Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
ATP-dependent Clp protease ATP-binding subunit ClpC1 (Mycobacterium tuberculosis) | BDBM50540273 (CHEMBL4637575) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 620 | n/a | n/a | n/a | n/a | n/a |
University of Illinois at Chicago Curated by ChEMBL | Assay Description Binding affinity to recombinant Mycobacterium tuberculosis H37Rv N-terminal His6-tagged ClpC1 (1 to 145 residues) expressed in Escherichia coli BL21 ... | J Nat Prod 83: 657-667 (2020) Article DOI: 10.1021/acs.jnatprod.9b01095 BindingDB Entry DOI: 10.7270/Q2959N3R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATP-dependent Clp protease ATP-binding subunit ClpC1 (Mycobacterium tuberculosis) | BDBM50540283 (CHEMBL4643756) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 1.50E+3 | n/a | n/a | n/a | n/a | n/a |
University of Illinois at Chicago Curated by ChEMBL | Assay Description Binding affinity to recombinant full length Mycobacterium tuberculosis H37Rv ClpC1 (1 to 842 residues) expressed in Escherichia coli BL21 cells by su... | J Nat Prod 83: 657-667 (2020) Article DOI: 10.1021/acs.jnatprod.9b01095 BindingDB Entry DOI: 10.7270/Q2959N3R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATP-dependent Clp protease ATP-binding subunit ClpC1 (Mycobacterium tuberculosis) | BDBM50540275 (CHEMBL4649631) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 1.10E+3 | n/a | n/a | n/a | n/a | n/a |
University of Illinois at Chicago Curated by ChEMBL | Assay Description Binding affinity to recombinant Mycobacterium tuberculosis H37Rv N-terminal His6-tagged ClpC1 (1 to 145 residues) expressed in Escherichia coli BL21 ... | J Nat Prod 83: 657-667 (2020) Article DOI: 10.1021/acs.jnatprod.9b01095 BindingDB Entry DOI: 10.7270/Q2959N3R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATP-dependent Clp protease ATP-binding subunit ClpC1 (Mycobacterium tuberculosis) | BDBM50540276 (CHEMBL4643598) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 1.20E+3 | n/a | n/a | n/a | n/a | n/a |
University of Illinois at Chicago Curated by ChEMBL | Assay Description Binding affinity to recombinant Mycobacterium tuberculosis H37Rv N-terminal His6-tagged ClpC1 (1 to 145 residues) expressed in Escherichia coli BL21 ... | J Nat Prod 83: 657-667 (2020) Article DOI: 10.1021/acs.jnatprod.9b01095 BindingDB Entry DOI: 10.7270/Q2959N3R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATP-dependent Clp protease ATP-binding subunit ClpC1 (Mycobacterium tuberculosis) | BDBM50540277 (CHEMBL4649342) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 310 | n/a | n/a | n/a | n/a | n/a |
University of Illinois at Chicago Curated by ChEMBL | Assay Description Binding affinity to recombinant Mycobacterium tuberculosis H37Rv N-terminal His6-tagged ClpC1 (1 to 145 residues) expressed in Escherichia coli BL21 ... | J Nat Prod 83: 657-667 (2020) Article DOI: 10.1021/acs.jnatprod.9b01095 BindingDB Entry DOI: 10.7270/Q2959N3R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATP-dependent Clp protease ATP-binding subunit ClpC1 (Mycobacterium tuberculosis) | BDBM50540278 (CHEMBL4647204) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 300 | n/a | n/a | n/a | n/a | n/a |
University of Illinois at Chicago Curated by ChEMBL | Assay Description Binding affinity to recombinant Mycobacterium tuberculosis H37Rv N-terminal His6-tagged ClpC1 (1 to 145 residues) expressed in Escherichia coli BL21 ... | J Nat Prod 83: 657-667 (2020) Article DOI: 10.1021/acs.jnatprod.9b01095 BindingDB Entry DOI: 10.7270/Q2959N3R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATP-dependent Clp protease ATP-binding subunit ClpC1 (Mycobacterium tuberculosis) | BDBM50540279 (CHEMBL4637113) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 60 | n/a | n/a | n/a | n/a | n/a |
University of Illinois at Chicago Curated by ChEMBL | Assay Description Binding affinity to recombinant Mycobacterium tuberculosis H37Rv N-terminal His6-tagged ClpC1 (1 to 145 residues) expressed in Escherichia coli BL21 ... | J Nat Prod 83: 657-667 (2020) Article DOI: 10.1021/acs.jnatprod.9b01095 BindingDB Entry DOI: 10.7270/Q2959N3R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATP-dependent Clp protease ATP-binding subunit ClpC1 (Mycobacterium tuberculosis) | BDBM50540280 (CHEMBL4648320) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 1.70E+3 | n/a | n/a | n/a | n/a | n/a |
