Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Beta-glucuronidase (Escherichia coli (Enterobacteria)) | BDBM152586 (D-Saccharic acid 1,4 lactone | D-Saccharic acid 1,...) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 4.84E+4 | n/a | n/a | n/a | n/a | 7.0 | 37 |
University of Karachi | Assay Description β-Glucuronidase inhibitory activity was evaluated by a biochemical assay, based on the measurement of the absorbance of p-nitrophenol at 405 nm,... | J Enzyme Inhib Med Chem 27: 348-55 (2012) Article DOI: 10.3109/14756366.2011.590804 BindingDB Entry DOI: 10.7270/Q2N29VV5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-glucuronidase (Escherichia coli (Enterobacteria)) | BDBM50223368 (3beta-hydroxyandrost-5-en-17-one | CHEMBL90593 | D...) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG MMDB PC cid PC sid PDB UniChem Patents Similars | Article PubMed | n/a | n/a | 7.79E+4 | n/a | n/a | n/a | n/a | 7.0 | 37 |
University of Karachi | Assay Description β-Glucuronidase inhibitory activity was evaluated by a biochemical assay, based on the measurement of the absorbance of p-nitrophenol at 405 nm,... | J Enzyme Inhib Med Chem 27: 348-55 (2012) Article DOI: 10.3109/14756366.2011.590804 BindingDB Entry DOI: 10.7270/Q2N29VV5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-glucuronidase (Escherichia coli (Enterobacteria)) | BDBM236514 (Androst-4-ene-3β,7β,17β-triol (8)) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.91E+5 | n/a | n/a | n/a | n/a | 7.0 | 37 |
University of Karachi | Assay Description β-Glucuronidase inhibitory activity was evaluated by a biochemical assay, based on the measurement of the absorbance of p-nitrophenol at 405 nm,... | J Enzyme Inhib Med Chem 27: 348-55 (2012) Article DOI: 10.3109/14756366.2011.590804 BindingDB Entry DOI: 10.7270/Q2N29VV5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-glucuronidase (Escherichia coli (Enterobacteria)) | BDBM236513 (Androst-4-ene-3β-ol-6,17-dione (7)) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 2.22E+5 | n/a | n/a | n/a | n/a | 7.0 | 37 |
University of Karachi | Assay Description β-Glucuronidase inhibitory activity was evaluated by a biochemical assay, based on the measurement of the absorbance of p-nitrophenol at 405 nm,... | J Enzyme Inhib Med Chem 27: 348-55 (2012) Article DOI: 10.3109/14756366.2011.590804 BindingDB Entry DOI: 10.7270/Q2N29VV5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-glucuronidase (Escherichia coli (Enterobacteria)) | BDBM236512 (Androstane-3,17-dione (2)) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.74E+5 | n/a | n/a | n/a | n/a | 7.0 | 37 |
University of Karachi | Assay Description β-Glucuronidase inhibitory activity was evaluated by a biochemical assay, based on the measurement of the absorbance of p-nitrophenol at 405 nm,... | J Enzyme Inhib Med Chem 27: 348-55 (2012) Article DOI: 10.3109/14756366.2011.590804 BindingDB Entry DOI: 10.7270/Q2N29VV5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-glucuronidase (Escherichia coli (Enterobacteria)) | BDBM91713 (Androst-4-en-3,17-dione, 2 | Androst-4-ene-3,17-di...) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase DrugBank KEGG MMDB PC cid PC sid PDB UniChem Patents Similars | Article PubMed | n/a | n/a | 4.30E+5 | n/a | n/a | n/a | n/a | 7.0 | 37 |
University of Karachi | Assay Description β-Glucuronidase inhibitory activity was evaluated by a biochemical assay, based on the measurement of the absorbance of p-nitrophenol at 405 nm,... | J Enzyme Inhib Med Chem 27: 348-55 (2012) Article DOI: 10.3109/14756366.2011.590804 BindingDB Entry DOI: 10.7270/Q2N29VV5 | |||||||||||
More data for this Ligand-Target Pair |