 60 | n/a | n/a | n/a | n/a |
Sanwa Kagaku Kenkyusho Co., Ltd Curated by ChEMBL | Assay Description Agonist activity at mouse GPR119 receptor expressed in CHO-K1 cells assessed as cAMP accumulation after 30 mins by HTRF assay | Bioorg Med Chem Lett 22: 5123-8 (2012) Article DOI: 10.1016/j.bmcl.2012.05.117 BindingDB Entry DOI: 10.7270/Q2TD9ZC4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Mus musculus) | BDBM50387907 (CHEMBL2058668) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 139 | n/a | n/a | n/a | n/a |
Sanwa Kagaku Kenkyusho Co., Ltd Curated by ChEMBL | Assay Description Agonist activity at mouse GPR119 receptor expressed in CHO-K1 cells assessed as cAMP accumulation after 30 mins by HTRF assay | Bioorg Med Chem Lett 22: 5123-8 (2012) Article DOI: 10.1016/j.bmcl.2012.05.117 BindingDB Entry DOI: 10.7270/Q2TD9ZC4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Mus musculus) | BDBM50387910 (CHEMBL2058671) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 1.02E+3 | n/a | n/a | n/a | n/a |
Sanwa Kagaku Kenkyusho Co., Ltd Curated by ChEMBL | Assay Description Agonist activity at mouse GPR119 receptor expressed in CHO-K1 cells assessed as cAMP accumulation after 30 mins by HTRF assay | Bioorg Med Chem Lett 22: 5123-8 (2012) Article DOI: 10.1016/j.bmcl.2012.05.117 BindingDB Entry DOI: 10.7270/Q2TD9ZC4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Mus musculus) | BDBM50387911 (CHEMBL2058672) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 812 | n/a | n/a | n/a | n/a |
Sanwa Kagaku Kenkyusho Co., Ltd Curated by ChEMBL | Assay Description Agonist activity at mouse GPR119 receptor expressed in CHO-K1 cells assessed as cAMP accumulation after 30 mins by HTRF assay | Bioorg Med Chem Lett 22: 5123-8 (2012) Article DOI: 10.1016/j.bmcl.2012.05.117 BindingDB Entry DOI: 10.7270/Q2TD9ZC4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Mus musculus) | BDBM50387912 (CHEMBL2058673) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 167 | n/a | n/a | n/a | n/a |
Sanwa Kagaku Kenkyusho Co., Ltd Curated by ChEMBL | Assay Description Agonist activity at mouse GPR119 receptor expressed in CHO-K1 cells assessed as cAMP accumulation after 30 mins by HTRF assay | Bioorg Med Chem Lett 22: 5123-8 (2012) Article DOI: 10.1016/j.bmcl.2012.05.117 BindingDB Entry DOI: 10.7270/Q2TD9ZC4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Mus musculus) | BDBM50387913 (CHEMBL2058674) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 158 | n/a | n/a | n/a | n/a |
Sanwa Kagaku Kenkyusho Co., Ltd Curated by ChEMBL | Assay Description Agonist activity at mouse GPR119 receptor expressed in CHO-K1 cells assessed as cAMP accumulation after 30 mins by HTRF assay | Bioorg Med Chem Lett 22: 5123-8 (2012) Article DOI: 10.1016/j.bmcl.2012.05.117 BindingDB Entry DOI: 10.7270/Q2TD9ZC4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Homo sapiens (Human)) | BDBM50387900 (CHEMBL2058401) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 550 | n/a | n/a | n/a | n/a |
Sanwa Kagaku Kenkyusho Co., Ltd Curated by ChEMBL | Assay Description Agonist activity at human GPR119 receptor expressed in CHO-K1 cells assessed as cAMP accumulation after 30 mins by HTRF assay | Bioorg Med Chem Lett 22: 5123-8 (2012) Article DOI: 10.1016/j.bmcl.2012.05.117 BindingDB Entry DOI: 10.7270/Q2TD9ZC4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Mus musculus) | BDBM50387889 (CHEMBL2058666) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 159 | n/a | n/a | n/a | n/a |
Sanwa Kagaku Kenkyusho Co., Ltd Curated by ChEMBL | Assay Description Agonist activity at mouse GPR119 receptor expressed in CHO-K1 cells assessed as cAMP accumulation after 30 mins by HTRF assay | Bioorg Med Chem Lett 22: 5123-8 (2012) Article DOI: 10.1016/j.bmcl.2012.05.117 BindingDB Entry DOI: 10.7270/Q2TD9ZC4 | |||||||||||
More data for this Ligand-Target Pair |