University of Illinois at Chicago Curated by ChEMBL | Assay Description Binding affinity to recombinant Mycobacterium tuberculosis H37Rv N-terminal His6-tagged ClpC1 (1 to 145 residues) expressed in Escherichia coli BL21 ... | J Nat Prod 83: 657-667 (2020) Article DOI: 10.1021/acs.jnatprod.9b01095 BindingDB Entry DOI: 10.7270/Q2959N3R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATP-dependent Clp protease ATP-binding subunit ClpC1 (Mycobacterium tuberculosis) | BDBM50540281 (CHEMBL4642233) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 1.20E+3 | n/a | n/a | n/a | n/a | n/a |
University of Illinois at Chicago Curated by ChEMBL | Assay Description Binding affinity to recombinant Mycobacterium tuberculosis H37Rv N-terminal His6-tagged ClpC1 (1 to 145 residues) expressed in Escherichia coli BL21 ... | J Nat Prod 83: 657-667 (2020) Article DOI: 10.1021/acs.jnatprod.9b01095 BindingDB Entry DOI: 10.7270/Q2959N3R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATP-dependent Clp protease ATP-binding subunit ClpC1 (Mycobacterium tuberculosis) | BDBM50540282 (CHEMBL4638710) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 60 | n/a | n/a | n/a | n/a | n/a |
University of Illinois at Chicago Curated by ChEMBL | Assay Description Binding affinity to recombinant Mycobacterium tuberculosis H37Rv N-terminal His6-tagged ClpC1 (1 to 145 residues) expressed in Escherichia coli BL21 ... | J Nat Prod 83: 657-667 (2020) Article DOI: 10.1021/acs.jnatprod.9b01095 BindingDB Entry DOI: 10.7270/Q2959N3R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATP-dependent Clp protease ATP-binding subunit ClpC1 (Mycobacterium tuberculosis) | BDBM50540283 (CHEMBL4643756) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 1.50E+3 | n/a | n/a | n/a | n/a | n/a |
University of Illinois at Chicago Curated by ChEMBL | Assay Description Binding affinity to recombinant Mycobacterium tuberculosis H37Rv N-terminal His6-tagged ClpC1 (1 to 145 residues) expressed in Escherichia coli BL21 ... | J Nat Prod 83: 657-667 (2020) Article DOI: 10.1021/acs.jnatprod.9b01095 BindingDB Entry DOI: 10.7270/Q2959N3R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATP-dependent Clp protease ATP-binding subunit ClpC1 (Mycobacterium tuberculosis) | BDBM50540273 (CHEMBL4637575) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 500 | n/a | n/a | n/a | n/a | n/a |
University of Illinois at Chicago Curated by ChEMBL | Assay Description Binding affinity to recombinant full length Mycobacterium tuberculosis H37Rv ClpC1 (1 to 842 residues) expressed in Escherichia coli BL21 cells by su... | J Nat Prod 83: 657-667 (2020) Article DOI: 10.1021/acs.jnatprod.9b01095 BindingDB Entry DOI: 10.7270/Q2959N3R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATP-dependent Clp protease ATP-binding subunit ClpC1 (Mycobacterium tuberculosis) | BDBM50540274 (CHEMBL4641855) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 1.30E+3 | n/a | n/a | n/a | n/a | n/a |
University of Illinois at Chicago Curated by ChEMBL | Assay Description Binding affinity to recombinant full length Mycobacterium tuberculosis H37Rv ClpC1 (1 to 842 residues) expressed in Escherichia coli BL21 cells by su... | J Nat Prod 83: 657-667 (2020) Article DOI: 10.1021/acs.jnatprod.9b01095 BindingDB Entry DOI: 10.7270/Q2959N3R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATP-dependent Clp protease ATP-binding subunit ClpC1 (Mycobacterium tuberculosis) | BDBM50540275 (CHEMBL4649631) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 1.10E+3 | n/a | n/a | n/a | n/a | n/a |
University of Illinois at Chicago Curated by ChEMBL | Assay Description Binding affinity to recombinant full length Mycobacterium tuberculosis H37Rv ClpC1 (1 to 842 residues) expressed in Escherichia coli BL21 cells by su... | J Nat Prod 83: 657-667 (2020) Article DOI: 10.1021/acs.jnatprod.9b01095 BindingDB Entry DOI: 10.7270/Q2959N3R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATP-dependent Clp protease ATP-binding subunit ClpC1 (Mycobacterium tuberculosis) | BDBM50540276 (CHEMBL4643598) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 5.70E+3 | n/a | n/a | n/a | n/a | n/a |
University of Illinois at Chicago Curated by ChEMBL | Assay Description Binding affinity to recombinant full length Mycobacterium tuberculosis H37Rv ClpC1 (1 to 842 residues) expressed in Escherichia coli BL21 cells by su... | J Nat Prod 83: 657-667 (2020) Article DOI: 10.1021/acs.jnatprod.9b01095 BindingDB Entry DOI: 10.7270/Q2959N3R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATP-dependent Clp protease ATP-binding subunit ClpC1 (Mycobacterium tuberculosis) | BDBM50540277 (CHEMBL4649342) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 450 | n/a | n/a | n/a | n/a | n/a |
