Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Leucine--tRNA ligase (Mycobacterium tuberculosis (strain ATCC 25618 / H3...) | BDBM50241779 (CHEMBL4082159) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 216 | n/a | n/a | n/a | n/a | n/a | n/a |
Russian Academy of Science Curated by ChEMBL | Assay Description Inhibition of Mycobacterium tuberculosis LeuRS expressed in Escherichia coli Rosetta (DE3) cells | J Med Chem 63: 8917-8955 (2020) Article DOI: 10.1021/acs.jmedchem.9b02075 BindingDB Entry DOI: 10.7270/Q21Z480D | |||||||||||
More data for this Ligand-Target Pair |