University of Illinois at Chicago Curated by ChEMBL | Assay Description Binding affinity to recombinant full length Mycobacterium tuberculosis H37Rv ClpC1 (1 to 842 residues) expressed in Escherichia coli BL21 cells by su... | J Nat Prod 83: 657-667 (2020) Article DOI: 10.1021/acs.jnatprod.9b01095 BindingDB Entry DOI: 10.7270/Q2959N3R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATP-dependent Clp protease ATP-binding subunit ClpC1 (Mycobacterium tuberculosis) | BDBM50540284 (CHEMBL4636448) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 1.50E+3 | n/a | n/a | n/a | n/a | n/a |
University of Illinois at Chicago Curated by ChEMBL | Assay Description Binding affinity to recombinant full length Mycobacterium tuberculosis H37Rv ClpC1 (1 to 842 residues) expressed in Escherichia coli BL21 cells by su... | J Nat Prod 83: 657-667 (2020) Article DOI: 10.1021/acs.jnatprod.9b01095 BindingDB Entry DOI: 10.7270/Q2959N3R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATP-dependent Clp protease ATP-binding subunit ClpC1 (Mycobacterium tuberculosis) | BDBM50540278 (CHEMBL4647204) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 280 | n/a | n/a | n/a | n/a | n/a |
University of Illinois at Chicago Curated by ChEMBL | Assay Description Binding affinity to recombinant full length Mycobacterium tuberculosis H37Rv ClpC1 (1 to 842 residues) expressed in Escherichia coli BL21 cells by su... | J Nat Prod 83: 657-667 (2020) Article DOI: 10.1021/acs.jnatprod.9b01095 BindingDB Entry DOI: 10.7270/Q2959N3R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATP-dependent Clp protease ATP-binding subunit ClpC1 (Mycobacterium tuberculosis) | BDBM50540279 (CHEMBL4637113) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 50 | n/a | n/a | n/a | n/a | n/a |
University of Illinois at Chicago Curated by ChEMBL | Assay Description Binding affinity to recombinant full length Mycobacterium tuberculosis H37Rv ClpC1 (1 to 842 residues) expressed in Escherichia coli BL21 cells by su... | J Nat Prod 83: 657-667 (2020) Article DOI: 10.1021/acs.jnatprod.9b01095 BindingDB Entry DOI: 10.7270/Q2959N3R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATP-dependent Clp protease ATP-binding subunit ClpC1 (Mycobacterium tuberculosis) | BDBM50540280 (CHEMBL4648320) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 540 | n/a | n/a | n/a | n/a | n/a |
University of Illinois at Chicago Curated by ChEMBL | Assay Description Binding affinity to recombinant full length Mycobacterium tuberculosis H37Rv ClpC1 (1 to 842 residues) expressed in Escherichia coli BL21 cells by su... | J Nat Prod 83: 657-667 (2020) Article DOI: 10.1021/acs.jnatprod.9b01095 BindingDB Entry DOI: 10.7270/Q2959N3R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATP-dependent Clp protease ATP-binding subunit ClpC1 (Mycobacterium tuberculosis) | BDBM50540281 (CHEMBL4642233) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 3.20E+3 | n/a | n/a | n/a | n/a | n/a |
University of Illinois at Chicago Curated by ChEMBL | Assay Description Binding affinity to recombinant full length Mycobacterium tuberculosis H37Rv ClpC1 (1 to 842 residues) expressed in Escherichia coli BL21 cells by su... | J Nat Prod 83: 657-667 (2020) Article DOI: 10.1021/acs.jnatprod.9b01095 BindingDB Entry DOI: 10.7270/Q2959N3R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATP-dependent Clp protease ATP-binding subunit ClpC1 (Mycobacterium tuberculosis) | BDBM50540282 (CHEMBL4638710) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 60 | n/a | n/a | n/a | n/a | n/a |
University of Illinois at Chicago Curated by ChEMBL | Assay Description Binding affinity to recombinant full length Mycobacterium tuberculosis H37Rv ClpC1 (1 to 842 residues) expressed in Escherichia coli BL21 cells by su... | J Nat Prod 83: 657-667 (2020) Article DOI: 10.1021/acs.jnatprod.9b01095 BindingDB Entry DOI: 10.7270/Q2959N3R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATP-dependent Clp protease ATP-binding subunit ClpC1 (Mycobacterium tuberculosis) | BDBM50540274 (CHEMBL4641855) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 1.60E+3 | n/a | n/a | n/a | n/a | n/a |
University of Illinois at Chicago Curated by ChEMBL | Assay Description Binding affinity to recombinant Mycobacterium tuberculosis H37Rv N-terminal His6-tagged ClpC1 (1 to 145 residues) expressed in Escherichia coli BL21 ... | J Nat Prod 83: 657-667 (2020) Article DOI: 10.1021/acs.jnatprod.9b01095 BindingDB Entry DOI: 10.7270/Q2959N3R | |||||||||||
More data for this Ligand-Target Pair |